未登录 An Imidazo[2,1-b][1,3,4]thiadiazole Derivative Inhibits the Virulence Factor α-Hemolysin by Blocking the Pullout of Its Stem Domain 咪唑并[2,1-b][1,3,4]噻二唑衍生物通过阻断其茎状域的拉出作用抑制毒力因子α-溶血素 Korotkov, Vadim S.; Lukat, Peer; Di Lucrezia, Raffaella; Shekhar, Aditya; Degenhart, Carsten; Diestel, Randi; Bilitewski, Ursula; Dinkel, Klaus; Blankenfeldt, Wulf; Bronstrup, Mark 分享 收藏
分享 收藏
分享 收藏
Synthesis and Microbiological Activities of 3-Nitropyrazolo-[1,5-d][1,2,4]triazin-7(6H)-ones and Derivatives Zapol’skii, V.A.; Munoz Castillo, D.C.; Pawletta, B.; Bilitewski, U.; Gjikaj, M.; Brüdigam, C.; Kaufmann, D.E. 3-硝基吡唑并[1,5-d][1,2,4]三嗪-7(6H)-酮及其衍生物的合成与微生物活性研究。Molecules 2025, 30, 3792. [Google Scholar] [CrossRef] Zapol'skii, Viktor A.; Munoz Castillo, Diana C.; Pawletta, Brigitte; Bilitewski, Ursula; Gjikaj, Mimoza; Brudigam, Christoff; Kaufmann, Dieter E. 分享 收藏
分享 收藏
Newly identified properties of known pharmaceuticals and myxobacterial small molecules revealed by screening for autophagy modulators 通过筛选自噬调节剂所揭示的已知药物和黏细菌小分子的新特性 Fichtner, Janine; Beer, Yan Yan; Ramm, H. G. Mauricio; Muhlen, Sabrina; Surup, Frank; Herrmann, Jennifer; Meister, Toni Luise; Pfaender, Stephanie; Bilitewski, Ursula; Bronstrup, Mark; Mueller, Rolf; Wirth, Manfred; Eskelinen, Eeva-Liisa; Schmitz, Ingo 分享 收藏
Highly potent quinoxalinediones inhibit a-hemolysin and ameliorate Staphylococcus aureus lung infections 高活性的喹喔啉二酮类化合物能够抑制α-溶血素并改善金黄色葡萄球菌肺部感染 Shekhar, Aditya; Di Lucrezia, Raffaella; Jerye, Karoline; Korotkov, Vadim S.; Harmrolfs, Kirsten; Rox, Katharina; Weich, Herbert A.; Ghai, Ishan; Delhommel, Florent; Becher, Isabelle; Degenhart, Carsten; Fansa, Eyad; Unger, Anke; Habenberger, Peter; Klebl, Bert; Lukat, Peer; Schmelz, Stefan; Henke, Steffi; Borgert, Sebastian; Lang, Julia C.; Sasse, Florenz; Diestel, Randi; Richter, Clementine; Schneider-Daum, Nicole; Hinkelmann, Bettina; Niemz, Jana; Lehr, Claus-Michael; Jaensch, Lothar; Huehn, Jochen; Alm, Richard; Savitski, Mikhail; Welte, Tobias; Hesterkamp, Thomas; Sattler, Michael; Winterhalter, Mathias; Blankenfeldt, Wulf; Medina, Eva; Bilitewski, Ursula; Dinkel, Klaus; Broenstrup, Mark 分享 收藏
分享 收藏
分享 收藏
Total Synthesis of Tosyl-Samroiyotmycin A and Its Biological Profiling Kolb, Benedikt; Schmid, Fabian; Weng, Jessica; Altevogt, Luca; Rebelo, Ruben Pereira; Wank, Bianca; Baro, Angelika; Zens, Anna; Shekhar, Aditya; Bilitewski, Ursula; Sax, Sibylle; Wittlin, Sergio; Taylor, Dale; Muller, Rudolf; Laschat, Sabine 分享 收藏
Repurposing screen identifies novel candidates for broad-spectrum coronavirus antivirals and druggable host targets 重新利用屏幕确定了广谱冠状病毒抗病毒药物和可药物宿主目标的新候选药物 Haid, Sibylle; Matthaei, Alina; Winkler, Melina; Sake, Svenja M.; Gunesch, Antonia P.; Milke, Vanessa; Koehler, Natalie M.; Rueckert, Jessica; Vieyres, Gabrielle; Kuehl, David; Nguyen, Tu-Trinh; Goehl, Matthias; Lasswitz, Lisa; Zapatero-Belinchon, Francisco J.; Brogden, Graham; Gerold, Gisa; Wiegmann, Bettina; Bilitewski, Ursula; Brown, Richard J. P.; Broenstrup, Mark; Schulz, Thomas F.; Pietschmann, Thomas 分享 收藏
分享 收藏
Selective killing of the human gastric pathogen Helicobacter pylori by mitochondrial respiratory complex I inhibitors Lettl, Clara; Schindele, Franziska; Mehdipour, Ahmad Reza; Steiner, Thomas; Ring, Diana; Brack-Werner, Ruth; Stecher, Baerbel; Eisenreich, Wolfgang; Bilitewski, Ursula; Hummer, Gerhard; Witschel, Matthias; Fischer, Wolfgang; Haas, Rainer 分享 收藏
分享 收藏
Identification of Antimotilins, Novel Inhibitors of Helicobacter pylori Flagellar Motility That Inhibit Stomach Colonization in a Mouse Model (vol 13, e03755-21, 2022) Suerbaum, Sebastian; Coombs, Nina; Patel, Lubna; Pscheniza, Dimitri; Rox, Katharina; Falk, Christine; Gruber, Achim D.; Kershaw, Olivia; Chhatwal, Patrick; Broenstrup, Mark; Bilitewski, Ursula; Josenhans, Christine 分享 收藏
分享 收藏
Reprogramming of Amino Acid Metabolism Differs between Community-Acquired Pneumonia and Infection-Associated Exacerbation of Chronic Obstructive Pulmonary Disease 氨基酸代谢的重编程在社区获得性肺炎和慢性阻塞性肺疾病感染相关加重之间存在差异 Arshad, Haroon; Siokis, Anastasios; Franke, Raimo; Habib, Aamna; Alfonso, Juan Carlos Lopez; Poliakova, Yuliya; Luecke, Eva; Michaelis, Katina; Broenstrup, Mark; Meyer-Hermann, Michael; Bilitewski, Ursula; Vila, Jordi; Abel, Laurent; Illig, Thomas; Schreiber, Jens; Pessler, Frank 分享 收藏
Identification of Antimotilins, Novel Inhibitors of Helicobacter pylori Flagellar Motility That Inhibit Stomach Colonization in a Mouse Model 在小鼠模型中抑制胃定植的抗幽门螺杆菌鞭毛运动的新型抑制剂antimatilins的鉴定 Suerbaum, Sebastian; Coombs, Nina; Patel, Lubna; Pscheniza, Dimitri; Rox, Katharina; Falk, Christine; Gruber, Achim D.; Kershaw, Olivia; Chhatwal, Patrick; Broenstrup, Mark; Bilitewski, Ursula; Josenhans, Christine 分享 收藏
Peptide microarrays coupled to machine learning reveal individual epitopes from human antibody responses with neutralizing capabilities against SARS-CoV-2 Hotop, Sven-Kevin; Reimering, Susanne; Shekhar, Aditya; Asgari, Ehsaneddin; Beutling, Ulrike; Dahlke, Christine; Fathi, Anahita; Khan, Fawad; Luetgehetmann, Marc; Ballmann, Rico; Gerstner, Andreas; Tegge, Werner; Cicin-Sain, Luka; Bilitewski, Ursula; McHardy, Alice C.; Broenstrup, Mark 分享 收藏
Dual Agents: Fungal Macrocidins and Synthetic Analogues with Herbicidal and Antibiofilm Activities Treiber, Laura; Pezolt, Christine; Zeng, Haoxuan; Schrey, Hedda; Jungwirth, Stefan; Shekhar, Aditya; Stadler, Marc; Bilitewski, Ursula; Erb-Brinkmann, Maike; Schobert, Rainer 分享 收藏