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收藏Targeting mTORC2-Dependent AKT/FOXO1/RNF125 signaling exploits a therapeutic vulnerability in c-MET-activated and β-catenin-mutated hepatocellular carcinoma靶向mTORC2依赖性AKT/FOXO1/RNF125信号通路利用了c-MET激活和β-catenin突变的肝细胞癌的治疗易损性
Wang, Xue; Zhou, Yi; Zhang, Shu; Farrar, Christine; Xie, Xuemei; Li, Jiaheng; Zhang, Sophia M.; Zhang, Zheng; Yonemura, Andrew; Haynes, Jonathan Toshio; Feng, Xuping; Shang, Runze; Xu, Zhong; Wu, Yanhui; Qiao, Yu; Cui, Guofei; Liao, Weiting; Li, Rong; Calvisi, Diego F.; Zhang, Shuxing; Xu, Meng; Chen, Xin; Wang, Haichuan
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收藏Uncoupling Metastasis and Epithelial-to-Mesenchymal Transition in sgP19/kRAS-Driven Spontaneous Metastatic Liver Tumor Model解耦sgP19/kRAS驱动的自发性转移性肝癌模型中的转移与上皮-间质转化
Wang, Jingwen; Xu, Zijing; Xu, Lei; Wang, Lishan; Geng, Jiahao; Wang, Xue; Xu, Meng; Superville, Daphne; Reeves, Melissa; Evert, Matthias; Calvisi, Diego F.; Chen, Xin; Song, Xinhua
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收藏Glutamine synthetase loss in β-catenin-mutant hepatocellular carcinoma promotes tumor burden through macrophage metabolic reprogramming
Delgado, Evan R.; Patel, Panari; Tao, Junyan; Krutsenko, Yekaterina; Liu, Silvia; Green, Daniel; Alzubali, Raghad; Lehrich, Brandon M.; Liu, Jai-Jun; Yasaka, Tyler; Poddar, Minakshi; Singh, Sucha; Meadows, Vik; Bell, Aaron W.; Chen, Xin; Singhi, Aatur; Monga, Satdarshan P.
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收藏Design, synthesis and biological evaluation of 3-amino-6-(2-hydroxy-phenyl)pyridazin-4-aryl derivatives as SMARCA2/4 degraders3-氨基-6-(2-羟基-苯基)吡啶azin-4-芳基衍生物的设计、合成及生物评价:作为SMARCA2/4降解剂
Yang, Tianqiong; Wei, Wei; Zhang, Qi; Chen, Xin; Xu, Kaiyan; Su, Xingping; Yue, Lin; Gao, Jiuyu; Wang, Ningyu; Cao, Yu; Yu, Luoting
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收藏PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models (vol 67, pg 1262, 2024)PROTACs靶向BRM(SMARCA2)可在体内实现对BRG1(SMARCA4)的选择性降解,并在BRG1突变异种移植肿瘤模型中表现出活性(vol 67, pg 1262, 2024)
Berlin, Michael; Cantley, Jennifer; Bookbinder, Mark; Bortolon, Elizabeth; Broccatelli, Fabio; Cadelina, Greg; Chan, Emily W.; Chen, Huifen; Chen, Xin; Cheng, Yunxing; Cheung, Tommy K.; Crew, Andrew P.; Davenport, Kim; Dinicola, Dean; Dong, Hanqing; Gordon, Debbie; Hamman, Brian D.; Harbin, Alicia; Haskell, Roy; He, Mingtao; Hole, Alison J.; Januario, Thomas; Kerry, Philip S.; Koenig, Stefan G.; Li, Limei; Merchant, Mark; Perez-Dorado, Inmaculada; Pizzano, Jennifer; Quinn, Connor; Rose, Christopher M.; Rousseau, Emma; Snyder, Lawrence B.; Soto, Leofal; Staben, Leanna R.; Sun, Hongming; Tian, Qingping; Wang, Gan; Wang, Jing; Wang, Weifeng; Ye, Crystal S.; Ye, Xiaofen; Zhang, Penghong; Zhou, Yuhui; Yauch, Robert; Dragovich, Peter S.
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收藏A conceptual exploration on the synergistic anti-tumor effects of high-order combination of OHSV2-DSTEFAP5/CD3, CAR-T cells, and immunotoxins in hepatocellular carcinoma关于HSV2-DSTEFAP5/CD3、CAR-T细胞和免疫毒素高级联合方案协同抗肿瘤效应的概念性探索:在肝细胞癌中的应用
Dong, Shuang; Chen, Xin; Li, Xiaoyu; Wang, Yang; Huang, Qing; Li, Yuanxiang; Jin, Jing; Zhu, Xianmin; Zhong, Yi; Cai, Qian; Xue, Chang; Guo, Fang; Huang, Le; Liu, Binlei
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