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J

James M. Cook

university of wisconsin─milwaukee

61H-index
869Paper Count
1.7WCitation Count
Published Papers 239
Publication Date
First Total Synthesis of the Unnatural (+)-Talcarpine and (−)-N4-Methyl; N4-21-secotalpinine
err2026-04-29
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errKamal Prasad Pandey; Md Toufiqur Rahman; Anna Benko; Gregory H. Imler; Jefferey R. Deschamps; James M. Cook
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Dual Pharmacology Strategies for a Wider Opioid Analgesic Therapeutic Window
err2025-03-01
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PREAI
errMadhuranthakam, Indu Nithra; Uribe, Sarah; Aldaghma, Danya; Afrin, Nadia; Kwitchoff, Drew T.; Philip, Jonathan; Didomenico, Eric; Conviser, Jason; Tapia, Yulitsa; Nambiar, Rohit; Ahmed, Shakil; Rahman, Mohammad A.; Donegan, Christa; Poe, Michael M.; Sharmin, Dishary; Cook, James M.; Bradford, Fischer D.; Keck, Thomas M.
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Procognitive and neurotrophic benefits of α5-GABA-A receptor positive allosteric modulation in a (3-amyloid deposition mouse model of Alzheimer's disease pathology
err2025-03-01
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errBernardo, Ashley M.; Marcotte, Michael; Wong, Kayla; Sharmin, Dishary; Pandey, Kamal P.; Cook, James M.; Sibille, Etienne L.; Prevot, Thomas D.
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Self-Administration of Benzodiazepines in Drug-Naïve and Cocaine-Experienced Rhesus Monkeys: Role of Alpha Subunit-Containing GABAA Receptors
err2025-03-01
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PREAI
errGilmore, Ihle; Piracha, Neha; Sharmin, Dishary; Mondal, Prithu; Cook, James M.; Doyle, William S.; Freeman, Kevin B.; Rowlett, James K.; Huskinson, Sally L.
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α6GABAA RECEPTOR-SELECTIVE POSITIVE ALLOSTERIC MODULATOR AS A POTENTIAL NOVEL THERAPY FOR AUTISM: A PRECLINICAL STUDY IN OFFSPRING OF VALPROIC ACID-TREATED RATS
err2025-02-12
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errPan, Yi-Ting; Wu, Chi-Chun; Chu, Ming-Chai; Yeh, Chen-Jiun; Sharmin, Dishary; Cook, James; Lin, Hui-Ching; Chiou, Lih-Chu
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Intravenous Nanoemulsions Loaded with Phospholipid Complex of a Novel Pyrazoloquinolinone Ligand for Enhanced Brain Delivery
err2025-02-11
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errStankovic, Tijana; Ilic, Tanja; Divovic Matovic, Branka; Petkovic, Milos; Dobricic, Vladimir; Jancic, Ivan; Bufan, Biljana; Jezdic, Kristina; Dokovic, Jelena; Pantelic, Ivana; Randjelovic, Danijela; Sharmin, Dishary; Cook, James M.; Savic, Miroslav M.; Savic, Snezana
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Development of non-sedating benzodiazepines with in vivo antischistosomal activity
err2024-09-04
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PREAI
errMian, Md Yeunus; Sharmin, Dishary; Mondal, Prithu; Belayet, Jawad Bin; Hossain, M. Mahmun; McCusker, Paul; Ryan, Kaetlyn T.; Fedorov, Alexander Y.; Green, Heather A.; Ericksen, Spencer S.; Zamanian, Mostafa; Tiruveedhula, V. V. N. Phani Babu; Cook, James M.; Chan, John D.
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An alpha 5-GABAA receptor positive allosteric modulator attenuates social and cognitive deficits without changing dopamine system hyperactivity in rats exposed to valproic acid in utero
err2024-06-22
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PREAI
errSouza, Adriana Jesus; Freitas, Icaro Silva; Sharmin, Dishary; Cook, James M.; Guimaraes, Francisco S.; Gomes, Felipe V.
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GABA(A) receptor activation drives GABARAP-Nix mediated autophagy to radiosensitize primary and metastatic lung adenocarcinoma tumors
err2024-03-22
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PREAI
errBhattacharya, Debanjan; Barrile, Riccardo; Toukam, Donatien Kamdem; Gawali, Vaibhavkumar S.; Kallay, Laura; Ahmed, Taukir; Brown, Hawley; Rezvanian, Sepideh; Karve, Aniruddha; Desai, Pankaj B.; Medvedovic, Mario; Wang, Kyle; Ionascu, Dan; Harun, Nusrat; Wang, Chenran; Baschnagel, Andrew M.; Kritzer, Joshua A.; Cook, James; Krummel, Daniel A. Pomeranz; Sengupta, Soma
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New Imidazodiazepine Analogue, 5-(8-Bromo-6-(pyridin-2-yl)-4H-benzo[f]imidazo[1,5-a][1,4]diazepin-3-yl)oxazole, Provides a Simplified Synthetic Scheme, High Oral Plasma and Brain Exposures, and Produces Antiseizure Efficacy in Mice, and Antiepileptogenic Activity in Neural Networks in Brain Slices from a Patient with Mesial Temporal Lobe Epilepsy
err2024-01-04
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PREAI
errSharmin, Dishary; Divovic, Branka; Ping, Xingjie; Cerne, Rok; Smith, Jodi L.; Rezvanian, Sepideh; Mondal, Prithu; Meyer, Michelle Jean; Kiley, Molly E.; Arnold, Leggy A.; Mian, Md Yeunus; Pandey, Kamal P.; Jin, Xiaoming; Mitrovic, Jelena R.; Djorovic, Djordje; Lippa, Arnold; Cook, James M.; Golani, Lalit K.; Scholze, Petra; Savic, Miroslav M.; Witkin, Jeffrey M.
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KRM-II-81 suppresses epileptifom activity across the neural network of cortical tissue from a patient with pharmacoresistant epilepsy
errHELIYON
IF3.6
err2024-01-01
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errSmith, Jodi L.; Wertz, Jeremy; Lippa, Arnold; Ping, Xingjie; Jin, Xiaoming; Cook, James M.; Witkin, Jeffrey M.; Cerne, Rok
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Freeze-dried nanocrystal dispersion of novel deuterated pyrazoloquinolinone ligand (DK-I-56-1): Process parameters and lyoprotectant selection through the stability study
err2023-10-01
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errMitrovic, Jelena R.; Ziberna, Maja Bjelosevic; Vukadinovic, Aleksandar; Knutson, Daniel E.; Sharmin, Dishary; Kremenovic, Aleksandar; Grabnar, Pegi Ahlin; Planinsekb, Odon; Lunter, Dominique; Cook, James M.; Savic, Miroslav M.; Savic, Snezana D.
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Synthesis and Receptor Binding Studies of α5 GABAAR Selective Novel Imidazodiazepines Targeted for Psychiatric and Cognitive Disorders
err2023-06-14
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errSharmin, Dishary; Mian, Md Yeunus; Marcotte, Michael; Prevot, Thomas D.; Sibille, Etienne; Witkin, Jeffrey M.; Cook, James M.
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Widening the Opioid Analgesia Therapeutic Window with a Dual Pharmacology Strategy
err2023-06-01
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errMadhuranthakam, Indu Mithra; Uribe, Sarah; Aldaghma, Danya; Kwitchoff, Drew; Philip, Jonathan; Williams, Aela A.; Nambiar, Rohit A.; Sharmin, Dishary; Cook, James; Fischer, Bradford; Keck, Thomas
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Structural Analogs of the GABAkine KRM-II-81 Are Orally Bioavailable Anticonvulsants without Sedation
err2023-04-01
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errPandey, Kamal P.; Divovic, Branka; Rashid, Farjana; Golani, Lalit K.; Cerne, Rok; Zahn, Nicolas M.; Meyer, Michelle Jean; Arnold, Leggy A.; Sharmin, Dishary; Mian, Md Yeunus; Smith, Jodi L.; Ping, Xingjie; Jin, Xiaoming; Lippa, Arnold; Tiruveedhula, V. V. N. Phani Babu; Cook, James M.; Savic, Miroslav M.; Witkin, Jeffrey M.
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Cerebellar α6GABAA Receptors as a Therapeutic Target for Essential Tremor: Proof-of-Concept Study with Ethanol and Pyrazoloquinolinones
err2023-03-01
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errHuang, Ya-Hsien; Lee, Ming Tatt; Hsueh, Han-Yun; Knutson, Daniel E.; Cook, James; Mihovilovic, Marko D.; Sieghart, Werner; Chiou, Lih-Chu
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Comparative anticonvulsant activity of the GABAkine KRM-II-81 and a deuterated analog
err2023-02-07
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errPing, Xingjie; Meyer, Michelle J.; Zahn, Nicolas M.; Golani, Lalit K.; Sharmin, Dishary; Pandey, Kamal P.; Revanian, Sepideh; Mondal, Prithu; Jin, Xiaoming; Arnold, Leggy A.; Cerne, Rok; Cook, James M.; Divovic, Branka; Savic, Miroslav M.; Lippa, Arnold; Smith, Jodi L.; Witkin, Jeffrey M.
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