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收藏Discovery and SAR of JTE-151: A Novel RORγ Inhibitor for Clinical Development
Maeba, Takaki; Hirata, Kazuyuki; Kotoku, Masayuki; Seki, Noriyoshi; Maeda, Katsuya; Hirashima, Shintaro; Yamanaka, Hiroshi; Sakai, Takayuki; Obika, Shingo; Hori, Akimi; Hara, Yoshinori; Noji, Satoru; Suwa, Yoshihiro; Yokota, Masahiro; Fujioka, Shingo; Yamaguchi, Takayuki; Katsuda, Yoshiaki; Hata, Takahiro; Miyagawa, Naoki; Arita, Kojo; Nomura, Yukihiro; Taniguchi, Toshio; Asahina, Kota; Aratsu, Yusuke; Naka, Yuichi; Adachi, Tsuyoshi; Nomura, Akihiro; Akai, Shota; Oshida, Shin-ichi; Pai, Sudhakar; Crowe, Paul; Bradley, Erin; Steensma, Ruo; Tao, Haiyan; Fenn, Morgan; Babine, Robert; Li, Xiaolin; Thacher, Scott; Soeta, Takahiro; Ukaji, Yutaka; Shiozaki, Makoto
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收藏A novel CoxNi1-xP/fs-Si self-supporting electrodes manufactured via femtosecond laser for highly efficient hydrogen evolution reaction
Xu, Lishuang; Zhang, Shuai; Huang, Licheng; Yang, Ying; Tao, Haiyan; Zhu, Jianmin; Yang, Chengyu; Li, Shuyang; Jin, Ruibo; Dong, Xiangting
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收藏β-Substituted Alkenyl Heteroarenes as Dipolarophiles in the Cu(I)-atalyzed Asymmetric 1,3-Dipolar Cycloaddition of Azomethine Ylides Empowered by a Dual Activation Strategy: Stereoselectivity and Mechanistic Insight
Chang, Xin; Yang, Yuhong; Shen, Chong; Xue, Kun-Shan; Wang, Zuo-Fei; Cong, Hengjiang; Tao, Hai-Yan; Chung, Lung Wa; Wang, Chun-Jiang
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收藏Discovery of Second Generation RORγ Inhibitors Composed of an Azole Scaffold
Kotoku, Masayuki; Maeba, Takaki; Fujioka, Shingo; Yokota, Masahiro; Seki, Noriyoshi; Ito, Keisuke; Suwa, Yoshihiro; Ikenogami, Taku; Hirata, Kazuyuki; Hase, Yasunori; Katsuda, Yoshiaki; Miyagawa, Naoki; Arita, Kojo; Asahina, Kota; Noguchi, Masato; Nomura, Akihiro; Doi, Satoki; Adachi, Tsuyoshi; Crowe, Paul; Tao, Haiyan; Thacher, Scott; Hashimoto, Hiromasa; Suzuki, Takayoshi; Shiozaki, Makoto
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收藏Ternary crystal structure of human RORγ ligand-binding-domain, an inhibitor and corepressor peptide provides a new insight into corepressor interaction
Noguchi, Masato; Nomura, Akihiro; Doi, Satoki; Yamaguchi, Keishi; Hirata, Kazuyuki; Shiozaki, Makoto; Maeda, Katsuya; Hirashima, Shintaro; Kotoku, Masayuki; Yamaguchi, Takayuki; Katsuda, Yoshiaki; Crowe, Paul; Tao, Haiyan; Thacher, Scott; Adachi, Tsuyoshi
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