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SaveCDK12/13 inactivation triggers STING-mediated antitumor immunity in preclinical models
Bao, Yi; Chang, Yu; Tien, Jean Ching-Yi; Cruz, Gabriel; Yang, Fan; Mannan, Rahul; Mahapatra, Somnath; Paturu, Radha; Cao, Xuhong; Su, Fengyun; Wang, Rui; Zhang, Yuping; Gondal, Mahnoor; Choi, Jae eun; Gurkan, Jonathan K.; Miner, Stephanie J.; Robinson, Dan R.; Wu, Yi-Mi; Zhou, Licheng; Wang, Zhen; Kryczek, Ilona; Wang, Xiaoju; Cieslik, Marcin; Qiao, Yuanyuan; Tsodikov, Alexander; Zou, Weiping; Ding, Ke; Chinnaiyan, Arul M.
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SaveTherapeutic benefit of the dual ALK/FAK inhibitor ESK440 in ALK-driven neuroblastoma
Chugh, Seema; Tien, Jean C.; Hon, Jennifer; Kenum, Carson; Mannan, Rahul; Cheng, Yunhui; Li, Chi Chiang; Taher, Zainab I.; Delekta, Andrew D.; Bawa, Pushpinder Singh; Apel, Ingrid J.; Miner, Stephanie J.; Cao, Xuhong; Mehra, Rohit; Dhanasekaran, Saravana M.; Qiao, Yuanyuan; Mody, Rajen; Chinnaiyan, Arul M.
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SaveTargeting PIKfyve-driven lipid metabolism in pancreatic cancer
Cheng, Caleb; Wisniewski, Jasmine P.; Peters, Sydney; Hu, Jing; Mannan, Rahul; Jackson, Bailey; Pakkan, Ruya; Morlacchi, Pietro; Magnuson, Brian; He, Tongchen; Bhattacharyya, Rupam; Qiao, Yuanyuan; Lyssiotis, Costas A.; Chinnaiyan, Arul M.
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SaveNSD2 is a requisite subunit of the AR/FOXA1 neo-enhanceosome in promoting prostate tumorigenesis
Parolia, Abhijit; Eyunni, Sanjana; Verma, Brijesh Kumar; Young, Eleanor; Liu, Yihan; Liu, Lianchao; George, James; Aras, Shweta; Das, Chandan Kanta; Mannan, Rahul; Rasool, Reyaz Ur; Mitchell-Velasquez, Erick; Mahapatra, Somnath; Luo, Jie; Carson, Sandra E.; Xiao, Lanbo; Gajjala, Prathibha R.; Venkatesh, Sharan; Jaber, Mustapha; Wang, Xiaoju; He, Tongchen; Qiao, Yuanyuan; Pang, Matthew; Zhang, Yuping; Tien, Jean Ching-Yi; Louw, Micheala; Alhusayan, Mohammed; Cao, Xuhong; Su, Fengyun; Tavana, Omid; Hou, Caiyun; Wang, Zhen; Ding, Ke; Chinnaiyan, Arul M.; Asangani, Irfan A.
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SavePIKfyve, expressed by CD11c-positive cells, controls tumor immunity
Choi, Jae Eun; Qiao, Yuanyuan; Kryczek, Ilona; Yu, Jiali; Gurkan, Jonathan; Bao, Yi; Gondal, Mahnoor; Tien, Jean Ching-Yi; Maj, Tomasz; Yazdani, Sahr; Parolia, Abhijit; Xia, Houjun; Zhou, Jiajia; Wei, Shuang; Grove, Sara; Vatan, Linda; Lin, Heng; Li, Gaopeng; Zheng, Yang; Zhang, Yuping; Cao, Xuhong; Su, Fengyun; Wang, Rui; He, Tongchen; Cieslik, Marcin; Green, Michael D.; Zou, Weiping; Chinnaiyan, Arul M.
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SaveClinically Relevant Humanized Mouse Models of Metastatic Prostate Cancer Facilitate Therapeutic Evaluation
Kostlan, Raymond J.; Phoenix, John T.; Budreika, Audris; Ferrari, Marina G.; Khurana, Neetika; Choi, Jae E.; Juckette, Kristin; Mahapatra, Somnath; McCollum, Brooke L.; Moskal, Russell; Mannan, Rahul; Qiao, Yuanyuan; Vander Griend, Donald J.; Chinnaiyan, Arul M.; Kregel, Steven
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SaveDiscovery of LLC0424 as a Potent and Selective in Vivo NSD2 PROTAC Degrader
Liu, Lianchao; Parolia, Abhijit; Liu, Yihan; Hou, Caiyun; He, Tongchen; Qiao, Yuanyuan; Eyunni, Sanjana; Luo, Jie; Li, Chungen; Wang, Yongxing; Zhou, Fengtao; Huang, Weixue; Ren, Xiaomei; Wang, Zhen; Chinnaiyan, Arul M.; Ding, Ke
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SaveTargeting the SWI/SNF complex in POU2F-POU2AF transcription factor-driven malignancies
Xiao, Lanbo; He, Tongchen; Klingbeil, Olaf; Eleanor, Young; Wu, Xiaoli; Qiao, Yuanyuan; Parolia, Abhijit; Eyunni, Sanjana; Mannan, Rahul; Mahapatra, Somnath; Kim, NamHoon; Zheng, Heng; Su, Fengyun; Cao, Xuhong; Samajdar, Susanta; Ramachandra, Murali; Vakoc, Christopher R.; Chinnaiyan, Arul M.
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SaveTargeting the lipid kinase PIKfyve upregulates surface expression of MHC class I to augment cancer immunotherapy
Borker, Parth; Bao, Yi; Qiao, Yuanyuan; Chinnaiyan, Arul; Choi, Jae Eun; Zhang, Yuping; Mannan, Rahul; Cheng, Caleb; He, Tongchen; Zheng, Yang; Yu, Jiali; Gondal, Mahnoor; Cruz, Gabriel; Grove, Sara Sara; Cao, Xuhong; Su, Fengyun; Wang, Rui; Chang, Yu; Kryczek, Ilona; Cieslik, Marcin; Green, Michael D.; Zou, Weiping
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