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收藏JMC14: a novel dual PI3Kδ/CSF1R inhibitor with potent antitumor activity in hematological and solid tumorsJMC14:一种新型的PI3Kδ/CSF1R双靶点抑制剂,在血液肿瘤和实体瘤中表现出显著的抗肿瘤活性
Zhang, X; Sun, P; Wang, Y; Xu, L; Li, HY; Tong, LJ; Tan, C; Ding, J; Yang, CH; Meng, LH
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收藏Mechanism of astragaloside A against lung adenocarcinoma based on network pharmacology combined with molecular dynamics simulation technique基于网络药理学结合分子动力学模拟技术的黄芪甲苷抗肺腺癌作用机制研究
Ding, Jian; Xue, Qian; Guo, Weizhen; Cheng, Gang; Zhang, Lu; Huang, Tantan; Wu, Di; Tong, Jiabing; Yang, Cheng; Gao, Yating; Li, Zegeng
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收藏USP7 V517F mutation as a mechanism of inhibitor resistanceUSP7 V517F突变作为抑制剂耐药的机制
Miao, Yu-Ling; Fan, Fengying; Cheng, Yong-Jun; Jia, Li; Song, Shan-Shan; Huan, Xia-Juan; Bao, Xu-Bin; Ding, Jian; Yu, Xuekui; He, Jin-Xue
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收藏Design, Synthesis and Biological Activity Study of γ-Aminobutyric Acid (GABA) Derivatives Containing Bridged Bicyclic Skeletons as BCAT1 Inhibitors
Luo, Wen; Pan, Zilu; Zhu, Xinyuan; Li, Yan; Li, Yong; Zhang, Yudi; Pan, Jiamin; Ding, Jian; Xie, Hua; Zhao, Guilong
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收藏Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer1,2,3,4-四氢苯并呋喃[2,3-c]吡啶衍生物的设计、合成及药理学评价:作为p21活化激酶4抑制剂用于胰腺癌治疗
Li, Yang; Fang, Yan; Chen, Xiaoyu; Tong, Linjiang; Feng, Fang; Zhou, Qianqian; Chen, Shulun; Ding, Jian; Xie, Hua; Zhang, Ao
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收藏Discovery of a Covalent Inhibitor That Overcame Resistance to Venetoclax in AML Cells Overexpressing BFL-1
Lou, Jianfeng; Zhou, Qianqian; Lyu, Xilin; Cen, Xinyi; Liu, Chen; Yan, Ziqin; Li, Yan; Tang, Haotian; Liu, Qiupei; Ding, Jian; Lu, Ye; Huang, He; Xie, Hua; Zhao, Yujun
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收藏Discovery of a novel BTK inhibitor S-016 and identification of a new strategy for the treatment of lymphomas including BTK inhibitor-resistant lymphomas发现新的BTK抑制剂S-016并确定治疗淋巴瘤 (包括BTK抑制剂耐药淋巴瘤) 的新策略
Song, Pei-ran; Wan, Zhi-peng; Huang, Ge-ge; Song, Zi-lan; Zhang, Tao; Tong, Lin-jiang; Fang, Yan; Tang, Hao-tian; Xue, Yu; Zhan, Zheng-sheng; Feng, Fang; Li, Yan; Shi, Wen-hao; Huang, Yu-qing; Chen, Yi; Duan, Wen-hu; Ding, Jian; Zhang, Ao; Xie, Hua
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收藏A Novel IRAK4 Inhibitor DW18134 Ameliorates Peritonitis and Inflammatory Bowel Disease新型IRAK4抑制剂DW18134改善腹膜炎和炎症性肠病
Huang, Yuqing; Ning, Yi; Chen, Zhiwei; Song, Peiran; Tang, Haotian; Shi, Wenhao; Wan, Zhipeng; Huang, Gege; Liu, Qiupei; Chen, Yun; Zhou, Yu; Li, Yuantong; Zhan, Zhengsheng; Ding, Jian; Duan, Wenhu; Xie, Hua
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