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SaveWithaferin A, a natural thioredoxin reductase 1 (TrxR1) inhibitor, synergistically enhances the antitumor efficacy of sorafenib through ROS-mediated ER stress and DNA damage in hepatocellular carcinoma cells
Chen, Xi; Zhu, Ning; Wu, Yajie; Zhang, Ye; Zhang, Yuxuan; Jin, Kaiwen; Zhou, Zhiyi; Chen, Guang; Wang, Jiabing
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SavePhase 1 study of BPI-23314, a novel BET inhibitor and degrader, in advanced myeloid leukemia (AML)
Sun, Mingyuan; Jin, Xiangyu; Guo, Jing; Liu, Xiaoyun; Xu, Yan; Lan, Hong; Wang, Jiabing; Zhen, Jiangnan; Yang, Jing; Ding, Lieming; Qi, Junyuan
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SaveBPI-501836: A highly potent small molecule inhibitor targeting KRASG12D mutation
Yang, Xiang; Lu, Yuan; Xu, Renqi; Kong, Xiaoqiang; Sun, Yongqing; Zhu, Xingjie; Liu, Xiaoyun; Zou, Zhengyao; Chen, Haibo; Liu, Yanju; Sun, Jialing; Han, Han; Yang, Cheng; Guo, Jing; Lan, Hong; Zhou, Quan; Ding, Lieming; Wu, Hao; Wang, Jiabing
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SaveDiscovery of a potent small molecule MALT1 protease inhibitor for the treatment of cancer
Zhou, Yuzhen; Fu, Bang; Chen, Jie; Cai, Weidong; Sun, Xiao; Li, Yinlong; Ren, Wei; Shen, Qichao; Du, Guolong; Zhou, Xiaojun; Zou, Zhengyao; Chen, Haibo; Liu, Xiaoyun; Yang, Cheng; Liu, Xiangyong; Guo, Jing; Wu, Hao; Ding, Lieming; Wang, Jiabing; Lan, Hong
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SaveBPI-511966,a potent and selective HPK1 inhibitor with robust single-agent efficacy for cancer immunotherapy
Zhang, Yong; Zhu, Xiaoguan; Wu, Wenmao; Xia, Zhifang; Zou, Zhengyao; Han, Han; Yang, Cheng; Chen, Haibo; Ma, Tianyi; Liu, Xiaoyun; Guo, Jing; Wu, Hao; Lan, Hong; Ding, Lieming; Wang, Jiabing; Zhou, Quan
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SaveBPI-520105, a highly potent, CNS- penetrant 4th generation EGFR inhibitor overcoming major EGFR resistance mutations in NSCLC
Guo, Jing; Liu, Lijia; Liu, Xiangyong; Fu, Bang; Bai, Guangcan; Qiu, Changyong; Ren, Wei; Song, Xiaodong; Du, Guolong; Sun, Xiao; Zhang, Yongchun; Cai, Weidong; Wang, Pingping; Chen, Haibo; Liu, Xiaoyun; Zou, Zhengyao; Zhao, Jiayu; Jv, Xuepeng; Lan, Hong; Ding, Lieming; Wang, Jiabing
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SaveBPI-472372: a potent and orally bioavailable small molecule inhibitor of CD73 for cancer immunotherapy
Han, Han; Yang, Xiaofeng; Zhao, Ying; Wang, Jin; Yang, Xiang; Ju, Xuepeng; Zhao, Jiayu; Zou, Zhengyao; Chen, Haibo; Liu, Xiaoyun; Guo, Jing; Yang, Cheng; Lan, Hong; Wu, Hao; Ding, Lieming; Wang, Jiabing
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SaveDesign, synthesis and biological evaluation of chalcone analogues with novel dual antioxidant mechanisms as potential anti-ischemic stroke agents (vol 9, pg 335, 2019)
Wang, Jiabing; Huang, Lili; Chen, Chanchan; Li, Ge; Xie, Jingwen; Shen, Mengya; Chen, Qian; Li, Wulan; He, Wenfei; Qiu, Peihong; Wu, Jianzhang
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