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收藏Python-derived 16α-Hydroxylated Bile Acid, Pythocholic Acid is a ligand for TGR5, not farnesoid X receptors and vitamin D receptors由Python衍生而来的16α-羟基化胆汁酸,Pythocholic Acid是TGR5的配体,而非法尼醇X受体和维生素D受体。
Kiaei, Nicole; Malik, Afsin; Idahosa, Sydney O.; Lee, Kevin K.; Endo-Umeda, Kaori; Makishima, Makoto; Kawamura, Akira; Higuchi, Sei
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收藏Transcriptional coregulator Ess2 controls survival of post-thymic CD4+ T cells through the Myc and IL-7 signaling pathways
Takada, Ichiro; Hidano, Shinya; Takahashi, Sayuri; Yanaka, Kaori; Ogawa, Hidesato; Tsuchiya, Megumi; Yokoyama, Atsushi; Sato, Shingo; Ochi, Hiroki; Nakagawa, Tohru; Kobayashi, Takashi; Nakagawa, Shinichi; Makishima, Makoto
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收藏Myeloid LXR (Liver X Receptor) Deficiency Induces Inflammatory Gene Expression in Foamy Macrophages and Accelerates Atherosclerosis
Endo-Umeda, Kaori; Kim, Eunyoung; Thomas, David G.; Liu, Wenli; Dou, Huijuan; Yalcinkaya, Mustafa; Abramowicz, Sandra; Xiao, Tong; Antonson, Per; Gustafsson, Jan-Ake; Makishima, Makoto; Reilly, Muredach P.; Wang, Nan; Tall, Alan R.
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收藏A deficiency of Dec2 triggers periodontal inflammation and pyroptosis
Oka, Shunichi; Li, Xiaoyan; Sato, Fuyuki; Zhang, Fengzhu; Tewari, Nitesh; Kim, Il-Shin; Zhong, Liangjun; Hamada, Nobushiro; Makishima, Makoto; Liu, Yi; Bhawal, Ujjal K.
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收藏Convenient Retinoid X Receptor Binding Assay Based on Fluorescence Change of the Antagonist NEt-C343
Yukawa-Takamatsu, Kayo; Wang, Yifei; Watanabe, Masaki; Takamura, Yuta; Fujihara, Michiko; Nakamura-Nakayama, Mariko; Yamada, Shoya; Kikuzawa, Shota; Makishima, Makoto; Kawasaki, Mayu; Ito, Sohei; Nakano, Shogo; Kakuta, Hiroki
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收藏Discovery of a Gatekeeper Antagonist that Blocks Entry Pathway to Retinoid X Receptors (RXRs) without Allosteric Ligand Inhibition in Permissive RXR Heterodimers
Watanabe, Masaki; Fujihara, Michiko; Motoyama, Tomoharu; Kawasaki, Mayu; Yamada, Shoya; Takamura, Yuta; Ito, Sohei; Makishima, Makoto; Nakano, Shogo; Kakuta, Hiroki
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收藏Dec2 attenuates autophagy in inflamed periodontal tissues
Oka, Shunichi; Li, Xiaoyan; Sato, Fuyuki; Zhang, Fengzhu; Tewari, Nitesh; Chen, Chongchong; Zhong, Liangjun; Makishima, Makoto; Liu, Yi; Bhawal, Ujjal K.
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收藏Development of Selective TGR5 Ligands Based on the 5,6,7,8-Tetrahydro-5,5,8,8-tetramethylnaphthalene Skeleton基于5,6,7,8-四氢-5,5,8,8-四甲基萘骨架的选择性TGR5配体的开发
Terui, Ryusei; Yanase, Yuta; Yokoo, Hidetomo; Suhara, Yoshitomo; Makishima, Makoto; Demizu, Yosuke; Misawa, Takashi
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