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Luke Wharton

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12H-index
63Paper Count
372Citation Count
Published Papers 29
Publication Date
Challenging the Macrocycle Paradigm: Four-Arm; High-Denticity Acyclic Chelators for Radiopharmaceuticals Incorporating Actinium and Lanthanides
err2026-03-17
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errOAAI
errDaniel Fernández-Pavón; Andrés de Blas; María Martínez-Cabanas; José L. Barriada; Brian O. Patrick; Chris Orvig; François Bénard; Hua Yang; Luke Wharton; María de Guadalupe Jaraquemada-Peláez; Teresa Rodríguez-Blas
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Is Thiourea the Weak Link? An Investigation of the In Vitro and In Vivo Destabilization of [203Pb]- and [212Pb]Pb2+ Thiourea-Based Bioconjugates
err2025-12-01
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PREAI
errMcNeil, Brooke L.; Wharton, Luke; Chen, Chao-Cheng; Merkens, Helen; Colovic, Milena; Rodriguez-Rodriguez, Cristina; Wilson, John; Mair, Stefan; Zhang, Chengcheng; Mcdonagh, Anthony W.; Lin, Kuo-Shyan; Benard, Francois; Wuest, Frank; Schaffer, Paul; Ramogida, Caterina F.
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Carboxylic- and Amide Donor-Functionalized Pyridine-N-trans-Substituted Cyclen-Based Chelators for 203Pb/212Pb Theranostic Radiopharmaceuticals
err2025-10-24
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PREAI
errSimona Mastroianni; Thomas E. Karpiuk; Marianna Tosato; Parmissa Randhawa; Brooke L. McNeil; Luke Wharton; Scott W. McNeil; Hua Yang; Caterina F. Ramogida
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Synthesis and evaluation of HOPO-O8-Methyl-tetrazine as a bifunctional chelator for use in [89Zr]Zr4+, [161Tb]Tb3+ and [227Th]Th4+ radioimmunoconjugates
err2025-09-15
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errOAAI
errImma Carbo-Bague; Parmissa Randhawa; Marianna Tosato; Brooke L. McNeil; Milena Čolović; Lucas London; Cristina Rodríguez-Rodríguez; Maryam Osooly; Luke Wharton; Helen Merkens; Michiel Van De Voorde; Maarten Ooms; Hua Yang; François Bénard; Caterina F. Ramogida
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Chelating [227Th]Th4+ for Peptide Receptor Radionuclide Therapy of Neuroendocrine Tumors
err2025-05-10
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PREAI
errWharton, Luke; McNeil, Scott W.; Meeres, Harrison; Zhang, Diduo; Ingham, Aidan; Merkens, Helen; Osooly, Maryam; Rodriguez-Rodriguez, Cristina; Benard, Francois; Yang, Hua
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Preclinical evaluation of [225Ac]Ac-crown-TATE - An alpha-emitting radiopharmaceutical for neuroendocrine tumors
err2024-11-01
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PREAI
errIngham, Aidan; Wharton, Luke; Koniar, Helena; Merkens, Helen; Mcneil, Scott; Sekar, Sathiya; Osooly, Maryam; Rodriguez-Rodriguez, Cristina; Benard, Francois; Schaffer, Paul; Yang, Hua
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The H2S x macropa Series: Increasing the Chemical Softness of H2macropa with Sulfur Atoms to Chelate Radiometals [213Bi]Bi3+ and [203Pb]Pb2+ for Radiopharmaceutical Applications
err2024-10-22
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PREAI
errRandhawa, Parmissa; Kadassery, Karthika J.; McNeil, Brooke L.; MacMillan, Samantha N.; Wharton, Luke; Yang, Hua; Wilson, Justin J.; Ramogida, Caterina F.
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Preclinical Evaluation of 226Ac as a Theranostic Agent: Imaging, Dosimetry, and Therapy
err2024-10-03
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PREAI
errKoniar, Helena; Wharton, Luke; Ingham, Aidan; Oliver, Ana Paulina Morales; Merkens, Helen; Rodriguez-Rodriguez, Cristina; Kunz, Peter; Radchenko, Valery; Yang, Hua; Rahmim, Arman; Uribe, Carlos; Schaffer, Paul
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Quantitative SPECT imaging of 155Tb and 161Tb for preclinical theranostic radiopharmaceutical development
err2024-09-14
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errOAAI
errKoniar, Helena; McNeil, Scott; Wharton, Luke; Ingham, Aidan; van de Voorde, Michiel; Ooms, Maarten; Sekar, Sathiya; Rodriguez-Rodriguez, Cristina; Kunz, Peter; Radchenko, Valery; Rahmim, Arman; Uribe, Carlos; Yang, Hua; Schaffer, Paul
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Preclinical evaluation of MC1R targeting theranostic pair [ 155 Tb] Tb-crown- α MSH and [ 161 Tb]Tb-crown- α MSH
err2024-09-01
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PREAI
errWharton, Luke; Mcneil, Scott W.; Zhang, Chengcheng; Engudar, Gokce; Van de Voorde, Michiel; Zeisler, Jutta; Koniar, Helena; Sekar, Sathiya; Yuan, Zheliang; Schaffer, Paul; Radchenko, Valery; Ooms, Maarten; Kunz, Peter; Benard, Francois; Yang, Hua
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In vivo quantitative SPECT imaging of actinium-226: feasibility and proof-of-concept
err2024-07-16
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errOAAI
errKoniar, Helena; Wharton, Luke; Ingham, Aidan; Rodriguez-Rodriguez, Cristina; Kunz, Peter; Radchenko, Valery; Yang, Hua; Rahmim, Arman; Uribe, Carlos; Schaffer, Paul
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Rearmed Bifunctional Chelating Ligand for 225Ac/155Tb Precision-Guided Theranostic Radiopharmaceuticals-H4noneunpaX
err2023-09-22
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PREAI
errWharton, Luke; Yang, Hua; Jaraquemada-Pelaez, Maria de Guadalupe; Merkens, Helen; Engudar, Gokce; Ingham, Aidan; Koniar, Helena; Radchenko, Valery; Kunz, Peter; Schaffer, Paul; Benard, Francois; Orvig, Chris
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Separation of 44mSc/44gSc Nuclear Isomers Based on After-Effects
err2023-08-25
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PREAI
errKurakina, Elena Sergeevna; Wharton, Luke; Khushvaktov, Jurabek; Magomedbekov, Eldar Parpachevich; Radchenko, Valery; Filosofov, Dmitry
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Preclinical Evaluation of [155/161Tb]Tb-Crown-TATE-A Novel SPECT Imaging Theranostic Agent Targeting Neuroendocrine Tumours
err2023-04-01
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errOAAI
errWharton, Luke; McNeil, Scott W.; Merkens, Helen; Yuan, Zheliang; van de Voorde, Michiel; Engudar, Gokce; Ingham, Aidan; Koniar, Helena; Rodriguez-Rodriguez, Cristina; Radchenko, Valery; Ooms, Maarten; Kunz, Peter; Benard, Francois; Schaffer, Paul; Yang, Hua
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H3TPAN-Triazole-Bn-NH2: Tripicolinate Clicked-Bifunctional Chelate for [225Ac]/[111In] Theranostics
err2022-11-15
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PREAI
errWharton, Luke; Zhang, Chengcheng; Zeisler, Jutta; Rodriguez-Rodriguez, Cristina; Osooly, Maryam; Radchenko, Valery; Yang, Hua; Lin, Kuo-Shyan; Benard, Francois; Schaffer, Paul; Orvig, Chris
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Trastuzumab-conjugated oxine-based ligand for [89Zr]Zr4+ immunoPET
err2022-10-01
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PREAI
errSouthcott, Lily; Wharton, Luke; Rousseau, Julie; Merkens, Helen; Yang, Hua; Benard, Francois; Orvig, Chris
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H4picoopa-Robust Chelate for 225Ac/111In Theranostics
err2022-09-20
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PREAI
errWharton, Luke; Jaraquemada-Pelaez, Maria de Guadalupe; Zhang, Chengcheng; Zeisler, Jutta; Rodriguez-Rodriguez, Cristina; Osooly, Maryam; Radchenko, Valery; Yang, Hua; Lin, Kuo-Shyan; Benard, Francois; Schaffer, Paul; Orvig, Chris
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Toward Bifunctional Chelators for Thallium-201 for Use in Nuclear Medicine
err2022-07-08
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errOAAI
errRigby, Alex; Firth, George; Rivas, Charlotte; Pham, Truc; Kim, Jana; Phanopoulos, Andreas; Wharton, Luke; Ingham, Aidan; Li, Lily; Ma, Michelle; Orvig, Chris; Blower, Philip J.; Terry, Samantha Y. A.; Abbate, Vincenzo
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H2ampa-Versatile Chelator for [203Pb]Pb2+, [213Bi]Bi3+, and [225Ac]Ac3+
err2022-06-09
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PREAI
errIngham, Aidan; Wharton, Luke; El Sayed, Tarek; Southcott, Lily; McNeil, Brooke L.; Ezhova, Maria B.; Patrick, Brian O.; Jaraquemada-Pelaez, Maria de Guadalupe; Orvig, Chris
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Bis(amido)bis(oxinate)diamine Ligands for theranostic radiometals
err2022-06-01
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PREAI
errSouthcott, Lily; Whetter, Jennifer N.; Wharton, Luke; Patrick, Brian O.; Zarschler, Kristof; Kubeil, Manja; Stephan, Holger; Jaraquemada-Pelaez, Maria de Guadalupe; Orvig, Chris
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