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H

Helge Prinz

university of munster

H指数:24

被引数:1,693

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Targeting Human Protein Kinase CK2 by a Library of Indeno[1,2-b]Indoles: Contribution of Thermal Shift Assay to Pre-Screening and Co-Crystallization to Post-Screening

靶向人蛋白激酶CK2的 inden o[1,2-<i>b</i>]吲哚文库：热迁移分析对预筛选的贡献和共晶化对后筛选的贡献

Archiv der Pharmazie

IF3.6

2026-09-070

OAAI

Small molecule-induced degradation of the full length and V7 truncated variant forms of human androgen receptor

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2018-09-0116

PREAI

Oxadiazole-substituted naphtho[2,3-b]thiophene-4,9-diones as potent inhibitors of keratinocyte hyperproliferation. Structure-activity relationships of the tricyclic quinone skeleton and the oxadiazole substituent

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2017-07-0112

PREAI

N-Heterocyclic (4-Phenylpiperazin-1-yl)methanones Derived from Phenoxazine and Phenothiazine as Highly Potent Inhibitors of Tubulin Polymerization

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2017-01-1332

PREAI

8-Halo-substituted naphtho[2,3-b]thiophene-4,9-diones as redox-active inhibitors of keratinocyte hyperproliferation with reduced membrane-damaging properties

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2016-03-0113

PREAI

Inhibitory effect of phenothiazine- and phenoxazine-derived chloroacetamides on Leishmania major growth and Trypanosoma brucei trypanothione reductase

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2016-01-0121

PREAI

Synthesis and Structure-Activity Relationships of Lapacho Analogues. 2. Modification of the Basic Naphtho[2,3-b]furan-4,9-dione, Redox Activation, and Suppression of Human Keratinocyte Hyperproliferation by 8-Hydroxynaphtho[2,3-b]thiophene-4,9-diones

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2014-07-0740

PREAI

Characterization of a New Class of Androgen Receptor Antagonists with Potential Therapeutic Application in Advanced Prostate Cancer

MOLECULAR CANCER THERAPEUTICS

IF5.5

2013-11-0627

OA

Natural Product Derived Antiprotozoal Agents: Synthesis, Biological Evaluation, and Structure-Activity Relationships of Novel Chromene and Chromane Derivatives

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2013-09-0954

PREAI

Synthesis and Structure-Activity Relationships of Lapacho Analogues. 1. Suppression of Human Keratinocyte Hyperproliferation by 2-Substituted Naphtho[2,3-b]furan-4,9-diones, Activation by Enzymatic One- and Two-Electron Reduction, and Intracellular Generation of Superoxide

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2012-08-0780

PREAI

Phenylimino-10H-anthracen-9-ones as novel antimicrotubule agents-synthesis, antiproliferative activity and inhibition of tubulin polymerization

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2011-07-0121

PRE

N-Benzoylated Phenoxazines and Phenothiazines: Synthesis, Antiproliferative Activity, and Inhibition of Tubulin Polymerization

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2011-05-2664

PRE

Synthesis and biological evaluation of novel 10-benzyl-substituted 4,5-dichloro-10H-anthracen-9-ones as inhibitors of keratinocyte hyperproliferation

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2010-11-019

PREAI

Structure-activity relationship studies of acridones as potential antipsoriatic agents. 2. Synthesis and antiproliferative activity of 10-substituted hydroxy-10H-acridin-9-ones against human keratinocyte growth

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2010-11-0121

PREAI

Synthesis, antiproliferative activity and inhibition of tubulin polymerization by anthracenone-based oxime derivatives

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2010-08-0122

PREAI

Structure-activity relationship studies of acridones as potential antipsoriatic agents. 1. Synthesis and antiproliferative activity of simple N-unsubstituted 10H-acridin-9-ones against human keratinocyte growth

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2010-08-0133

PREAI

Synthesis, antiproliferative activity and inhibition of tubulin polymerization by 1,5-and 1,8-disubstituted 10H-anthracen-9-ones bearing a 10-benzylidene or 10-(2-oxo-2-phenylethylidene) moiety

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2010-08-0122

PREAI

Synthesis of 2,6-Aceanthrylenedione, a Cyclic Vinylog of Anthraquinone

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2010-05-113

PREAI

10-(2-oxo-2-Phenylethylidene)-10H-anthracen-9-ones as Highly Active Antimicrotubule Agents: Synthesis, Antiproliferative Activity, and Inhibition of Tubulin Polymerization

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2009-02-1628

PREAI

9-benzylidene-naphtho[2,3-b]thiophen-4-ones and benzylidene-9(10H)-anthracenones as novel tubulin interacting agents with high apoptosis-inducing activity

EUROPEAN JOURNAL OF PHARMACOLOGY

IF4.7

2007-12-0118

PREAI