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CDK9 inhibition constrains multiple oncogenic transcriptional and epigenetic pathways in prostate cancer (vol 131, pg 1092, 2024) Rahman, Razia; Rahaman, Muhammed H.; Hanson, Adrienne R.; Choo, Nicholas; Xie, Jianling; Townley, Scott L.; Shrestha, Raj; Hassankhani, Ramin; Islam, Saiful; Ramm, Susanne; Simpson, Kaylene J.; Risbridger, Gail P.; Best, Giles; Centenera, Margaret M.; Balk, Steven P.; Kichenadasse, Ganessan; Taylor, Renea A.; Butler, Lisa M.; Tilley, Wayne D.; Conn, Simon J.; Lawrence, Mitchell G.; Wang, Shudong; Selth, Luke A. Share Save
CDK9 inhibition inhibits multiple oncogenic transcriptional and epigenetic pathways in prostate cancer Rahman, Razia; Rahaman, Muhammed H.; Hanson, Adrienne R.; Choo, Nicholas; Xie, Jianling; Townley, Scott L.; Shrestha, Raj; Hassankhani, Ramin; Islam, Saiful; Ramm, Susanne; Simpson, Kaylene J.; Risbridger, Gail P.; Best, Giles; Centenera, Margaret M.; Balk, Steven P.; Kichenadasse, Ganessan; Taylor, Renea A.; Butler, Lisa M.; Tilley, Wayne D.; Conn, Simon J.; Lawrence, Mitchell G.; Wang, Shudong; Selth, Luke A. Share Save
ACSM1 and ACSM3 Regulate Fatty Acid Metabolism to Support Prostate Cancer Growth and Constrain Ferroptosis Shrestha, Raj K.; Nassar, Zeyad D.; Hanson, Adrienne R.; Iggo, Richard; Townley, Scott L.; Dehairs, Jonas; Mah, Chui Y.; Helm, Madison; Alizadeh-Ghodsi, Mohammadreza; Pickering, Marie; Ghesquiere, Bart; Watt, Matthew J.; Quek, Lake-Ee; Hoy, Andrew J.; Tilley, Wayne D.; Swinnen, Johannes V.; Butler, Lisa M.; Selth, Luke A. Share Save
Library size confounds biology in spatial transcriptomics data Bhuva, Dharmesh D.; Tan, Chin Wee; Salim, Agus; Marceaux, Claire; Pickering, Marie A.; Chen, Jinjin; Kharbanda, Malvika; Jin, Xinyi; Liu, Ning; Feher, Kristen; Putri, Givanna; Tilley, Wayne D.; Hickey, Theresa E.; Asselin-Labat, Marie-Liesse; Phipson, Belinda; Davis, Melissa J. Share Save
The androgen receptor interacts with GATA3 to transcriptionally regulate a luminal epithelial cell phenotype in breast cancer Hosseinzadeh, Leila; Kikhtyak, Zoya; Laven-Law, Geraldine; Pederson, Stephen M.; Puiu, Caroline G.; D'Santos, Clive S.; Lim, Elgene; Carroll, Jason S.; Tilley, Wayne D.; Dwyer, Amy R.; Hickey, Theresa E. Share Save
Selective inhibition of CDK9 in triple negative breast cancer Mustafa, Ebtihal H.; Laven-Law, Geraldine; Kikhtyak, Zoya; Nguyen, Van; Ali, Simak; Pace, Alex A.; Iggo, Richard; Kebede, Alemwork; Noll, Ben; Wang, Shudong; Winter, Jean M.; Dwyer, Amy R.; Tilley, Wayne D.; Hickey, Theresa E. Share Save
Luminal breast cancer identity is determined by loss of glucocorticoid receptor activity Prekovic, Stefan; Chalkiadakis, Theofilos; Roest, Merel; Roden, Daniel; Lutz, Catrin; Schuurman, Karianne; Opdam, Mark; Hoekman, Liesbeth; Abbott, Nina; Tesselaar, Tanja; Wajahat, Maliha; Dwyer, Amy R.; Mayayo-Peralta, Isabel; Gomez, Gabriela; Altelaar, Maarten; Beijersbergen, Roderick; Gyorffy, Balazs; Young, Leonie; Linn, Sabine; Jonkers, Jos; Tilley, Wayne; Hickey, Theresa; Vareslija, Damir; Swarbrick, Alexander; Zwart, Wilbert Share Save
Designing Fluorescent Nuclear Permeable Peptidomimetics to Target Proliferating Cell Nuclear Antigen Horsfall, Aimee J.; Chav, Theresa; Pederick, Jordan L.; Kikhtyak, Zoya; Vandborg, Bethiney C.; Kowalczyk, Wioleta; Scanlon, Denis B.; Tilley, Wayne D.; Hickey, Theresa E.; Abell, Andrew D.; Bruning, John B. Share Save
Selective Androgen Receptor Modulators in combination with CDK4/6 inhibitors demonstrate anti-cancer activity in preclinical treatment resistant ER plus AR plus breast cancer models Freelander, Allegra; Laven-Law, Geraldine; Eshraghi, Leila; Geetha, Nimmy; Somerville, Peta; Pickering, Marie; Alexandrou, Sarah; Caldon, C. Elizabeth; Tilley, Wayne D.; Hickey, Theresa E.; Lim, Elgene Share Save
Combination CDK4/6 inhibition and AR agonism suppresses the growth of CDK4/6 inhibitor resistant breast cancers Freelander, Allegra; Laven-Law, Geraldine; Eshraghi, Leila; Chia, Kee Ming; Pickering, Marie; Yong, Aliza; Wilkinson, Ashleigh; Alexandrou, Sarah; Caldon, C. Elizabeth; Hickey, Theresa E.; Tilley, Wayne D.; Lim, Elgene Share Save
Opposing transcriptional programs of KLF5 and AR emerge during therapy for advanced prostate cancer Che, Meixia; Chaturvedi, Aashi; Munro, Sarah A.; Pitzen, Samuel P.; Ling, Alex; Zhang, Weijie; Mentzer, Josh; Ku, Sheng-Yu; Puca, Loredana; Zhu, Yanyun; Bergman, Andries M.; Severson, Tesa M.; Forster, Colleen; Liu, Yuzhen; Hildebrand, Jacob; Daniel, Mark; Wang, Ting-You; Selth, Luke A.; Hickey, Theresa; Zoubeidi, Amina; Gleave, Martin; Bareja, Rohan; Sboner, Andrea; Tilley, Wayne; Carroll, Jason S.; Tan, Winston; Kohli, Manish; Yang, Rendong; Hsieh, Andrew C.; Murugan, Paari; Zwart, Wilbert; Beltran, Himisha; Huang, R. Stephanie; Dehm, Scott M. Share Save
An androgen receptor switch underlies lineage infidelity in treatment-resistant prostate cancer Davies, Alastair; Nouruzi, Shaghayegh; Ganguli, Dwaipayan; Namekawa, Takeshi; Thaper, Daksh; Linder, Simon; Karaoglanoglu, Fatih; Omur, Meltem E.; Kim, Soojin; Kobelev, Maxim; Kumar, Sahil; Sivak, Olena; Bostock, Chiara; Bishop, Jennifer; Hoogstraat, Marlous; Talal, Amina; Stelloo, Suzan; van der Poel, Henk; Bergman, Andries M.; Ahmed, Musaddeque; Fazli, Ladan; Huang, Haojie; Tilley, Wayne; Goodrich, David; Feng, Felix Y.; Gleave, Martin; He, Housheng Hansen; Hach, Faraz; Zwart, Wilbert; Beltran, Himisha; Selth, Luke; Zoubeidi, Amina Share Save
Lipidomic Profiling of Clinical Prostate Cancer Reveals Targetable Alterations in Membrane Lipid Composition Butler, Lisa M.; Mah, Chui Yan; Machiels, Jelle; Vincent, Andrew D.; Irani, Swati; Mutuku, Shadrack M.; Spotbeen, Xander; Bagadi, Muralidhararao; Waltregny, David; Moldovan, Max; Dehairs, Jonas; Vanderhoydonc, Frank; Bloch, Katarzyna; Das, Rajdeep; Stahl, Jurgen; Kench, James G.; Gevaert, Thomas; Derua, Rita; Waelkens, Etienne; Nassar, Zeyad D.; Selth, Luke A.; Trim, Paul J.; Snel, Marten F.; Lynn, David J.; Tilley, Wayne D.; Horvath, Lisa G.; Centenera, Margaret M.; Swinnen, Johannes, V Share Save
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ELOVL5 Is a Critical and Targetable Fatty Acid Elongase in Prostate Cancer Centenera, Margaret M.; Scott, Julia S.; Machiels, Jelle; Nassar, Zeyad D.; Miller, Deanna C.; Zinonos, Irene; Dehairs, Jonas; Burvenich, Ingrid J. G.; Zadra, Giorgia; Chetta, Paolo M.; Bango, Clyde; Evergren, Emma; Ryan, Natalie K.; Gillis, Joanna L.; Mah, Chui Yan; Tieu, Terence; Hanson, Adrienne R.; Carelli, Ryan; Bloch, Katarzyna; Panagopoulos, Vasilios; Waelkens, Etienne; Derua, Rita; Williams, Elizabeth D.; Evdokiou, Andreas; Cifuentes-Rius, Anna; Voelcker, Nicolas H.; Mills, Ian G.; Tilley, Wayne D.; Scott, Andrew M.; Loda, Massimo; Selth, Luke A.; Swinnen, Johannes, V; Butler, Lisa M. Share Save
The androgen receptor is a tumor suppressor in estrogen receptor-positive breast cancer Hickey, Theresa E.; Selth, Luke A.; Chia, Kee Ming; Laven-Law, Geraldine; Milioli, Heloisa H.; Roden, Daniel; Jindal, Shalini; Hui, Mun; Finlay-Schultz, Jessica; Ebrahimie, Esmaeil; Birrell, Stephen N.; Stelloo, Suzan; Iggo, Richard; Alexandrou, Sarah; Caldon, C. Elizabeth; Abdel-Fatah, Tarek M.; Ellis, Ian O.; Zwart, Wilbert; Palmieri, Carlo; Sartorius, Carol A.; Swarbrick, Alex; Lim, Elgene; Carroll, Jason S.; Tilley, Wayne D. Share Save
Trans-ancestry genome-wide association meta-analysis of prostate cancer identifies new susceptibility loci and informs genetic risk prediction Conti, David, V; Darst, Burcu F.; Moss, Lilit C.; Saunders, Edward J.; Sheng, Xin; Chou, Alisha; Schumacher, Fredrick R.; Al Olama, Ali Amin; Benlloch, Sara; Dadaev, Tokhir; Brook, Mark N.; Sahimi, Ali; Hoffmann, Thomas J.; Takahashi, Atushi; Matsuda, Koichi; Momozawa, Yukihide; Fujita, Masashi; Muir, Kenneth; Lophatananon, Artitaya; Wan, Peggy; Le Marchand, Loic; Wilkens, Lynne R.; Stevens, Victoria L.; Gapstur, Susan M.; Carter, Brian D.; Schleutker, Johanna; Tammela, Teuvo L. J.; Sipeky, Csilla; Auvinen, Anssi; Giles, Graham G.; Southey, Melissa C.; MacInnis, Robert J.; Cybulski, Cezary; Wokolorczyk, Dominika; Lubinski, Jan; Neal, David E.; Donovan, Jenny L.; Hamdy, Freddie C.; Martin, Richard M.; Nordestgaard, Borge G.; Nielsen, Sune F.; Weischer, Maren; Bojesen, Stig E.; Roder, Martin Andreas; Iversen, Peter; Batra, Jyotsna; Chambers, Suzanne; Moya, Leire; Horvath, Lisa; Clements, Judith A.; Tilley, Wayne; Risbridger, Gail P.; Gronberg, Henrik; Aly, Markus; Szulkin, Robert; Eklund, Martin; Nordstrom, Tobias; Pashayan, Nora; Dunning, Alison M.; Ghoussaini, Maya; Travis, Ruth C.; Key, Tim J.; Riboli, Elio; Park, Jong Y.; Sellers, Thomas A.; Lin, Hui-Yi; Albanes, Demetrius; Weinstein, Stephanie J.; Mucci, Lorelei A.; Giovannucci, Edward; Lindstrom, Sara; Kraft, Peter; Hunter, David J.; Penney, Kathryn L.; Turman, Constance; Tangen, Catherine M.; Goodman, Phyllis J.; Thompson, Ian M., Jr.; Hamilton, Robert J.; Fleshner, Neil E.; Finelli, Antonio; Parent, Marie-Elise; Stanford, Janet L.; Ostrander, Elaine A.; Geybels, Milan S.; Koutros, Stella; Freeman, Laura E. Beane; Stampfer, Meir; Wolk, Alicja; Hakansson, Niclas; Andriole, Gerald L.; Hoover, Robert N.; Machiela, Mitchell J.; Sorensen, Karina Dalsgaard; Borre, Michael; Blot, William J.; Zheng, Wei; Yeboah, Edward D.; Mensah, James E.; Lu, Yong-Jie; Zhang, Hong-Wei; Feng, Ninghan; Mao, Xueying; Wu, Yudong; Zhao, Shan-Chao; Sun, Zan; Thibodeau, Stephen N.; McDonnell, Shannon K.; Schaid, Daniel J.; West, Catharine M. L.; Burnet, Neil; Barnett, Gill; Maier, Christiane; Schnoeller, Thomas; Luedeke, Manuel; Kibel, Adam S.; Drake, Bettina F.; Cussenot, Olivier; Cancel-Tassin, Geraldine; Menegaux, Florence; Truong, Therese; Koudou, Yves Akoli; John, Esther M.; Grindedal, Eli Marie; Maehle, Lovise; Khaw, Kay-Tee; Ingles, Sue A.; Stern, Mariana C.; Vega, Ana; Gomez-Caamano, Antonio; Fachal, Laura; Rosenstein, Barry S.; Kerns, Sarah L.; Ostrer, Harry; Teixeira, Manuel R.; Paulo, Paula; Brandao, Andreia; Watya, Stephen; Lubwama, Alexander; Bensen, Jeannette T.; Fontham, Elizabeth T. H.; Mohler, James; Taylor, Jack A.; Kogevinas, Manolis; Llorca, Javier; Castano-Vinyals, Gemma; Cannon-Albright, Lisa; Teerlink, Craig C.; Huff, Chad D.; Strom, Sara S.; Multigner, Luc; Blanchet, Pascal; Brureau, Laurent; Kaneva, Radka; Slavov, Chavdar; Mitev, Vanio; Leach, Robin J.; Weaver, Brandi; Brenner, Hermann; Cuk, Katarina; Holleczek, Bernd; Saum, Kai-Uwe; Klein, Eric A.; Hsing, Ann W.; Kittles, Rick A.; Murphy, Adam B.; Logothetis, Christopher J.; Kim, Jeri; Neuhausen, Susan L.; Steele, Linda; Ding, Yuan Chun; Isaacs, William B.; Nemesure, Barbara; Hennis, Anselm J. M.; Carpten, John; Pandha, Hardev; Michael, Agnieszka; De Ruyck, Kim; De Meerleer, Gert; Ost, Piet; Xu, Jianfeng; Razack, Azad; Lim, Jasmine; Teo, Soo-Hwang; Newcomb, Lisa F.; Lin, Daniel W.; Fowke, Jay H.; Neslund-Dudas, Christine; Rybicki, Benjamin A.; Gamulin, Marija; Lessel, Davor; Kulis, Tomislav; Usmani, Nawaid; Singhal, Sandeep; Parliament, Matthew; Claessens, Frank; Joniau, Steven; Van den Broeck, Thomas; Gago-Dominguez, Manuela; Castelao, Jose Esteban; Martinez, Maria Elena; Larkin, Samantha; Townsend, Paul A.; Aukim-Hastie, Claire; Bush, William S.; Aldrich, Melinda C.; Crawford, Dana C.; Srivastava, Shiv; Cullen, Jennifer C.; Petrovics, Gyorgy; Casey, Graham; Roobol, Monique J.; Jenster, Guido; van Schaik, Ron H. N.; Hu, Jennifer J.; Sanderson, Maureen; Varma, Rohit; McKean-Cowdin, Roberta; Torres, Mina; Mancuso, Nicholas; Berndt, Sonja, I; Van den Eeden, Stephen K.; Easton, Douglas F.; Chanock, Stephen J.; Cook, Michael B.; Wiklund, Fredrik; Nakagawa, Hidewaki; Witte, John S.; Eeles, Rosalind A.; Kote-Jarai, Zsofia; Haiman, Christopher A. Share Save
Post-transcriptional Gene Regulation by MicroRNA-194 Promotes Neuroendocrine Transdifferentiation in Prostate Cancer Fernandes, Rayzel C.; Toubia, John; Townley, Scott; Hanson, Adrienne R.; Dredge, B. Kate; Pillman, Katherine A.; Bert, Andrew G.; Winter, Jean M.; Iggo, Richard; Das, Rajdeep; Obinata, Daisuke; Sandhu, Shahneen; Risbridger, Gail P.; Taylor, Renea A.; Lawrence, Mitchell G.; Butler, Lisa M.; Zoubeidi, Amina; Gregory, Philip A.; Tilley, Wayne D.; Hickey, Theresa E.; Goodall, Gregory J.; Selth, Luke A. Share Save
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