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Jan Kihlberg

uppsala university

56H指数
317论文数
1.2W被引数
收录论文 103
发表时间
Docking of virtual libraries identifies small-molecule agonists of neurotensin receptors with analgesic activity虚拟库的对接鉴定出具有镇痛活性的神经tensin受体小分子激动剂
err2026-07-22
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errNicolas Panel; Duy Duc Vo; Harald Hübner; Mattia Deluigi; Szymon Pach; Félix Bélair; Dorothee Weikert; Christoph Klenk; Mark Hilge; Niharika Shiva; Isabelle Brochu; Jean-Michel Longpré; Frida Bällgren; Aljona Saleh; Huabin Hu; Jon Kapla; Stefanie Kampen; Israel Cabeza de Vaca; Jan Kihlberg; Nina Wettschureck; Philippe Sarret; Andreas Plückthun; Peter Gmeiner; Jens Carlsson
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Autoantibodies to Joint-Related Peptides Are Associated with Onset of Rheumatoid Arthritis in Presymptomatic Seronegative Individuals关节相关肽的自体抗体与无症状期类风湿关节炎血清阴性个体的发病相关
err2026-04-17
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errOuti Sareila PhD; Linda Johansson MD, PhD; Anders Lundquist PhD; Monica Leu Agelii PhD; Lei Cheng PhD; Yibo He PhD; Erik Lönnblom PhD; Maria Andersson PhD; Jan Kihlberg PhD; Anders Esberg PhD; Inger Gjertsson MD, PhD; Rikard Holmdahl MD, PhD; Solbritt Rantapää-Dahlqvist MD, PhD
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Ultra-large virtual screening unveils potent agonists of the neuromodulatory orphan receptor GPR139超大规模虚拟筛选揭示了神经调节孤核受体GPR139的强效激动剂
err2025-12-09
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errIsrael Cabeza de Vaca; Boris Trapkov; Ling Shen; Duy Duc Vo; Xiaoqun Zhang; Yunting Yang; Mitra Pezeshki; Xuehan Zhang; Frida Bällgren; Aljona Saleh; Andrii V. Tarnovskiy; Dmytro S. Radchenko; Yurii S. Moroz; Hans Bräuner-Osborne; Per Svenningsson; Jan Kihlberg; Zhi-Jie Liu; Alexander Sebastian Hauser; Jens Carlsson
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Conformational Trajectory of the Molecular Chameleon Grazoprevir from Formulation to Target-Bound
err2025-12-01
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errWieske, Lianne H. E.; Bu, Guanhong; Erdelyi, Mate; Kihlberg, Jan; Gonen, Tamir; Danelius, Emma Rova
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Tolerogenic antigen-specific vaccine induces VISTA-enriched regulatory T cells and protects against arthritis in DRB1∗04:01 mice耐受原特异性疫苗诱导VISTA富集的调节性T细胞,并保护DRB1∗04:01小鼠免受关节炎侵害
err2025-04-24
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errLaura Romero-Castillo; Rajan Kumar Pandey; Bingze Xu; Christian M. Beusch; Ana Oliveira-Coelho; Kejsi Zeqiraj; Carolin Svensson; Zhongwei Xu; Huqiao Luo; Outi Sareila; Pierre Sabatier; Changrong Ge; Lei Cheng; Vilma Urbonaviciute; Alexander Krämer; Cecilia Lindgren; Sabrina Haag; Johan Viljanen; Roman A. Zubarev; Jan Kihlberg; Anna Linusson; Harald Burkhardt; Rikard Holmdahl
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Impact of Linker Composition on VHL PROTAC Cell Permeability接头组成对VHL PROTAC细胞通透性的影响
err2024-12-18
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errAbeje, Yordanos Esubalew; Wieske, Lianne H. E.; Poongavanam, Vasanthanathan; Maassen, Stefanie; Atilaw, Yoseph; Cromm, Philipp; Lehmann, Lutz; Erdelyi, Mate; Meibom, Daniel; Kihlberg, Jan
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Discovery of a Series of Macrocycles as Potent Inhibitors of Leishmania Infantum
err2024-10-08
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errRiu, Federico; Ruppitsch, Larissa Alena; Vo, Duc Duy; Hong, Richard S.; Tyagi, Mohit; Matheeussen, An; Hendrickx, Sarah; Poongavanam, Vasanthanathan; Caljon, Guy; Sheikh, Ahmad Y.; Sjo, Peter; Kihlberg, Jan
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Beware of extreme calculated lipophilicity when designing cyclic peptides
err2024-09-19
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PREAI
errPoongavanam, Vasanthanathan; Vo, Duc Duy; Kihlberg, Jan
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Exploring the chemical space of orally bioavailable PROTACs
err2024-04-01
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errApprato, Giulia; Poongavanam, Vasanthanathan; Jimenez, Diego Garcia; Atilaw, Yoseph; Erdelyi, Mate; Ermondi, Giuseppe; Caron, Giulia; Kihlberg, Jan
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Molecular chameleons in drug discovery药物发现中的分子变色龙
err2023-12-20
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PREAI
errPoongavanam, Vasanthanathan; Wieske, Lianne H. E.; Peintner, Stefan; Erdelyi, Mate; Kihlberg, Jan
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Antigen-presenting autoreactive B cells activate regulatory T cells and suppress autoimmune arthritis in mice ( vol 220 , e20230101 , 2023)
err2023-10-03
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errAoun, Mike; Coelho, Ana; Kramer, Alexander; Saxena, Amit; Sabatier, Pierre; Beusch, Christian Michel; Lonnblom, Erik; Geng, Manman; Do, Nhu-Nguyen; Xu, Zhongwei; Zhang, Jingdian; He, Yibo; Castillo, Laura Romero; Abolhassani, Hassan; Xu, Bingze; Viljanen, Johan; Rorbach, Joanna; Lahore, Gonzalo Fernandez; Gjertsson, Inger; Kastbom, Alf; Sjowall, Christopher; Kihlberg, Jan; Zubarev, Roman A.; Burkhardt, Harald; Holmdahl, Rikard
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Antigen-presenting autoreactive B cells activate regulatory T cells and suppress autoimmune arthritis in mice
err2023-09-11
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errAoun, Mike; Coelho, Ana; Kramer, Alexander; Saxena, Amit; Sabatier, Pierre; Beusch, Christian Michel; Lonnblom, Erik; Geng, Manman; Do, Nhu-Nguyen; Xu, Zhongwei; Zhang, Jingdian; He, Yibo; Romero Castillo, Laura; Abolhassani, Hassan; Xu, Bingze; Viljanen, Johan; Rorbach, Joanna; Fernandez Lahore, Gonzalo; Gjertsson, Inger; Kastbom, Alf; Sjowall, Christopher; Kihlberg, Jan; Zubarev, Roman A.; Burkhardt, Harald; Holmdahl, Rikard
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Structure-based virtual screening discovers potent and selective adenosine A1 receptor antagonists
err2023-09-01
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errMatricon, Pierre; Nguyen, Anh T. N.; Vo, Duc Duy; Baltos, Jo-Anne; Jaiteh, Mariama; Luttens, Andreas; Kampen, Stefanie; Christopoulos, Arthur; Kihlberg, Jan; May, Lauren Therese; Carlsson, Jens
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Therapy targeting antigen-specific T cells by a peptide-based tolerizing vaccine against autoimmune arthritis通过针对自身免疫性关节炎的基于肽的耐受疫苗靶向抗原特异性T细胞的治疗
err2023-06-12
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errOAAI
errUrbonaviciute, Vilma; Romero-Castillo, Laura; Xu, Bingze; Luo, Huqiao; Schneider, Nadine; Weisse, Sylvia; Do, Nhu-Nguyen; Oliveira-Coelho, Ana; Lahore, Gonzalo Fernandez; Li, Taotao; Sabatier, Pierre; Beusch, Christian M.; Viljanen, Johan; Zubarev, Roman A.; Kihlberg, Jan; Baecklund, Johan; Burkhardt, Harald; Holmdahl, Rikard
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Autoantibodies to Disease-Related Proteins in Joints as Novel Biomarkers for the Diagnosis of Rheumatoid Arthritis
err2023-04-27
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errLonnblom, Erik; Leu Agelii, Monica; Sareila, Outi; Cheng, Lei; Xu, Bingze; Viljanen, Johan; Hafstrom, Ingiald; Andersson, Maria L. E.; Bergstrom, Goran; Ekwall, Anna-Karin Hultgard; Rudin, Anna; Kastbom, Alf; Sjowall, Christopher; Jacobsson, Lennart T. H.; Kihlberg, Jan; Gjertsson, Inger; Holmdahl, Rikard
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Predictive Modeling of PROTAC Cell Permeability with Machine Learning
err2023-02-01
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errPoongavanam, Vasanthanathan; Koelling, Florian; Giese, Anja; Goeller, Andreas H.; Lehmann, Lutz; Meibom, Daniel; Kihlberg, Jan
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Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction (vol 65, pg 2204, 2022)
err2023-01-26
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errBegnini, Fabio; Geschwindner, Stefan; Johansson, Patrik; Wissler, Lisa; Lewis, Richard J.; Danelius, Emma; Luttens, Andreas; Matricon, Pierre; Carlsson, Jens; Lenders, Stijn; Koenig, Beate; Friedel, Anna; Sjoe, Peter; Schiesser, Stefan; Kihlberg, Jan
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