Jean‐Luc Galzi - Publications, H-index & Citations

Jean‐Luc Galzi

centre national de la recherche scientifique (cnrs)

38H指数

119论文数

6.5K被引数

收录论文 40

发表时间

DMSO Solubility Assessment for Fragment-Based Screening

MOLECULES

IF4.6

2021-06-28

OAAI

Baybekov, Shamkhal; Marcou, Gilles; Ramos, Pascal; Saurel, Olivier; Galzi, Jean-Luc; Varnek, Alexandre

Discovery of a Locally and Orally Active CXCL12 Neutraligand (LIT-927) with Anti-inflammatory Effect in a Murine Model of Allergic Airway Hypereosinophilia

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2018-08-14

OAAI

Regenass, Pierre; Abboud, Dayana; Daubeuf, Francois; Lehalle, Christine; Gizzi, Patrick; Riche, Stephanie; Hachet-Haas, Muriel; Rohmer, Francois; Gasparik, Vincent; Boeglin, Damien; Haiech, Jacques; Knehans, Tim; Rognan, Didier; Heissler, Denis; Marsol, Claire; Villa, Pascal; Galzi, Jean-Luc; Hibert, Marcel; Frossard, Nelly; Bonnet, Dominique

A strategy to discover decoy chemokine ligands with an anti-inflammatory activity

SCIENTIFIC REPORTS

IF3.9

2015-10-07

OAAI

Abboud, Dayana; Daubeuf, Francois; Quoc Tuan Do; Utard, Valerie; Villa, Pascal; Haiech, Jacques; Bonnet, Dominique; Hibert, Marcel; Bernard, Philippe; Galzi, Jean-Luc; Frossard, Nelly

New Fluorescein Precursors for Live Bacteria Detection

ANALYTICAL CHEMISTRY

IF6.7

2015-08-20

OAAI

Guilini, Celia; Baehr, Corinne; Schaeffer, Etienne; Gizzi, Patrick; Rufi, Frederic; Haiech, Jacques; Weiss, Etienne; Bonnet, Dominique; Galzi, Jean-Luc

Neuropeptide Y receptor mediates activation of ERK1/2 via transactivation of the IGF receptor

CELLULAR SIGNALLING

IF3.7

2015-07-01

OAAI

Lecat, Sandra; Belemnaba, Lazare; Galzi, Jean-Luc; Bucher, Bernard

Discovery and Characterization of an Endogenous CXCR4 Antagonist

CELL REPORTS

IF6.9

2015-05-01

OAAI

Zirafi, Onofrio; Kim, Kyeong-Ae; Staendker, Ludger; Mohr, Katharina B.; Sauter, Daniel; Heigele, Anke; Kluge, Silvia F.; Wiercinska, Eliza; Chudziak, Doreen; Richter, Rudolf; Moepps, Barbara; Gierschik, Peter; Vas, Virag; Geiger, Hartmut; Lamla, Markus; Weil, Tanja; Burster, Timo; Zgraja, Andreas; Daubeuf, Francois; Frossard, Nelly; Hachet-Haas, Muriel; Heunisch, Fabian; Reichetzeder, Christoph; Galzi, Jean-Luc; Perez-Castells, Javier; Canales-Mayordomo, Angeles; Jimenez-Barbero, Jesus; Gimenez-Gallego, Guillermo; Schneider, Marion; Shorter, James; Telenti, Amalio; Hocher, Berthold; Forssmann, Wolf-Georg; Bonig, Halvard; Kirchhoff, Frank; Muench, Jan

A Fluorescent Live Imaging Screening Assay Based on Translocation Criteria Identifies Novel Cytoplasmic Proteins Implicated in G Protein-coupled Receptor Signaling Pathways

MOLECULAR & CELLULAR PROTEOMICS

IF5.5

2015-05-01

OAAI

Lecat, Sandra; Matthes, Hans W. D.; Pepperkok, Rainer; Simpson, Jeremy C.; Galzi, Jean-Luc

Hypoxia differentially regulated CXCR4 and CXCR7 signaling in colon cancer

MOLECULAR CANCER

IF33.9

2014-03-14

OAAI

Romain, Benoit; Hachet-Haas, Muriel; Rohr, Serge; Brigand, Cecile; Galzi, Jean-Luc; Gaub, Marie-Pierre; Pencreach, Erwan; Guenot, Dominique

Quantitative Structure-Property Relationship Modeling: A Valuable Support in High-Throughput Screening Quality Control

ANALYTICAL CHEMISTRY

IF6.7

2014-02-12

OAAI

Ruggiu, Fiorella; Gizzi, Patrick; Galzi, Jean-Luc; Hibert, Marcel; Haiech, Jacques; Baskin, Igor; Horvath, Dragos; Marcou, Gilles; Varnek, Alexandre

Exploration of the Orthosteric/Allosteric Interface in Human M1 Muscarinic Receptors by Bitopic Fluorescent Ligands

MOLECULAR PHARMACOLOGY

IF3

2013-07-01

OAAI

Daval, Sandrine B.; Kellenberger, Esther; Bonnet, Dominique; Utard, Valerie; Galzi, Jean-Luc; Ilien, Brigitte

An Antedrug of the CXCL12 Neutraligand Blocks Experimental Allergic Asthma without Systemic Effect in Mice

JOURNAL OF BIOLOGICAL CHEMISTRY

IF3.9

2013-04-01

OAAI

Daubeuf, Francois; Hachet-Haas, Muriel; Gizzi, Patrick; Gasparik, Vincent; Bonnet, Dominique; Utard, Valerie; Hibert, Marcel; Frossard, Nelly; Galzi, Jean-Luc

Plasma membrane translocation of REDD1 governed by GPCRs contributes to mTORC1 activation

JOURNAL OF CELL SCIENCE

IF3.6

2013-01-01

OAAI

Michel, Gregory; Matthes, Hans W. D.; Hachet-Haas, Muriel; El Baghdadi, Keltouma; de Mey, Jan; Pepperkok, Rainer; Simpson, Jeremy C.; Galzi, Jean-Luc; Lecat, Sandra

Fluorescent Derivatives of AC-42 To Probe Bitopic Orthosteric/Allosteric Binding Mechanisms on Muscarinic M1 Receptors

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2012-02-27

OAAI

Daval, Sandrine B.; Valant, Celine; Bonnet, Dominique; Kellenberger, Esther; Hibert, Marcel; Galzi, Jean-Luc; Ilien, Brigitte

Prodrugs of a CXC Chemokine-12 (CXCL12) Neutraligand Prevent Inflammatory Reactions in an Asthma Model in Vivo CXC Chemokine-12 (CXCL12) 的前药在体内中和预防哮喘模型中的炎症反应

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2011-12-16

OAAI

Gasparik, Vincent; Daubeuf, Francois; Hachet-Haas, Muriel; Rohmer, Francois; Gizzi, Patrick; Haiech, Jacques; Galzi, Jean-Luc; Hibert, Marcel; Bonnet, Dominique; Frossard, Nelly

TRPA1 mediates spinal antinociception induced by acetaminophen and the cannabinoid Δ9-tetrahydrocannabiorcol

NATURE COMMUNICATIONS

IF15.7

2011-11-22

249

OAAI

Andersson, David A.; Gentry, Clive; Alenmyr, Lisa; Killander, Dan; Lewis, Simon E.; Andersson, Anders; Bucher, Bernard; Galzi, Jean-Luc; Sterner, Olov; Bevan, Stuart; Hogestatt, Edward D.; Zygmunt, Peter M.

Contribution of a tyrosine-based motif to cellular trafficking of wild-type and truncated NPY Y1 receptors

CELLULAR SIGNALLING

IF3.7

2011-01-01

OAAI

Lecat, Sandra; Ouedraogo, Moussa; Cherrier, Thomas; Noulet, Fanny; Ronde, Philippe; Glasser, Nicole; Galzi, Jean-Luc; Mely, Yves; Takeda, Kenneth; Bucher, Bernard

Neutralizing endogenous chemokines with small molecules Principles and potential therapeutic applications

PHARMACOLOGY & THERAPEUTICS

IF12.5

2010-04-01

OAAI

Galzi, Jean-Luc; Hachet-Haas, Muriel; Bonnet, Dominique; Daubeuf, Francois; Lecat, Sandra; Hibert, Marcel; Haiech, Jacques; Frossard, Nelly

Identification and pharmacological properties of E339-3D6, the first nonpeptidic apelin receptor agonist

FASEB JOURNAL

IF4.2

2009-12-29

109

OAAI

Iturrioz, Xavier; Alvear-Perez, Rodrigo; De Mota, Nadia; Franchet, Christel; Guillier, Fabrice; Leroux, Vincent; Dabire, Hubert; Le Jouan, Melissande; Chabane, Hadjila; Gerbier, Romain; Bonnet, Dominique; Berdeaux, Alain; Maigret, Bernard; Galzi, Jean-Luc; Hibert, Marcel; Llorens-Cortes, Catherine

Pirenzepine Promotes the Dimerization of Muscarinic M1 Receptors through a Three-step Binding Process

JOURNAL OF BIOLOGICAL CHEMISTRY

IF3.9

2009-07-01

OAAI

Ilien, Brigitte; Glasser, Nicole; Clamme, Jean-Pierre; Didier, Pascal; Piemont, Etienne; Chinnappan, Raja; Daval, Sandrine B.; Galzi, Jean-Luc; Mely, Yves

THE FUNCTIONAL ARCHITECTURE OF THE ACETYLCHOLINE NICOTINIC RECEPTOR EXPLORED BY AFFINITY LABELING AND SITE-DIRECTED MUTAGENESIS

QUARTERLY REVIEWS OF BIOPHYSICS

IF5.3

2009-03-17

181

OAAI

CHANGEUX, JP; GALZI, JL; DEVILLERSTHIERY, A; BERTRAND, D

研究方向