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PIEZO1 regulates smooth muscle cell plasticity by integrating mechanical stretch with glycolytic metabolism Cao, Yapeng; Xu, Liran; Zhang, Min; Su, Ailing; Wang, Siyu; Li, Ting; Liu, Siyu; Mao, Ziyang; He, Yu; Shao, Zehua; Zhang, Jiamin; Wang, Youhua; Tian, Huijing; Sun, Yuzhuo; Li, Yongxin; Yan, Luqin; Zhang, Guangjian; Sun, Shiquan; Mei, Na; Chen, Fangyuan; Xiong, Ying; Liang, Guozheng; Offermanns, Stefan; Yan, Yang; Yuan, Zuyi; Wang, Shengpeng Share Save
The Concise Guide to PHARMACOLOGY 2025/26: Ion channels Alexander, Stephen P. H.; Striessnig, Jorg; Gibb, Alasdair J.; Mathie, Alistair A.; Veale, Emma L.; Kelly, Eamonn; Peach, Chloe J.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Aldrich, Richard W.; Attali, Bernard; Baggetta, Austin M.; Becirovic, Elvir; Beech, David J.; Biel, Martin; Bill, Roslyn M.; Caceres, Ana I.; Catterall, William A.; Chua, Han Chow; Conner, Alex C.; Danahay, Henry; Davies, Paul; De Clerq, Katrien; Delling, Markus; Di Virgilio, Francesco; Falzoni, Simonetta; Fang, Wei; Fenske, Stefanie; Fortuny-gomez, Anna; Fountain, Samuel; Chandy, George K.; Ghovanloo, Mohammad-reza; Goldstein, Steve A. N.; Gosling, Martin; Grimm, Christian; Grissmer, Stephan; Ha, Kotdaji; Hales, Tim G.; Hammelmann, Verena; Hanukoglu, Israel; Hu, Meiqin; Ijzerman, Ad P.; Jabba, Sairam V.; Jarvis, Mike; Jensen, Anders A.; Jordt, Sven E.; Kaczmarek, Leonard K.; Kellenberger, Stephan; Kennedy, Charles; King, Brian; Kitchen, Philip; Liu, Qiang; Lynch, Joseph W.; Manville, Rian W.; Meades, Jessica; Mehlfeld, Verena; Nicke, Annette; Offermanns, Stefan; Perez-reyes, Edward; Plant, Leigh D.; Pless, Stephan A.; Rash, Lachlan D.; Ren, Dejian; Rubaiy, Hussein N.; Salman, Mootaz M.; Sieghart, Werner; Sivilotti, Lucia G.; Smart, Trevor G.; Snutch, Terrance P.; Tammaro, Paolo; Tian, Jinbin; Trimmer, James S.; Van Den Eynde, Charlotte; Vergani, Paola; Vriens, Joris; Waxman, Stephen G.; Wei, Aguan D.; Winn, Brenda T.; Wulff, Heike; Xu, Haoxing; Yang, Fan; Yue, Lixia; Zhang, Xiaoli; Zhu, Michael Share Save
The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors Alexander, Stephen P. H.; Davenport, Anthony P.; Kelly, Eamonn; Gibb, Alasdair J.; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George R.; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bennett, Kirstie A.; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria A.; Bonaventure, Pascal; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Brown, Andrew J.; Burnstock, Geoffrey; Busnelli, Marta; Calo, Girolamo; Caruso, Vanni; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Christopoulos, Arthur; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dautzenberg, Frank M.; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Dubocovich, Margarita L.; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Forsman, Huamei Fu; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gbahou, Florence; Gerard, Craig; Gershengorn, Marvin; Glass, Michelle; Gloriam, David E.; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gruber, Christian; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hartman, Deborah S.; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Heitman, Laura; Herr, Deron R.; Hollenberg, Morley D.; Holliday, Nicholas D.; Holst, Birgitte; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Insel, Paul A.; Jacobson, Kenneth A.; Jacobson, Laura H.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kinsolving, Julia; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Laishram, Luxmichan; Langenhan, Tobias; Langmead, Christopher J.; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Leurs, Rob; Li, Xaria X.; Liebscher, Ines; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet J.; Malfacini, Davide; Manning, Maurice; Marangon, Davide; Martemyanov, Kirill; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Neubig, Richard R.; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Perry-Hauser, Nicole; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Qin, Helena Chengxue; Quinn, Mark; Raffaele, Stefano; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Buzon, Alejandro Romeral; Rondard, Philippe; Rosenkilde, Mette M.; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Scholz, Nicole; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Shukla, Arun K.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Smith, Nicola J.; Staeubert, Claudia; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David M.; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Verbalis, Joseph G.; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Wu, Huixian; Yang, Cheng; Yao, Chengcan; Ye, Richard D.; Zaidman, Nathan Share Save
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Butyrate receptor HCAR2/GPR109A controls imiquimod-induced psoriasis-like skin inflammation Leko, Lucija; Simic, Darija; Martins, Timna Valera; da Silva, Gabriel Victor Lucena; Maillet, Isabelle; Savigny, Florence; Vuksan, Lara; Rodrigues, Dorian de Moura; Le Bert, Marc; Offermanns, Stefan; Riteau, Nicolas; Togbe, Dieudonnee; Quesniaux, Valerie F.; Russo, Remo Castro Share Save
FFAR4-mediated IL-6 release from islet macrophages promotes insulin secretion and is compromised in type-2 diabetes Chen, Xinyi; Shao, Jingchen; Brandenburger, Isabell; Qian, Weikun; Hahnefeld, Lisa; Bonnavion, Remy; Cho, Haaglim; Wang, ShengPeng; Hidalgo, Juan; Wettschureck, Nina; Geisslinger, Gerd; Gurke, Robert; Wang, Zheng; Offermanns, Stefan Share Save
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ALPK2 prevents cardiac diastolic dysfunction in heart failure with preserved ejection fraction Yoshida, Tatsuya; Yoshida, Satoya; Inukai, Kohei; Kato, Katsuhiro; Yura, Yoshimitsu; Hattori, Tomoki; Taki, Kentaro; Enomoto, Atsushi; Ohashi, Koji; Okumura, Takahiro; Ouchi, Noriyuki; Kawase, Haruya; Wettschureck, Nina; Offermanns, Stefan; Murohara, Toyoaki; Takefuji, Mikito Share Save
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SPMs exert anti- inflammatory and pro- resolving effects through positive allosteric modulation of the prostaglandin EP4 receptor Alnouri, Mohamad Wessam; Roquid, Kenneth Anthony; Bonnavion, Remy; Cho, Haaglim; Heering, Jan; Kwon, Jeonghyeon; Jaeger, Yannick; Wang, ShengPeng; Guenther, Stefan; Wettschureck, Nina; Geisslingerb, Gerd; Gurke, Robert; Mueller, Christa E.; Proschak, Ewgenij; Offermanns, Stefan Share Save
Protein kinase N promotes cardiac fibrosis in heart failure by fibroblast-to-myofibroblast conversion Yoshida, Satoya; Yoshida, Tatsuya; Inukai, Kohei; Kato, Katsuhiro; Yura, Yoshimitsu; Hattori, Tomoki; Enomoto, Atsushi; Ohashi, Koji; Okumura, Takahiro; Ouchi, Noriyuki; Kawase, Haruya; Wettschureck, Nina; Offermanns, Stefan; Murohara, Toyoaki; Takefuji, Mikito Share Save
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Bitter tastants relax the mouse gallbladder smooth muscle independent of signaling through tuft cells and bitter taste receptors Keshavarz, Maryam; Ruppert, Anna-Lena; Meiners, Mirjam; Poharkar, Krupali; Liu, Shuya; Mahmoud, Wafaa; Winterberg, Sarah; Hartmann, Petra; Mermer, Petra; Perniss, Alexander; Offermanns, Stefan; Kummer, Wolfgang; Schuetz, Burkhard Share Save
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