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Michel Bouvier

université de montreal

108H指数
808论文数
4.0W被引数
收录论文 258
发表时间
The structure of the dopamine D3 receptor bound to cariprazine reveals principles for partial agonists with designed pharmacology多巴胺D3受体与卡利拉赞结合的结构揭示了具有设计药理学特性的部分激动剂的原则
err2026-08-28
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errEliane Hadas Yardeni; Dóra Judit Kiss; Julie Sanchez; Keshet Shavit; Dénes Szepesi Kovács; Attila Egyed; Caleb D. Vogt; Supriya A. Gaitonde; Jacqueline Glenn; Meritxell Canals; Michel Bouvier; Amy Hauck Newman; J. Robert Lane; György M. Keserű; Moran Shalev-Benami
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Screening apelin analogues and a small molecule agonist as effective cardiovascular therapeutics against reperfusion injury筛选阿皮林类似物和小分子激动剂作为防治再灌注损伤的有效心血管治疗药物
err2025-12-20
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errAnjalee Wijewardane; Kleinberg X. Fernandez; Anran Zhang; Conrad Fischer; Dineth P. Nagahawatta; Xavier Iturrioz; Charlotte Avet; Bethan L. Heard; Catherine Llorens-Cortes; Gavin Y. Oudit; Michel Bouvier; John C. Vederas
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The impact of secondary site interactions on the binding specificity of bitopic dopamine D2/D3 receptor ligands次级位点相互作用对双拓扑多巴胺D2/D3受体配体结合特异性的影响
err2025-10-20
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errAttila Egyed; Dóra Judit Kiss; Zsófia Pável; Keve Rajna; Supriya A. Gaitonde; Mariam Dubiel; María Isabel Loza; Edina Szűcs; Éva Borbély; Zsófia Hajna; Grzegorz Satala; Márton Vass; Pál Szabó; Katalin Jósvay; Andrzej J. Bojarski; Holger Stark; Zsuzsanna Helyes; Erika Pintér; Michel Bouvier; György M. Keserű
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MRAP2 modifies the signaling and oligomerization state of the melanocortin-4 receptorMRAP2修饰黑皮素-4受体的信号传导和寡聚化状态
err2025-09-25
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errIqra Sohail; Suli-Anne Laurin; Gunnar Kleinau; Vidicha Chunilal; Andrew Morton; Alfonso Brenlla; Zeynep Cansu Uretmen Kagiali; Marie-José Blouin; Javier A. Tello; Annette G. Beck-Sickinger; Martin J. Lohse; Patrick Scheerer; Michel Bouvier; Peter McCormick; Paolo Annibale; Heike Biebermann
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Intracrine FFA4 signaling controls lipolysis at lipid droplets内源性FFA4信号通路控制脂滴中的脂解作用
err2025-08-05
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errShannon L. O’Brien; Emma Tripp; Natasja Barki; Elodie Blondel-Tepaz; Gabrielle Smith; Adam Boufersaoui; Jennie Roberts; Jeremy A. Pike; Joao Correia; Tamara Miljus; Michel Bouvier; Daniel A. Tennant; Brian D. Hudson; Zachary Gerhart-Hines; Graeme Milligan; Thue W. Schwartz; Davide Calebiro
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The cell adhesion molecule CD44 acts as a modulator of 5-HT7 receptor functions
err2024-11-23
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errBorsdorf, Saskia; Zeug, Andre; Wu, Yuxin; Mitroshina, Elena; Vedunova, Maria; Gaitonde, Supriya A.; Bouvier, Michel; Wehr, Michael C.; Labus, Josephine; Ponimaskin, Evgeni
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G protein selectivity profile of GPR56/ADGRG1 and its effect on downstream effectorsGPR56/ADGRG1的g蛋白选择性特征及其对下游效应子的影响
err2024-09-04
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errJallouli, Raida; Moreno-Salinas, Ana L.; Laniel, Andreanne; Holleran, Brian; Avet, Charlotte; Jacob, Joan; Hoang, Trang; Lavoie, Christine; Carmon, Kendra S.; Bouvier, Michel; Leduc, Richard
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Role of the V2R-βarrestin-Gβγ complex in promoting G protein translocation to endosomes
err2024-07-07
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errSokrat, Badr; Nguyen, Anthony H.; Thomsen, Alex R. B.; Huang, Li-Yin; Kobayashi, Hiroyuki; Kahsai, Alem W.; Kim, Jihee; Ho, Bing X.; Ma, Symon; Little, John; Ehrhart, Catherine; Pyne, Ian; Hammond, Emmery; Bouvier, Michel
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Conformation- and activation-based BRET sensors differentially report on GPCR-G protein coupling
err2024-06-18
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errWright, Shane C.; Avet, Charlotte; Gaitonde, Supriya A.; Muneta-Arrate, Itziar; Le Gouill, Christian; Hogue, Mireille; Breton, Billy; Koutsilieri, Stefania; Alarcia, Rebeca Diez; Heroux, Madeleine; Lauschke, Volker M.; Bouvier, Michel
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G protein-specific mechanisms in the serotonin 5-HT2A receptor regulate psychosis-related effects and memory deficits
err2024-05-29
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errKossatz, Elk; Diez-Alarcia, Rebeca; Gaitonde, Supriya A.; Ramon-Duaso, Carla; Stepniewski, Tomasz Maciej; Aranda-Garcia, David; Muneta-Arrate, Itziar; Tepaz, Elodie; Saen-Oon, Suwipa; Soliva, Robert; Shahraki, Aida; Moreira, David; Brea, Jose; Loza, Maria Isabel; de la Torre, Rafael; Kolb, Peter; Bouvier, Michel; Meana, J. Javier; Robledo, Patricia; Selent, Jana
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In Memoriam Professor Philippe Crine: a hero for children with hypophosphatasia
err2024-04-16
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errChretien, Michel; Hoang, Trang; Bouvier, Michel; Marcinkiewicz, Mieczyslaw; Whyte, Michael; Rockman-Greenberg, Cheryl
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Pharmacological fingerprint of antipsychotic drugs at the serotonin 5-HT2A receptor
err2024-04-02
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errGaitonde, Supriya A.; Avet, Charlotte; Revenga, Mario de la Fuente; Blondel-Tepaz, Elodie; Shahraki, Aida; Pastor, Adrian Morales; Talagayev, Valerij; Robledo, Patricia; Kolb, Peter; Selent, Jana; Gonzalez-Maeso, Javier; Bouvier, Michel
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EGFR signaling and pharmacology in oncology revealed with innovative BRET-based biosensors基于BRET的创新生物传感器揭示了肿瘤学中的EGFR信号和药理学
err2024-03-01
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errGross, Florence; Mancini, Arturo; Breton, Billy; Kobayashi, Hiroyuki; Pereira, Pedro Henrique Scarpelli; Le Gouill, Christian; Bouvier, Michel; Schann, Stephan; Leroy, Xavier; Sabbagh, Laurent
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How carvedilol does not activate β2-adrenoceptors卡维地洛如何不激活 β2-肾上腺素受体
err2023-11-30
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errLefkowitz, Robert J.; Rockman, Howard A.; Shim, Paul J.; Liu, Samuel; Ahn, Seungkirl; Pani, Biswaranjan; Rajagopal, Sudarshan; Shenoy, Sudha K.; Bouvier, Michel; Benovic, Jeffrey L.; Liggett, Stephen B.; Ruffolo, Robert R.; Bristow, Michael R.; Packer, Milton
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GLP-1R signaling neighborhoods associate with the susceptibility to adverse drug reactions of incretin mimetics
err2023-10-09
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errWright, Shane C.; Motso, Aikaterini; Koutsilieri, Stefania; Beusch, Christian M.; Sabatier, Pierre; Berghella, Alessandro; Blondel-Tepaz, Elodie; Mangenot, Kimberley; Pittarokoilis, Ioannis; Sismanoglou, Despoina-Christina; Le Gouill, Christian; Olsen, Jesper V.; Zubarev, Roman A.; Lambert, Nevin A.; Hauser, Alexander S.; Bouvier, Michel; Lauschke, Volker M.
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The ubiquitination status of the glucagon receptor determines signal bias
err2023-05-01
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errKaur, Suneet; Sokrat, Badr; Capozzi, Megan E.; El, Kimberley; Bai, Yushi; Jazic, Aeva; Han, Bridgette; Kumar, Kaavya Krishna; D'Alessio, David A.; Campbell, Jonathan E.; Bouvier, Michel; Shenoy, Sudha K.
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