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SaveAPR-246 increases tumor antigenicity independent of p53
Michels, Judith; Venkatesh, Divya; Liu, Cailian; Budhu, Sadna; Zhong, Hong; George, Mariam M.; Thach, Daniel; Yao, Zhong-Ke; Ouerfelli, Ouathek; Liu, Hengrui; Stockwell, Brent R.; Campesato, Luis Felipe; Zamarin, Dmitriy; Zappasodi, Roberta; Wolchok, Jedd D.; Merghoub, Taha
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SaveDevelopment of optimized drug-like small molecule inhibitors of the SARS-CoV-2 3CL protease for treatment of COVID-19
Liu, Hengrui; Iketani, Sho; Zask, Arie; Khanizeman, Nisha; Bednarova, Eva; Forouhar, Farhad; Fowler, Brandon; Hong, Seo Jung; Mohri, Hiroshi; Nair, Manoj S.; Huang, Yaoxing; Tay, Nicholas E. S.; Lee, Sumin; Karan, Charles; Resnick, Samuel J.; Quinn, Colette; Li, Wenjing; Shion, Henry; Xia, Xin; Daniels, Jacob D.; Bartolo-Cruz, Michelle; Farina, Marcelo; Rajbhandari, Presha; Jurtschenko, Christopher; Lauber, Matthew A.; McDonald, Thomas; Stokes, Michael E.; Hurst, Brett L.; Rovis, Tomislav; Chavez, Alejandro; Ho, David D.; Stockwell, Brent R.
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SaveCharacterization of a patient-derived variant of GPX4 for precision therapy
Liu, Hengrui; Forouhar, Farhad; Seibt, Tobias; Saneto, Russell; Wigby, Kristen; Friedman, Jennifer; Xia, Xin; Shchepinov, Mikhail S.; Ramesh, Sanath Kumar; Conrad, Marcus; Stockwell, Brent R.
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SaveInhibitors of Coronavirus 3CL Proteases Protect Cells from Protease-Mediated Cytotoxicity
Resnick, Samuel J.; Iketani, Sho; Hong, Seo Jung; Zask, Arie; Liu, Hengrui; Kim, Sungsoo; Melore, Schuyler; Lin, Fang-Yu; Nair, Manoj S.; Huang, Yaoxing; Lee, Sumin; Tay, Nicholas E. S.; Rovis, Tomislav; Yang, Hee Won; Xing, Li; Stockwell, Brent R.; Ho, David D.; Chavez, Alejandro
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SaveLead compounds for the development of SARS-CoV-2 3CL protease inhibitors (vol 12, 2016, 2021)
Iketani, Sho; Forouhar, Farhad; Liu, Hengrui; Hong, Seo Jung; Lin, Fang-Yu; Nair, Manoj S.; Zask, Arie; Huang, Yaoxing; Xing, Li; Stockwell, Brent R.; Chavez, Alejandro; Ho, David D.
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SaveLead compounds for the development of SARS-CoV-2 3CL protease inhibitors
Iketani, Sho; Forouhar, Farhad; Liu, Hengrui; Hong, Seo Jung; Lin, Fang-Yu; Nair, Manoj S.; Zask, Arie; Huang, Yaoxing; Xing, Li; Stockwell, Brent R.; Chavez, Alejandro; Ho, David D.
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SaveFINO2 initiates ferroptosis through GPX4 inactivation and iron oxidation
Gaschler, Michael M.; Andia, Alexander A.; Liu, Hengrui; Csuka, Joleen M.; Hurlocker, Brisa; Vaiana, Christopher A.; Heindel, Daniel W.; Zuckerman, Dylan S.; Bos, Pieter H.; Reznik, Eduard; Ye, Ling F.; Tyurina, Yulia Y.; Lin, Annie J.; Shchepinov, Mikhail S.; Chan, Amy Y.; Peguero-Pereira, Eveliz; Fomich, Maksim A.; Daniels, Jacob. D.; Bekish, Andrei V.; Shmanai, Vadim V.; Kagan, Valerian E.; Mahal, Lara K.; Woerpel, K. A.; Stockwell, Brent R.
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