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Hai‐Yan Tao

orphagen pharmaceuticals

43H指数
162论文数
4.0K被引数
收录论文 55
发表时间
A potent and selective RORγ inhibitor for the treatment of autoimmune diseases一种强效且选择性的RORγ抑制剂,用于治疗自身免疫性疾病
err2025-12-08
err0
PREAI
errTaku Ikenogami; Masahiro Yokota; Shingo Fujioka; Naoki Ogawa; Masato Noguchi; Akihiro Nomura; Tsuyoshi Adachi; Yoshiaki Katsuda; Kojo Arita; Naoki Miyagawa; Yusuke Aratsu; Kota Asahina; Paul Crowe; Haiyan Tao; Scott Thacher; Makoto Shiozaki
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A Concise and Modular Approach to Generate Novel RORγ Agonists一种简洁且模块化的方法以生成新型RORγ激动剂
err2025-07-18
err0
PREAI
errShunichi Fukuda; Taku Ikenogami; Kazuki Otake; Shohei Miwa; Katsuya Maeda; Tomoya Yamashita; Tasuku Inami; Masahiro Yokota; Yanhui Lu; Akira Suma; Yutaro Hirono; Naoki Ogawa; Teruhiko Inoue; Kazuhito Harada; Keishi Yamaguchi; Shota Akai; Akihiro Nomura; Tsuyoshi Adachi; Tsuyoshi Terawaki; Akane Suzukawa; Mari Kitamoto; Minako Tanimoto; Toru Noguchi; Takahiro Hata; Iichiro Kawahara; Kazuhiko Iwamoto; Kazuma Kondo; Yoshihiro Kitagawa; Yuichi Naka; Paul Crowe; Haiyan Tao; Morgan Fenn; Scott Thacher; Makoto Oba; Makoto Shiozaki
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Synergistic Dual Catalysis in Stereodivergent Synthesis立体发散合成中的协同双重催化
err2024-02-23
err24
PREAI
errWei, Liang; Fu, Cong; Wang, Zuo-Fei; Tao, Hai-Yan; Wang, Chun-Jiang
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Discovery and SAR of JTE-151: A Novel RORγ Inhibitor for Clinical Development
err2024-01-03
err0
PREAI
errMaeba, Takaki; Hirata, Kazuyuki; Kotoku, Masayuki; Seki, Noriyoshi; Maeda, Katsuya; Hirashima, Shintaro; Yamanaka, Hiroshi; Sakai, Takayuki; Obika, Shingo; Hori, Akimi; Hara, Yoshinori; Noji, Satoru; Suwa, Yoshihiro; Yokota, Masahiro; Fujioka, Shingo; Yamaguchi, Takayuki; Katsuda, Yoshiaki; Hata, Takahiro; Miyagawa, Naoki; Arita, Kojo; Nomura, Yukihiro; Taniguchi, Toshio; Asahina, Kota; Aratsu, Yusuke; Naka, Yuichi; Adachi, Tsuyoshi; Nomura, Akihiro; Akai, Shota; Oshida, Shin-ichi; Pai, Sudhakar; Crowe, Paul; Bradley, Erin; Steensma, Ruo; Tao, Haiyan; Fenn, Morgan; Babine, Robert; Li, Xiaolin; Thacher, Scott; Soeta, Takahiro; Ukaji, Yutaka; Shiozaki, Makoto
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A novel CoxNi1-xP/fs-Si self-supporting electrodes manufactured via femtosecond laser for highly efficient hydrogen evolution reaction
err2022-08-01
err10
PREAI
errXu, Lishuang; Zhang, Shuai; Huang, Licheng; Yang, Ying; Tao, Haiyan; Zhu, Jianmin; Yang, Chengyu; Li, Shuyang; Jin, Ruibo; Dong, Xiangting
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A new entry to highly functionalized pyrroles via a cascade reaction of α-amino esters and alkynals
err2020-01-01
err9
PREAI
errWei, Liang; Xu, Shi-Ming; Jia, Ziqi; Tao, Hai-Yan; Wang, Chun-Jiang
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Asymmetric synthesis of quaternary α-trifluoromethyl α-amino acids by Ir-catalyzed allylation followed by kinetic resolution
err2020-01-01
err22
PREAI
errSun, Xi-Shang; Qiu Ou-Yang; Xu, Shi-Ming; Wang, Xing-Heng; Tao, Hai-Yan; Chung, Lung Wa; Wang, Chun-Jiang
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Stereodivergent assembly of tetrahydro-γ-carbolines via synergistic catalytic asymmetric cascade reaction
err2019-12-05
err120
errOAAI
errXu, Shi-Ming; Wei, Liang; Shen, Chong; Xiao, Lu; Tao, Hai-Yan; Wang, Chun-Jiang
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Synergistic catalysis for cascade allylation and 2-aza-cope rearrangement of azomethine ylides
err2019-04-08
err65
errOAAI
errWei, Liang; Zhu, Qiao; Xiao, Lu; Tao, Hai-Yan; Wang, Chun-Jiang
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Discovery of Second Generation RORγ Inhibitors Composed of an Azole Scaffold
err2019-02-18
err26
PREAI
errKotoku, Masayuki; Maeba, Takaki; Fujioka, Shingo; Yokota, Masahiro; Seki, Noriyoshi; Ito, Keisuke; Suwa, Yoshihiro; Ikenogami, Taku; Hirata, Kazuyuki; Hase, Yasunori; Katsuda, Yoshiaki; Miyagawa, Naoki; Arita, Kojo; Asahina, Kota; Noguchi, Masato; Nomura, Akihiro; Doi, Satoki; Adachi, Tsuyoshi; Crowe, Paul; Tao, Haiyan; Thacher, Scott; Hashimoto, Hiromasa; Suzuki, Takayoshi; Shiozaki, Makoto
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Copper(I)-Catalyzed Kinetic Resolution of exo-3-Oxodicyclopentadienes and endo-3-Oxodicyclopentadiene
err2019-02-01
err15
PREAI
errChang, Xin; Sun, Xi-Shang; Che, Chao; Hu, Yuan-Zheng; Tao, Hai-Yan; Wang, Chun-Jiang
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Ternary crystal structure of human RORγ ligand-binding-domain, an inhibitor and corepressor peptide provides a new insight into corepressor interaction
err2018-11-26
err16
errOAAI
errNoguchi, Masato; Nomura, Akihiro; Doi, Satoki; Yamaguchi, Keishi; Hirata, Kazuyuki; Shiozaki, Makoto; Maeda, Katsuya; Hirashima, Shintaro; Kotoku, Masayuki; Yamaguchi, Takayuki; Katsuda, Yoshiaki; Crowe, Paul; Tao, Haiyan; Thacher, Scott; Adachi, Tsuyoshi
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