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Single versus dual EGFR/PARP inhibition: Mechanistic rationale, synthetic approaches, pharmacophoric features, structure-activity relationships, and therapeutic perspectives 单药与联合EGFR/PARP抑制:作用机制依据、合成方法、药效团特征、构效关系及治疗前景 Elkafoury, Eman M.; El-Moselhy, Tarek F.; El-Hamamsy, Mervat H.; El-Bastawissy, Eman A.; Rabea, Esraa Y.; Afarinkia, Kamyar; Sidhom, Peter A. 分享 收藏
Michael like formation of isoquinoline-based pyrido[2,1 a]isoquinoline-carbonitriles: X-Ray structure confirmation, antibacterial activity, and molecular docking studies 迈克尔加成反应形成异喹啉基吡啶[2,1-a]异喹啉-碳腈:X射线结构确认、抗菌活性及分子对接研究 Teleb, Mohamed A. Mohamed; Hassaneen, Hamdi M.; Abdelhamid, Ismail A.; Ibrahim, Nada S.; Alaasar, Mohamed; Wagner, Christoph; Saleh, Fatma M. 分享 收藏
Crystal structure and computational study of a multifunctional 3-Spi-ro-2-oxindole derivative: Ethyl 4-[2-(2′-oxospiro[1,3-dioxolane-2,3′-indol]-1′(2′H)-yl)acetamido]benzoate 一种多功能3-螺-2-氧代吲哚衍生物的晶体结构与计算研究:乙基4-[2-(2′-氧代螺[1,3-二氧杂环戊烷-2,3′-吲哚]-1′(2′H)-基)乙酰胺基]苯甲酸酯 Sweify, Islam R.; El-Wahab, Hend A. A. Abdel; Qayed, Wesam S.; Bandaru, Siva S. M.; Schulzke, Carola; Aboul-Fadl, Tarek 分享 收藏
Strategic synthesis, antimicrobial evaluation, and computational insights into novel thieno[2,3-d]pyrimidines: From scaffold diversification to stable DHFR inhibition 战略性合成、抗菌活性评价及计算研究:新型噻吩[2,3-d]嘧啶类化合物的骨架多样化与稳定DHFR抑制 Sayed, Mostafa; Naguib, Menna A.; El-Rashedy, Ahmed A.; Hamed, Mahmoud M.; Hassanien, Reda; Ahmed, Mostafa; Tolba, Mahmoud S. 分享 收藏
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Synthesis, characterization, theoretical investigation, and biological evaluation of guanosine-based Ni(II), Cu(II), Pd(II), and Pt(II) complexes 基于鸟嘌呤的Ni(II)、Cu(II)、Pd(II)和Pt(II)配合物的合成、表征、理论研究和生物评价 Al-Farraj, Eida S.; El-Reash, Yasmeen G. Abou; El-Reash, Gaber M. I. Abu; Younis, Adel M. 分享 收藏
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STING organelle stress sensing in the liver drives hepatocyte fate and remodeling STING细胞器应激传感在肝脏中驱动肝细胞命运和重塑 Hamad, Rabab S.; Elmorsy, Elsayed A.; Elnaghy, Fatma; Amer, Maha M.; Abdel-Hamed, Mohamed R.; Farrag, Alshaimaa A.; Eissa, Hanan; El-kott, Attalla F.; Negm, Sally; AlShehri, Mohammed A.; Ali, Mohamed A. M.; Chaudhary, Anis Ahmad; Saber, Sameh 分享 收藏
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Impact of high-fat diet on the expression and distribution of Aquaporins 1, 3, 7, 8, and 9 in the rat parotid gland 高脂饮食对大鼠腮腺中水通道蛋白1、3、7、8和9的表达及分布的影响 Eldesoqui, Mamdouh; Sherif, Rania N.; Erfan, Omnia S.; Mohamed, Shrouk B.; Albadawi, Emad A.; Embaby, Eman M.; Hamada, Amal Saber; El-Desoky, Manal M.; Hendawy, Mahmoud 分享 收藏
Posterior versus anterior circulation infarct location and outcomes after breakthrough ischemic stroke in orally anticoagulated patients for atrial fibrillation: An ASPERA-R inverse probability-weighted analysis 心房颤动口服抗凝患者突破性缺血性卒中后,后循环与前循环梗死部位的比较及预后:一项ASPERA-R逆概率加权分析 Foschi, Matteo; D'Anna, Lucio; Gabriele, Francesca; Ornello, Raffaele; Zini, Andrea; Paolucci, Matteo; Forlivesi, Stefano; Migliaccio, Ludovica; Viola, Maria Maddalena; Rizzo, Angelo Cascio; Sessa, Maria; Schwarz, Ghil; Tortorella, Rachele; Jaffar, Muhammad; Prandin, Gabriele; Pantoni, Leonardo; Mele, Francesco; Scopelliti, Giuseppe; Cova, Ilaria; Valente, Mariarosaria; Maisano, Domenico; Antonelli, Luca; Bagnato, Maria Rosaria; Di Mauro, Giovanni; Bernocchi, Francesca; Di Donna, Martina Gaia; Casolla, Barbara; Ciacciarelli, Antonio; Bruno, Chiara; Alvarez, Baptiste; Gonzalez-Martin, Laura; Rigual, Ricardo; Fuentes, Blanca; Hervas, Carlos; Candelaresi, Paolo; Andreone, Vincenzo; De Mase, Antonio; Spina, Emanuele; de Sousa, Diana Aguiar; Souza, Mariana Almudi; Fior, Alberto; Serodio, Miguel; Caliandro, Pietro; Zauli, Aurelia; Reale, Giuseppe; Abdelalim, Ahmed; Ahmed, Sandra; Soliman, Nourhan Mohamed; Zhang, Liqun; Latimer, Tara; Elboghday, Muhammad; Elbassiouny, Ahmed Aly; Roushdy, Tamer; Shokri, Hossam; Ferrari, Federica; Loizzo, Nicola Davide; Mazzacane, Federico; Guarino, Maria; Barone, Valentina; Forti, Paola; Rinaldi, Giuseppe; Rossi, Marco Vito; Laterza, Vincenzo; Frisullo, Giovanni; Rizzo, Pier Andrea; Broccolini, Aldobrando; Mannino, Marina; Terruso, Valeria; Caggiula, Marcella; Rizzo, Annalisa; Fonseca, Ana Catarina; Antunes, Bernardo; Barbosa, Ana M.; Budincevic, Hrvoje; Crnac, Petra; Viticchi, Giovanna; Silvestrini, Mauro; Barba, Lorenzo; Musienko, Viktoria; Otto, Markus; Lochner, Piergiorgio; Landau, Benjamin; Buddha, Sandeep; Khalil, Roumeisa; Miserocchi, Ludovica Maria; Balducci, Giorgia; Piscaglia, Maria Grazia; Minguzzi, Elena; Zedde, Marialuisa; Nasreldein, Ahmed; Vinciguerra, Luisa; Costa, Luis; Elsayed, Ahmed Elsaid; AlBanna, Mona; Tudisco, Laura; Merlino, Giovanni; Polymeris, Alexandros; De Santis, Federico; Sacco, Simona 分享 收藏
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VPS13C-mediated endoplasmic reticulum-lysosome tethering in neuronal stress responses VPS13C介导的内质网-溶酶体连接在神经元应激反应中的作用 Hamad, Rabab S.; Hamza, Eman; Abdel-Aal, Ebtehal M.; Elmorsy, Elsayed A.; Eissa, Hanan; Farrag, Alshaimaa A.; Shata, Ahmed; Nassar, Ghada M.; Morsy, Nesreen Elsayed; El-Mansy, Ahmed A.; Hamad, Ahmed G.; Abdellatif, Eman R.; Saber, Sameh 分享 收藏
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Lactose-decorated, alginate-coated chitosan nanoparticles loaded with Coomassie Brilliant Blue G-250 protect colonic barrier integrity in experimental colitis 乳糖修饰、海藻酸钠包被的壳聚糖纳米粒子负载考马斯亮蓝G-250可保护实验性结肠炎中的结肠屏障完整性 Amer, Maha M.; Kira, Ahmed Y.; Saber, Sameh; Alsalloom, Abdulaziz A.; Khodeir, Mostafa M.; Elashry, Hala A.; Hamad, Rabab S.; Alhomaidi, Adel; Alsaykhan, Hamad; Alorini, Mohammed; Abdel-Hamed, Mohamed R.; Eltayeb, Huda; Hasan, Tabinda; El-Sayed, Abdelrahman; Elmorsy, Elsayed A. 分享 收藏
Beyond its mucolytic mechanism, carbocisteine protects against cyclophosphamide-induced lung injury by modulating TLR-4/NF-κB signaling, oxidative stress, and PPARγ 除其黏痰溶解机制外,羧甲司坦通过调控TLR-4/NF-κB信号通路、氧化应激和PPARγ来对抗环磷酰胺诱导的肺损伤 Alruhaimi, Reem S.; Hassanein, Emad H. M.; Aldawood, Nouf; Al-Thubiani, Wafa S.; Mahdi, Somya E.; Abd El-Ghafar, Omnia A. M.; Alotaibi, Mohammed F.; Mahmoud, Ayman M. 分享 收藏