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Repurposing disulfiram, an alcohol-abuse drug, in neuroblastoma causes KAT2A downregulation and in vivo activity with a water/oil emulsion Beaudry, Annie; Jacques-Ricard, Simon; Darracq, Anais; Sgarioto, Nicolas; Garcia, Araceli; Garcia, Teresita Rode; Lemieux, William; Beland, Kathie; Haddad, Elie; Cordeiro, Paulo; Duval, Michel; Mcgraw, Serge; Richer, Chantal; Caron, Maxime; Marois, Francois; St-Onge, Pascal; Sinnett, Daniel; Banquy, Xavier; Raynal, Noel J. -M. Share Save
The Lipid Metabolism as Target and Modulator of BOLD-100 Anticancer Activity: Crosstalk with Histone Acetylation Baier, Dina; Mendrina, Theresa; Schoenhacker-Alte, Beatrix; Pirker, Christine; Mohr, Thomas; Rusz, Mate; Regner, Benedict; Schaier, Martin; Sgarioto, Nicolas; Raynal, Noel J. -M.; Nowikovsky, Karin; Schmidt, Wolfgang M.; Heffeter, Petra; Meier-Menches, Samuel M.; Koellensperger, Gunda; Keppler, Bernhard K.; Berger, Walter Share Save
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TACIMA-218: A Novel Pro-Oxidant Agent Exhibiting Selective Antitumoral Activity Abusarah, Jamilah; Cui, Yun; El-Hachem, Nehme; El-Kadiry, Abed El-Hakim; Hammond-Martel, Ian; Wurtele, Hugo; Beaudry, Annie; Raynal, Noel J-M; Robert, Francis; Pelletier, Jerry; Jankovic, Maja; Mercier, Francois; Kamyabiazar, Samaneh; Annabi, Borhane; Rafei, Moutih Share Save
Targeting MYC overexpressing leukemia with cardiac glycoside proscillaridin through downregulation of histone acetyltransferases Da Costa, Elodie Marie; Armaos, Gregory; McInnes, Gabrielle; Beaudry, Annie; Moquin-Beaudry, Gael; Bertrand-Lehouillier, Virginie; Caron, Maxime; St-Onge, Pascal; Jonhson, Jeffrey R.; Krogan, Nevan; Sai, Yuka; Downey, Michale; Rafei, Moutih; Boileau, Meaghan; Eppert, Kolja; Florez-Diaz, Ema; Haman, Andre; Trang Hoang; Sinnett, Daniel; Beausejour, Christian; McGraw, Serge; Raynal, Noel J. Share Save
Heart failure drug proscillaridin A targets MYC overexpressing leukemia through global loss of lysine acetylation Da Costa, Elodie M.; Armaos, Gregory; McInnes, Gabrielle; Beaudry, Annie; Moquin-Beaudry, Gael; Bertrand-Lehouillier, Virginie; Caron, Maxime; Richer, Chantal; St-Onge, Pascal; Johnson, Jeffrey R.; Krogan, Nevan; Sai, Yuka; Downey, Michael; Rafei, Moutih; Boileau, Meaghan; Eppert, Kolja; Flores-Diaz, Ema; Haman, Andre; Hoang, Trang; Sinnett, Daniel; Beausejour, Christian; McGraw, Serge; Raynal, Noel J. -M. Share Save
Targeting histone acetyltransferases to reprogram high C-MYC expressing cancers Da Costa, Elodie M.; Armaos, Gregory; Beaudry, Annie; Richer, Chantal; Caron, Maxime; St-Onge, Pascal; Johnson, Jeffrey; Krogan, Nevan; Sai, Yuka; Downey, Michael; Sinnett, Daniel; McGraw, Serge; Raynal, Noel J. Share Save
Targeting CDK9 reactivates epigenetically silenced genes in cancer Zhang, Hanghang; Pandey, Somnath; Travers, Meghan; Khowsathit, Jittasak; Morton, George; Sum, Hongxing; Barrero, Carlos A.; Merali, Carmen; Okamoto, Yasuyuki; Sato, Takahiro; Garriga, Judit; Bhanu, Natarajan V.; Simithy, Johayra; Patel, Bela; Madzo, Jozef; Raynal, Noel; Garcia, Benjamin A.; Jacobson, Marlene A.; Merali, Salim; Zhang, Yi; Childers, Wayne; Abou-Gharbia, Magid; Karanicolas, John; Baylin, Stephen B.; Zahnow, Cynthia A.; Jelinek, Jaroslav; Grana, Xavier; Issa, Jean-Pierre J. Share Save
Identifying novel potential epigenetic anti-cancer drugs from natural compounds using a phenotypic-based screening Zhang, Hanghang; Raynal, Noel J-M; Sato, Takahiro; Okamoto, Yasuyuki; Garriga, Judith; Garcia, Benjamin; Morton, George; Childers, Wayne; Jacobson, Marlene A.; Baylin, Stephen B.; Grana, Xavier; Abou-Gharbia, Magid; Issa, Jean-Pierre J. Share Save
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A phenotypic cell-based screen to identify novel potential epigenetic anti-cancer drugs from natural compounds Zhang, Hanghang; Raynal, Noel J. -M; Sato, Takahiro; Okamoto, Yasuyuki; Garriga, Judit; Morton, George; Childers, Wayne; Jacobson, Marlene A.; Baylin, Stephen B.; Grana, Xavier; Abou-Gharbia, Magid; Issa, Jean-Pierre J. Share Save