未登录 Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A Bourahla, Khadidja; Guiheneuf, Solene; Limanton, Emmanuelle; Paquin, Ludovic; Le Guevel, Remy; Charlier, Thierry; Rahmouni, Mustapha; Durieu, Emilie; Lozach, Olivier; Carreaux, Francois; Meijer, Laurent; Bazureau, Jean-Pierre 分享 收藏
Lipid-Based Quaternary Ammonium Sophorolipid Amphiphiles with Antimicrobial and Transfection Activities Delbeke, Elisabeth I. P.; Everaert, Jonas; Lozach, Olivier; Le Gall, Tony; Berchel, Mathieu; Montier, Tristan; Jaffres, Paul-Alain; Rigole, Petra; Coenye, Tom; Brennich, Martha; Baccile, Niki; Roelants, Sophie L. K. W.; Soetaert, Wim; Van Bogaert, Inge N. A.; Van Geem, Kevin M.; Stevens, Christian, V 分享 收藏
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Synthesis and Biological Evaluation of Bolaamphiphilic Sophorolipids Delbeke, Elisabeth I. P.; Everaert, Jonas; Lozach, Olivier; Le Gall, Tony; Berchel, Mathieu; Montier, Tristan; Jaffres, Paul-Alain; Rigole, Petra; Coenye, Tom; Brennich, Martha; Baccile, Niki; Roelants, Sophie L. K. W.; Soetaert, Wim; van Bogaert, Inge N. A.; Van Geem, Kevin M.; Stevens, Christian V. 分享 收藏
Synthesis, biological evaluation and molecular modeling studies of imidazo[1,2-α]pyridines derivatives as protein kinase inhibitors Lawson, Marie; Rodrigo, Jordi; Baratte, Blandine; Robert, Thomas; Delehouze, Claire; Lozach, Olivier; Ruchaud, Sandrine; Bach, Stephane; Brion, Jean-Daniel; Alami, Mouad; Hamze, Abdallah 分享 收藏
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Novel optimization of valmerins (tetrahydropyrido[1,2-a] isoindolones) as potent dual CDK5/GSK3 inhibitors Ouach, Aziz; Boulahjar, Rajaa; Vala, Christine; Bourg, Stephane; Bonnet, Pascal; Guguen-Guillouzo, Christiane; Ravache, Myriam; Le Guevel, Remy; Lozach, Olivier; Lazar, Said; Troin, Yves; Meijer, Laurent; Ruchaud, Sandrine; Akssira, Mohamed; Guillaumet, Gerald; Routier, Sylvain 分享 收藏
Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors Boulahjar, Rajaa; Ouach, Aziz; Bourg, Stephane; Bonnet, Pascal; Lozach, Olivier; Meijer, Laurent; Guguen-Guillouzo, Christiane; Le Guevel, Remy; Lazar, Said; Akssira, Mohamed; Troin, Yves; Guillaumet, Gerald; Routier, Sylvain 分享 收藏
10-lodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A Falke, Hannes; Chaikuad, Apirat; Becker, Anja; Loaec, Nadege; Lozach, Olivier; Abu Jhaisha, Samira; Becker, Walter; Jones, Peter G.; Preu, Lutz; Baumann, Knut; Knapp, Stefan; Meijer, Laurent; Kunick, Conrad 分享 收藏
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Synthesis and optimization of an original V-shaped collection of 4-7-disubstituted Pyrido[3,2-d]pyrimidines as CDK5 and DYRK1A inhibitors Dehbi, Oussama; Tikad, Abdellatif; Bourg, Stephane; Bonnet, Pascal; Lozach, Olivier; Meijer, Laurent; Aadil, Mina; Akssira, Mohammed; Guillaumet, Gerald; Routier, Sylvain 分享 收藏
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Synthesis, Resolution, and Biological Evaluation of Atropisomeric (aR)- and (aS)-16-Methyllamellarins N: Unique Effects of the Axial Chirality on the Selectivity of Protein Kinases Inhibition Yoshida, Kenyu; Itoyama, Ryosuke; Yamahira, Masashi; Tanaka, Junji; Loaec, Nadege; Lozach, Olivier; Durieu, Emilie; Fukuda, Tsutomu; Ishibashi, Fumito; Meijer, Laurent; Iwao, Masatomo 分享 收藏
Natural Aristolactams and Aporphine Alkaloids as Inhibitors of CDK1/Cyclin B and DYRK1A Marti, Guillaume; Eparvier, Veronique; Morleo, Barbara; Le Ven, Jessica; Apel, Cecile; Bodo, Bernard; Amand, Severine; Dumontet, Vincent; Lozach, Olivier; Meijer, Laurent; Gueritte, Francoise; Litaudon, Marc 分享 收藏
Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors Loidreau, Yvonnick; Marchand, Pascal; Dubouilh-Benard, Carole; Nourrisson, Marie-Renee; Duflos, Muriel; Lozach, Olivier; Loaec, Nadege; Meijer, Laurent; Besson, Thierry 分享 收藏
Synthesis and biological evaluation of 2,3-diarylimidazo[1,2-a]pyridines as antileishmanial agents Marhadour, Sophie; Marchand, Pascal; Pagniez, Fabrice; Bazin, Marc-Antoine; Picot, Carine; Lozach, Olivier; Ruchaud, Sandrine; Antoine, Maud; Meijer, Laurent; Rachidi, Najma; Le Pape, Patrice 分享 收藏
Novel Inverse Binding Mode of Indirubin Derivatives Yields Improved Selectivity for DYRK Kinases Myrianthopoulos, Vassilios; Kritsanida, Marina; Gaboriaud-Kolar, Nicolas; Magiatis, Prokopios; Ferandin, Yoan; Durieu, Emilie; Lozach, Olivier; Cappel, Daniel; Soundararajan, Meera; Filippakopoulos, Panagis; Sherman, Woody; Knapp, Stefan; Meijer, Laurent; Mikros, Emmanuel; Skaltsounis, Alexios-Leandros 分享 收藏
Synthesis and biological evaluation of new 5-benzylated 4-oxo-3,4-dihydro-5H-pyridazino[4,5-b]indoles as PI3Kα inhibitors Bruel, Amelie; Loge, Cedric; de Tauzia, Marie-Ludivine; Ravache, Myriam; Le Guevel, Remy; Guillouzo, Christiane; Lohier, Jean-Francois; Santos, Jana Sopkova-de Oliveira; Lozach, Olivier; Meijer, Laurent; Ruchaud, Sandrine; Benedetti, Helene; Robert, Jean-Michel 分享 收藏
Novel Tetrahydropyrido[1,2-a]isoindolone Derivatives (Valmerins): Potent Cyclin-Dependent Kinase/Glycogen Synthase Kinase 3 Inhibitors with Antiproliferative Activities and Antitumor Effects in Human Tumor Xenografts Boulahjar, Rajaa; Ouach, Aziz; Matteo, Chiurato; Bourg, Stephane; Ravache, Myriam; le Guevel, Remy; Marionneau, Severine; Oullier, Thibauld; Lozach, Olivier; Meijer, Laurent; Guguen-Guillouzo, Christiane; Lazar, Said; Akssira, Mohamed; Troin, Yves; Guillaumet, Gerald; Routier, Sylvain 分享 收藏
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