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Sustainable Manufacturing of trans-4-Trifluoromethyl-l-proline via Stereochemical Editing: A Combined In Silico and Experimental Approach 通过立体化学编辑可持续制造trans-4-Trifluoromethyl-l-proline: 结合计算机和实验方法 Algera, Russell F.; Allais, Christophe; Cabrera, Pablo J.; Gonzalez-Esguevillas, Maria; Guan, Yanfei; James, Chintelle; Lee, Johnny W.; Massicott, Jeffrey M.; McInturff, Emma L.; Pearson, Robert J.; Risley, Hud; Watson, Rebecca B. 分享 收藏
Synthesis of Nirmatrelvir: Development of a Scalable Cobalt-Catalyzed Cyclopropanation for Manufacture of the Bicyclic [3.1.0]Proline-Building Block Algera, Russell F.; Allais, Christophe; Baldwin, Aaron F.; Busch, Torsten; Colombo, Federica; Colombo, Matteo; Depretz, Christelle; Dumond, Yves Rene; Faria Quintero, Andres R.; Heredia, Maria; Jung, Jorg; Lall, Amrita; Lee, Taegyo; Liu, Yizhou; Mandelli, Stefano; Mantel, Marvin; Morris, Ronald; Mustakis, Jason; Nguyen, Bao; Pearson, Robert; Piper, Jared L.; Ragan, John A.; Ruffin, Brigitte; Talicska, Courtney; Tcyrulnikov, Sergei; Uyeda, Christopher; Weekly, R. Matthew; Zeng, Ming 分享 收藏
Synthesis of Nirmatrelvir: Development of an Efficient, Scalable Process to Generate the Western Fragment Algera, Russell F.; Allais, Christophe; Baldwin, Aaron F.; Becirovic, Husein; Bowles, Paul; Brown, Adam R.; Buske, Jamie M.; Clarke, Hugh J.; Do, Nga M.; Doyle, Kevin; Fifer, Jonathan; Gray, Kaitlyn; Happe, Alan; Hardink, Mark; Hubbell, Aran K.; James, Chintelle; Khadamkar, Hrushikesh P.; Magano, Javier; McInturff, Emma L.; Mustakis, Jason; Ozbuyukkaya, Gizem; Piper, Jared L.; Place, David W.; Ragan, John A.; Rauschenberger, Blake; Reyes, Giselle; Shehadeh, Rawan; Stanchina, Corey; Stanley, Michael; Weekly, R. Matthew; Weinstein, Ethan; Weisenburger, Gerald A.; Wood, Ethan; Yayla, Hatice G.; Yu, Shu 分享 收藏
Synthesis of Nirmatrelvir: Development of Magnesium Sulfate-Mediated Aminolysis for the Manufacture of the Eastern Fragment Algera, Russell F.; Allais, Christophe; Becirovic, Husein; Brown, Adam R.; Chen, Bo; Clarke, Hugh J.; Concannon, Paul E.; Du, Yansheng; Georgian, William; Lee, Johnny W.; Lee, Taegyo; Magano, Javier; Mandry, Carlos Perez; Mehta, Ruchi; Mull, Eric; Pearson, Robert; Peng, Zhihui; Piper, Jared L.; Ragan, John A.; Reyes, Giselle; Shen, Haibo; Ward, Daniel W.; Weekly, R. Matthew; Weisenburger, Gerald A.; Xu, Pengcheng; Yayla, Hatice G.; Zhang, Mengtan 分享 收藏
Synthesis of Nirmatrelvir: Design and Optimization of an Efficient Telescoped Amidation-Dehydration Sequence Algera, Russell F.; Baldwin, Aaron F.; Bowles, Paul; Clarke, Hugh J.; Connor, Christina G.; Cordi, Eric M.; Do, Nga M.; Nicholson, Lindsay D.; Georgian, William; Happe, Alan; Herman, Madeline I.; Hilou, Elaa; James, Chintelle; Johnson, Amber M.; Kalinowski, Maciej; Kulkarni, Samir A.; Launer-Felty, Katherine D.; Lee, Johnny W.; Lee, Taegyo; Lopez, Jorge; Mcinturff, Emma L.; Piper, Jared L.; Place, David W.; Ragan, John A.; Rauschenberger, Blake; Ryder, Katherine; Stanley, Michael; Weisenburger, Gerald A.; Weekly, R. Matthew; Allais, Christophe 分享 收藏
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