Peter M. Blumberg - Publications, H-index & Citations

Peter M. Blumberg

ben gurion university

82H指数

558论文数

3.0W被引数

收录论文 202

发表时间

Discovery of Dual TRPA1 and TRPV1 Antagonists as Novel Therapeutic Agents for Pain

PHARMACEUTICALS

IF4.8

2024-09-13

OAAI

Do, Nayeon; Zuo, Dongxu; Kim, Miri; Kim, Minseok; Ha, Hee-Jin; Blumberg, Peter M.; Ann, Jihyae; Hwang, Sun Wook; Lee, Jeewoo

Tyrosine phosphorylation of protein kinase Cδ is essential for its apoptotic effect in response to etoposide

MOLECULAR AND CELLULAR BIOLOGY

IF2.7

2023-03-27

199

OAAI

Blass, M; Kronfeld, I; Kazimirsky, G; Blumberg, PM; Brodie, C

Discovery of Benzopyridone-Based Transient Receptor Potential Vanilloid 1 Agonists and Antagonists and the Structural Elucidation of Their Activity Shift

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2021-01-01

PREAI

Thorat, Shivaji A.; Lee, Yoonji; Jung, Aeran; Ann, Jihyae; Ahn, Songyeon; Baek, Jisoo; Zuo, Dongxu; Do, Nayeon; Jeong, Jin Ju; Blumberg, Peter M.; Esch, Timothy E.; Turcios, Noe A.; Pearce, Larry, V; Ha, Hee-Jin; Yoo, Young Dong; Hong, Sunhye; Choi, Sun; Lee, Jeewoo

Discovery of Nonpungent Transient Receptor Potential Vanilloid 1 (TRPV1) Agonist as Strong Topical Analgesic

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2019-11-08

PREAI

Ann, Jihyae; Kim, Ho Shin; Thorat, Shivaji A.; Kim, Hee; Ha, Hee-Jin; Choi, Kwanghyun; Kim, Young-Ho; Kim, Minseok; Hwang, Sun Wook; Pearce, Larry, V; Esch, Timothy E.; Turcios, Noe A.; Blumberg, Peter M.; Lee, Jeewoo

Discovery of dual-acting opioid ligand and TRPV1 antagonists as novel therapeutic agents for pain

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2019-11-01

OAAI

Lee, Hobin; Ahn, Songyeon; Ann, Jihyae; Ha, Heejin; Yoo, Young Dong; Kim, Young Ho; Hwang, Ji-Young; Hur, Kwang-Hyun; Jang, Choon-Gon; Pearce, Larry V.; Esch, Timothy E.; Lewin, Nancy E.; Blumberg, Peter M.; Lee, Jeewoo

Combination of a Rapidly Penetrating Agonist and a Slowly Penetrating Antagonist Affords Agonist Action of Limited Duration at the Cellular Level

BIOMOLECULES & THERAPEUTICS

IF3.2

2019-09-01

OAAI

Pearce, Larry, V; Ann, Jihyae; Blumberg, Peter M.; Lee, Jeewoo

Differential Regulation of Gene Expression in Lung Cancer Cells by Diacyglycerol-Lactones and a Phorbol Ester Via Selective Activation of Protein Kinase C Isozymes

SCIENTIFIC REPORTS

IF3.9

2019-04-15

OAAI

Cooke, Mariana; Casado-Medrano, Victoria; Ann, Jihyae; Lee, Jeewoo; Blumberg, Peter M.; Abba, Martin C.; Kazanietz, Marcelo G.

4-Aminophenyl acetamides and propanamides as potent transient receptor potential vanilloid 1 (TRPV1) ligands

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2018-08-01

PREAI

Kim, Changhoon; Ann, Jihyae; Lee, Sunho; Kim, Eunhye; Choi, Sun; Blumberg, Peter M.; Frank-Foltyn, Robert; Bahrenberg, Gregor; Stockhause, Hannelore; Christoph, Thomas; Lee, Jeewoo

α-Arylidene Diacylglycerol-Lactones (DAG-Lactones) as Selective Ras Guanine-Releasing Protein 3 (RasGRP3) Ligands

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2018-06-03

PREAI

Ann, Jihyae; Czikora, Agnes; Saini, Amandeep S.; Zhou, Xiaoling; Mitchell, Gary A.; Lewin, Nancy E.; Peach, Megan L.; Blumberg, Peter M.; Lee, Jeewoo

Characterization of AJH-836, a diacylglycerol-lactone with selectivity for novel PKC isozymes

JOURNAL OF BIOLOGICAL CHEMISTRY

IF3.9

2018-06-01

OAAI

Cooke, Mariana; Zhou, Xiaoling; Casado-Medrano, Victoria; Lopez-Haber, Cynthia; Baker, Martin J.; Garg, Rachana; Ann, Jihyae; Lee, Jeewoo; Blumberg, Peter M.; Kazanietz, Marcelo G.

The C1 domain of Vav3, a novel potential therapeutic target

CELLULAR SIGNALLING

IF3.7

2017-12-01

OAAI

Kelsey, Jessica S.; Geczy, Tamas; Kaler, Christopher J.; Blumberg, Peter M.

Novel Radiolabeled Vanilloid with Enhanced Specificity for Human Transient Receptor Potential Vanilloid 1 (TRPV1)

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2017-09-21

OAAI

Pearce, Larry V.; Ann, Jihyae; Jung, Aeran; Thorat, Shiyaii A.; Herold, Brienna K. A.; Habtemichael, Amelework D.; Blumberg, Peter M.; Lee, Jeewoo

Synthesis and Evaluation of Dimeric Derivatives of Diacylglycerol-Lactones as Protein Kinase C Ligands

BIOCONJUGATE CHEMISTRY

IF3.9

2017-07-21

OAAI

Ohashi, Nami; Kobayashi, Ryosuke; Nomura, Wataru; Kobayakawa, Takuya; Czikora, Agnes; Herold, Brienna K.; Lewin, Nancy E.; Blumberg, Peter M.; Tamamura, Hirokazu

Characterization by mass spectrometry of protein kinase C substrates differentially phosphorylated in LNCaP cells in response to phorbol ester and bryostatin 1 treatment

CANCER RESEARCH

IF16.6

2017-07-01

PREAI

Kedei, Noemi; Das, Sudipto; Andresson, Thorkell; Blumberg, Peter M.

Understanding the structural requirements of C1 domains for phorbol ester binding, analysis of the atypical C1 domain of STAC2

CANCER RESEARCH

IF16.6

2017-07-01

PREAI

Abramovitz, Adelle; Kedei, Noemi; Blumberg, Peter M.

Analysis of the distinct activities of the C1a and C1b domains of protein kinase C theta

CANCER RESEARCH

IF16.6

2017-07-01

PREAI

Czikora, Agnes; Pany, Satyabrata; You, Youngki; Saini, Amandeep; Kedei, Noemi; Lewin, Nancy E.; Abramovitz, Adelle; Das, Joydip; Blumberg, Peter M.

Exploring the influence of indololactone structure on selectivity for binding to the C1 domains of PKCα, PKCε, and RasGRP

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2017-06-01

OAAI

Elhalem, Eleonora; Gandolfi Donadio, Lucia; Zhou, Xiaoling; Lewin, Nancy E.; Garcia, Lia C.; Lai, Christopher C.; Kelley, James A.; Peach, Megan L.; Blumberg, Peter M.; Comin, Maria J.

t-Butyl pyridine and phenyl C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2017-04-01

OAAI

Lee, Sunho; Kang, Dong Wook; Ryu, HyungChul; Kim, Changhoon; Ann, Jihyae; Lee, Hobin; Kim, Eunhye; Hong, Sunhye; Choi, Sun; Blumberg, Peter M.; Frank-Foltyn, Robert; Bahrenberg, Gregor; Stockhausen, Hannelore; Christoph, Thomas; Lee, Jeewoo

Evaluation of Chromane-Based Bryostatin Analogues Prepared via Hydrogen-Mediated C-C Bond Formation: Potency Does Not Confer Bryostatin-like Biology

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

IF15.6

2016-09-27

OAAI

Ketcham, John M.; Volchkov, Ivan; Chen, Te-Yu; Blumberg, Peter M.; Kedei, Noemi; Lewin, Nancy E.; Krische, Michael J.

Synthesis and Biological Evaluation of Several Bryostatin Analogues Bearing a Diacylglycerol Lactone C-Ring

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2016-08-23

OAAI

Baumann, David O.; McGowan, Kevin M.; Kedei, Noemi; Peach, Megan L.; Blumberg, Peter M.; Keck, Gary E.

研究方向