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收藏Structure-based design and optimization lead to the identification of novel dihydrothiopyrano [3,2-d]pyrimidine derivatives as potent HIV-1 inhibitors against drug-resistant variants基于结构的设计和优化导致鉴定新型二氢噻喃 [3,2-d] 嘧啶衍生物作为抗耐药变体的有效HIV-1抑制剂
Wang, Zhao; Zhang, Heng; Gao, Zhen; Sang, Zihao; De Clercq, Erik; Pannecouque, Christophe; Kang, Dongwei; Zhan, Peng; Liu, Xinyong
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收藏Identification of Ebselen derivatives as novel SARS-CoV-2 main protease inhibitors: Design, synthesis, biological evaluation, and structure-activity relationships exploration
Zhang, Heng; Li, Jing; Toth, Karoly; Tollefson, Ann E.; Jing, Lanlan; Gao, Shenghua; Liu, Xinyong; Zhan, Peng
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收藏Structure-Based Optimization of 2,4,5-Trisubstituted Pyrimidines as Potent HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: Exploiting the Tolerant Regions of the Non-Nucleoside Reverse Transcriptase Inhibitors' Binding Pocket
Zhao, Fabao; Zhang, Heng; Xie, Minghui; Meng, Bairu; Liu, Na; Dun, Caiyun; Qin, Yanyang; Gao, Shenghua; De Clercq, Erik; Pannecouque, Christophe; Tang, Ya-Jie; Zhan, Peng; Liu, Xinyong; Kang, Dongwei
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收藏An interpretable machine learning model based on a quick pre-screening system enables accurate deterioration risk prediction for COVID-19
Jia, Lijing; Wei, Zijian; Zhang, Heng; Wang, Jiaming; Jia, Ruiqi; Zhou, Manhong; Li, Xueyan; Zhang, Hankun; Chen, Xuedong; Yu, Zheyuan; Wang, Zhaohong; Li, Xiucheng; Li, Tingting; Liu, Xiangge; Liu, Pei; Chen, Wei; Li, Jing; He, Kunlun
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收藏A cohort autopsy study defines COVID-19 systemic pathogenesis
Yao, Xiao-Hong; Luo, Tao; Shi, Yu; He, Zhi-Cheng; Tang, Rui; Zhang, Pei-Pei; Cai, Jun; Zhou, Xiang-Dong; Jiang, Dong-Po; Fei, Xiao-Chun; Huang, Xue-Quan; Zhao, Lei; Zhang, Heng; Wu, Hai-Bo; Ren, Yong; Liu, Zhen-Hua; Zhang, Hua-Rong; Chen, Cong; Fu, Wen-Juan; Li, Heng; Xia, Xin-Yi; Chen, Rong; Wang, Yan; Liu, Xin-Dong; Yin, Chang-Lin; Yan, Ze-Xuan; Wang, Juan; Jing, Rui; Li, Tai-Sheng; Li, Wei-Qin; Wang, Chao-Fu; Ding, Yan-Qing; Mao, Qing; Zhang, Ding-Yu; Zhang, Shu-Yang; Ping, Yi-Fang; Bian, Xiu-Wu
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