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Stuart L. Schreiber

MIT and Harvard

166H-index
1.3KPaper Count
13.3WCitation Count
Published Papers 370
Publication Date
Discovery of molecular glues that bind FKBP12 and structurally distinct targets using DNA-encoded libraries
err2026-04-22
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errOAAI
errTrevor A. Zandi; Michael J. Romanowski; Jessica S. Viscomi; Karl Gunderson; Zher Yin Tan; Bingqi Tong; Simone Bonazzi; Frédéric J. Zécri; Stuart L. Schreiber; Gregory A. Michaud
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Author Correction: Diversity-oriented synthesis yields novel multistage antimalarial inhibitors
errNature
IF48.5
err2025-11-28
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PREAI
errNobutaka Kato; Eamon Comer; Tomoyo Sakata-Kato; Arvind Sharma; Manmohan Sharma; Micah Maetani; Jessica Bastien; Nicolas M. Brancucci; Joshua A. Bittker; Victoria Corey; David Clarke; Emily R. Derbyshire; Gillian L. Dornan; Sandra Duffy; Sean Eckley; Maurice A. Itoe; Karin M. J. Koolen; Timothy A. Lewis; Ping S. Lui; Amanda K. Lukens; Emily Lund; Sandra March; Elamaran Meibalan; Bennett C. Meier; Jacob A. McPhail; Branko Mitasev; Eli L. Moss; Morgane Sayes; Yvonne Van Gessel; Mathias J. Wawer; Takashi Yoshinaga; Anne-Marie Zeeman; Vicky M. Avery; Sangeeta N. Bhatia; John E. Burke; Flaminia Catteruccia; Jon C. Clardy; Paul A. Clemons; Koen J. Dechering; Jeremy R. Duvall; Michael A. Foley; Fabian Gusovsky; Clemens H. M. Kocken; Matthias Marti; Marshall L. Morningstar; Benito Munoz; Daniel E. Neafsey; Amit Sharma; Elizabeth A. Winzeler; Dyann F. Wirth; Christina A. Scherer; Stuart L. Schreiber
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Publisher Correction: Mutant p53 protein accumulation is selectively targetable by proximity-inducing drugs
err2025-11-12
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errOAAI
errAnanthan Sadagopan; Maximilian Carson; Eriks J. Zamurs; Nicholas Garaffo; Heng-Jui Chang; Stuart L. Schreiber; Matthew Meyerson; William J. Gibson
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Mutant p53 protein accumulation is selectively targetable by proximity-inducing drugs
err2025-11-03
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errOAAI
errAnanthan Sadagopan; Maximilian Carson; Eriks J. Zamurs; Nicholas Garaffo; Heng-Jui Chang; Stuart L. Schreiber; Matthew Meyerson; William J. Gibson
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The Ulcerative Colitis-Associated Gene NXPE1 Catalyzes Glycan Modifications on Colonic Mucin
err2025-03-11
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errOAAI
errHumeidi, Ranad; Oshiro-Rapley, Noriko; Gu, Xiebin; An, Joon Soo; Ananthakrishnan, Ashwin N.; Creasey, Elizabeth A.; Daly, Mark J.; Schreiber, Stuart L.; Graham, Daniel B.; Seyedsayamdost, Mohammad R.; Xavier, Ramnik J.
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Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes
err2024-12-01
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errOAAI
errOgasawara, Daisuke; Konrad, David B.; Tan, Zher Yin; Carey, Kimberly L.; Luo, Jessica; Won, Sang Joon; Li, Haoxin; Carter, Trever R.; DeMeester, Kristen E.; Njomen, Evert; Schreiber, Stuart L.; Xavier, Ramnik J.; Melillo, Bruno; Cravatt, Benjamin F.
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Bicyclic Pyrrolidine Inhibitors of Toxoplasma gondii Phenylalanine t-RNA Synthetase with Antiparasitic Potency In Vitro and Brain Exposure
err2024-05-14
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PREAI
errEnce, Chloe C.; Uddin, Taher; Borrel, Julien; Mittal, Payal; Xie, Han; Zoller, Jochen; Sharma, Amit; Comer, Eamon; Schreiber, Stuart L.; Melillo, Bruno; Sibley, L. David; Chatterjee, Arnab K.
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Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders
err2024-04-03
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PREAI
errLiu, Zhonglin; Remsberg, Jarrett R.; Li, Haoxin; Njomen, Evert; Demeester, Kristen E.; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E.; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M.; Schreiber, Stuart L.; Melillo, Bruno; Cravatt, Benjamin F.
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Bifunctional Small Molecules That Induce Nuclear Localization and Targeted Transcriptional Regulation
err2023-11-22
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errOAAI
errGibson, William J.; Sadagopan, Ananthan; Shoba, Veronika M.; Choudhary, Amit; Meyerson, Matthew; Schreiber, Stuart L.
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Diversity-oriented synthesis encoded by deoxyoligonucleotides (vol 14, 4930, 2023)
err2023-11-21
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errHudson, Liam; Mason, Jeremy W.; Westphal, Matthias V.; Richter, Matthieu J. R.; Thielman, Jonathan R.; Hua, Bruce K.; Gerry, Christopher J.; Xia, Guoqin; Osswald, Heather L.; Knapp, John M.; Tan, Zher Yin; Kokkonda, Praveen; Tresco, Ben I. C.; Liu, Shuang; Reidenbach, Andrew G.; Lim, Katherine S.; Poirier, Jennifer; Capece, John; Bonazzi, Simone; Gampe, Christian M.; Smith, Nichola J.; Bradner, James E.; Coley, Connor W.; Clemons, Paul A.; Melillo, Bruno; Hon, C. Suk-Yee; Ottl, Johannes; Dumelin, Christoph E.; Schaefer, Jonas V.; Faust, Ann Marie E.; Berst, Frederic; Schreiber, Stuart L.; Zecri, Frederic J.; Briner, Karin
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DNA-encoded library-enabled discovery of proximity-inducing small molecules
err2023-11-02
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errOAAI
errMason, Jeremy W.; Chow, Yuen Ting; Hudson, Liam; Tutter, Antonin; Michaud, Gregory; Westphal, Matthias V.; Shu, Wei; Ma, Xiaolei; Tan, Zher Yin; Coley, Connor W.; Clemons, Paul A.; Bonazzi, Simone; Berst, Frederic; Briner, Karin; Liu, Shuang; Zecri, Frederic J.; Schreiber, Stuart L.
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Rational Screening for Cooperativity in Small-Molecule Inducers of Protein-Protein Associations
err2023-10-10
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errOAAI
errLiu, Shuang; Tong, Bingqi; Mason, Jeremy W.; Ostrem, Jonathan M.; Tutter, Antonin; Hua, Bruce K.; Tang, Sunny A.; Bonazzi, Simone; Briner, Karin; Berst, Frederic; Zecri, Frederic J.; Schreiber, Stuart L.
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Diversity-oriented synthesis encoded by deoxyoligonucleotides
err2023-08-15
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errOAAI
errHudson, Liam; Mason, Jeremy W.; Westphal, Matthias V.; Richter, Matthieu J. R.; Thielman, Jonathan R.; Hua, Bruce K.; Gerry, Christopher J.; Xia, Guoqin; Osswald, Heather L.; Knapp, John M.; Tan, Zher Yin; Kokkonda, Praveen; Tresco, Ben I. C.; Liu, Shuang; Reidenbach, Andrew G.; Lim, Katherine S.; Poirier, Jennifer; Capece, John; Bonazzi, Simone; Gampe, Christian M.; Smith, Nichola J.; Bradner, James E.; Coley, Connor W.; Clemons, Paul A.; Melillo, Bruno; Hon, C. Suk-Yee; Ottl, Johannes; Dumelin, Christoph E.; Schaefer, Jonas V.; Faust, Ann Marie E.; Berst, Frederic; Schreiber, Stuart L.; Zecri, Frederic J.; Briner, Karin
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Targeted Protein Degradation by Electrophilic PROTACs that Stereoselectively and Site-Specifically Engage DCAF1 (vol 144, pg 18688, 2022)
err2023-06-02
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PREAI
errTao, Yongfeng; Remillard, David; Vinogradova, Ekaterina V. V.; Yokoyama, Minoru; Banchenko, Sofia; Schwefel, David; Melillo, Bruno; Schreiber, Stuart L. L.; Zhang, Xiaoyu; Cravatt, Benjamin F. F.
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Proteomic discovery of chemical probes that perturb protein complexes in human cells
err2023-05-01
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errOAAI
errLazear, Michael R.; Remsberg, Jarrett R.; Jaeger, Martin G.; Rothamel, Katherine; Her, Hsuan-lin; DeMeester, Kristen E.; Njomen, Evert; Hogg, Simon J.; Rahman, Jahan; Whitby, Landon R.; Won, Sang Joon; Schafroth, Michael A.; Ogasawara, Daisuke; Yokoyama, Minoru; Lindsey, Garrett L.; Li, Haoxin; Germain, Jason; Barbas, Sabrina; Vaughan, Joan; Hanigan, Thomas W.; Vartabedian, Vincent F.; Reinhardt, Christopher J.; Dix, Melissa M.; Koo, Seong Joo; Heo, Inha; Teijaro, John R.; Simon, Gabriel M.; Ghosh, Brahma; Abdel-Wahab, Omar; Ahn, Kay; Saghatelian, Alan; Melillo, Bruno; Schreiber, Stuart L.; Yeo, Gene W.; Cravatt, Benjamin F.
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Mapping the landscape of genetic dependencies in chordoma
err2023-04-06
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errOAAI
errSharifnia, Tanaz; Wawer, Mathias J.; Goodale, Amy; Lee, Yenarae; Kazachkova, Mariya; Dempster, Joshua M.; Muller, Sandrine; Levy, Joan; Freed, Daniel M.; Sommer, Josh; Kalfon, Jeremie; Vazquez, Francisca; Hahn, William C.; Root, David E.; Clemons, Paul A.; Schreiber, Stuart L.
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ROS Induction Targets Persister Cancer Cells with Low Metabolic Activity in NRAS-Mutated Melanoma
err2023-03-22
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errOAAI
errEichhoff, Ossia M.; Stoffel, Corinne I.; Kasler, Jan; Briker, Luzia; Turko, Patrick; Karsai, Gergely; Zila, Nina; Paulitschke, Verena; Cheng, Phil F.; Leitner, Alexander; Bileck, Andrea; Zamboni, Nicola; Irmisch, Anja; Balazs, Zsolt; Tastanova, Aizhan; Pascoal, Susana; Johansen, Pal; Wegmann, Rebekka; Mena, Julien; Othman, Alaa; Viswanathan, Vasanthi S.; Wenzina, Judith; Aloia, Andrea; Saltari, Annalisa; Dzung, Andreas; Krauthammer, Michael; Schreiber, Stuart L.; Hornemann, Thorsten; Distel, Martin; Snijder, Berend; Dummer, Reinhard; Levesque, Mitchell P.
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Reference compounds for characterizing cellular injury in high-content cellular morphology assays
err2023-03-13
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errOAAI
errDahlin, Jayme L.; Hua, Bruce K.; Zucconi, Beth E.; Nelson, Shawn D.; Singh, Shantanu; Carpenter, Anne E.; Shrimp, Jonathan H.; Lima-Fernandes, Evelyne; Wawer, Mathias J.; Chung, Lawrence P. W.; Agrawal, Ayushi; O'Reilly, Mary; Barsyte-Lovejoy, Dalia; Szewczyk, Magdalena; Li, Fengling; Lak, Parnian; Cuellar, Matthew; Cole, Philip A.; Meier, Jordan L.; Thomas, Tim; Baell, Jonathan B.; Brown, Peter J.; Walters, Michael A.; Clemons, Paul A.; Schreiber, Stuart L.; Wagner, Bridget K.
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