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Veerabahu Shanmugasundaram

Pfizer

27H指数
86论文数
3.1K被引数
收录论文 35
发表时间
Uncovering hidden druggable sites: computational approaches to allosteric and cryptic pocket discovery—from molecular dynamics to AI揭示隐藏的可成药位点:别构和隐匿口袋发现的计算方法——从分子动力学到人工智能
err2026-10-01
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PREAI
errSirish Kaushik Lakkaraju; Olivia Pierce; Ahmet Mentes; Ivy Zhang; John Tokarski; Matthew Chalkley; Jissy Kuriappan; Goutam Mukherjee; Antonio Palmeri; Theresa Johnson; Veerabahu Shanmugasundaram
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Leveraging efficiency metrics for the optimization of CELMoDs™ as cereblon-based molecular glue degraders
err2025-03-01
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PREAI
errJia, Lei; Riggs, Jennifer R.; Weiss, Dahlia R.; Claus, Brian L.; Shanmugasundaram, Veerabahu; Johnson, Stephen R.; Zapf, Christoph W.
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Insights from protein frustration analysis of BRD4-cereblon degrader ternary complexes show separation of strong from weak degraders
err2025-01-01
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PREAI
errYang, Tianyi; Mukhaleva, Elizaveta; Wei, Wenyuan; Weiss, Dahlia; Ma, Ning; Shanmugasundaram, Veerabahu; Vaidehi, Nagarajan
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Asymmetric Dirhodium-Catalyzed Modification of Immunomodulatory Imide Drugs and Their Biological Assessment
err2024-08-23
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errOAAI
errTracy, William F.; Davies, Geraint H. M.; Jia, Lei; Evans, Ethan D.; Sun, Zhenghang; Buenviaje, Jennifer; Khambatta, Gody; Yu, Shan; Shi, Lihong; Shanmugasundaram, Veerabahu; Moreno, Jesus; Cherney, Emily C.; Davies, Huw M. L.
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Identification of Small Molecule Inhibitors and Ligand Directed Degraders of Calcium/Calmodulin Dependent Protein Kinase Kinase 1 and 2 (CaMKK1/2)
err2023-11-27
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PREAI
errChen, Young; Whitefield, Brandon; Nevius, Erin; Hill, Mark; DelRosario, Joselyn; Sinitsyna, Nadia; Shanmugasundaram, Veerabahu; Mukherjee, Debarati; Shi, Lihong; Mayne, Christopher Glenn; Rousseau, Anne-Marie; Bernard, Steffen M.; Buenviaje, Jennifer; Khambatta, Gody; El Samin, Miriam; Wallace, Michael; Nie, Zhe; Sivakumar, Pallavur; Hamann, Lawrence G.; McDonnell, Donald P.; D'Agostino, Laura Akullian
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On Ternary Complex Stability in Protein Degradation: In Silico Molecular Glue Binding Affinity Calculations
err2023-04-10
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PREAI
errWeiss, Dahlia R.; Bortolato, Andrea; Sun, Yongnian; Cai, Xianmei; Lai, Chon; Guo, Sixuan; Shi, Lihong; Shanmugasundaram, Veerabahu
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Epilogue to the Gerald Maggiora Festschrift: a tribute to an exemplary mentor, colleague, collaborator, and innovator
err2022-09-17
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errOAAI
errShanmugasundaram, Veerabahu; Bajorath, Juergen; Christoffersen, Ralph E.; Petke, James D.; Howe, W. Jeffrey; Johnson, Mark A.; Agrafiotis, Dimitris K.; Lee, Pil; Kuhn, Leslie A.; Goodwin, Jay T.; Holloway, M. Katharine; Doman, Thompson N.; Walters, W. Patrick; Schreyer, Suzanne; Medina-Franco, Jose L.; Martinez-Mayorga, Karina; Restifo, Linda L.
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The PROTACtable genome可替代的基因组
err2021-07-20
err143
PREAI
errSchneider, Melanie; Radoux, Chris J.; Hercules, Andrew; Ochoa, David; Dunham, Ian; Zalmas, Lykourgos-Panagiotis; Hessler, Gerhard; Ruf, Sven; Shanmugasundaram, Veerabahu; Hann, Michael M.; Thomas, Pam J.; Queisser, Markus A.; Benowitz, Andrew B.; Brown, Kris; Leach, Andrew R.
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Absence of GP130 cytokine receptor signaling causes extended Stuve-Wiedemann syndrome
err2020-01-08
err37
errOAAI
errChen, Yin-Huai; Grigelioniene, Giedre; Newton, Phillip T.; Gullander, Jacob; Elfving, Maria; Hammarsjo, Anna; Batkovskyte, Dominyka; Alsaif, Hessa S.; Kurdi, Wesam I. Y.; Abdulwahab, Firdous; Shanmugasundaram, Veerabahu; Devey, Luke; Bacrot, Severine; Brodszki, Jana; Huber, Celine; Hamel, Ben; Gisselsson, David; Papadogiannakis, Nikos; Jedrycha, Katarina; Gurtl-Lackner, Barbara; Chagin, Andrei S.; Nishimura, Gen; Aschenbrenner, Dominik; Alkuraya, Fowzan S.; Laurence, Arian; Cormier-Daire, Valerie; Uhlig, Holm H.
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Machine Learning for Prioritization of Thermostabilizing Mutations for G-Protein Coupled Receptors
err2019-12-01
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errOAAI
errMuk, Sanychen; Ghosh, Soumadwip; Achuthan, Srisairam; Chen, Xiaomin; Yao, XiaoJie; Sandhu, Manbir; Griffor, Matthew C.; Fennell, Kimberly F.; Che, Ye; Shanmugasundaram, Veerabahu; Qiu, Xiayang; Tate, Christopher G.; Vaidehi, Nagarajan
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Cyclic Peptide Design Guided by Residual Dipolar Couplings, J-Couplings, and Intramolecular Hydrogen Bond Analysis
err2019-01-03
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PREAI
errFarley, Kathleen A.; Che, Ye; Navarro-Vazquez, Armando; Limberakis, Chris; Anderson, Dennis; Yan, Jiangli; Shapiro, Michael; Shanmugasundaram, Veerabahu; Gil, Roberto R.
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TRPA1 ankyrin repeat six interacts with a small molecule inhibitor chemotype
err2018-11-14
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errOAAI
errTseng, Wei Chou; Pryde, David C.; Yoger, Katrina E.; Padilla, Karen M.; Antonio, Brett M.; Han, Seungil; Shanmugasundaram, Veerabahu; Gerlach, Aaron C.
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Delineating the role of cooperativity in the design of potent PROTACs for BTK
err2018-07-16
err296
errOAAI
errZorba, Adelajda; Chuong Nguyen; Xu, Yingrong; Starr, Jeremy; Borzilleri, Kris; Smith, James; Zhu, Hongyao; Farley, Kathleen A.; Ding, WeiDong; Schiemer, James; Feng, Xidong; Chang, Jeanne S.; Uccello, Daniel P.; Young, Jennifer A.; Garcia-Irrizary, Carmen N.; Czabaniuk, Lara; Schuff, Brandon; Oliver, Robert; Montgomery, Justin; Hayward, Matthew M.; Coe, Jotham; Chen, Jinshan; Niosi, Mark; Luthra, Suman; Shah, Jaymin C.; El-Kattan, Ayman; Qiu, Xiayang; West, Graham M.; Noe, Mark C.; Shanmugasundaram, Veerabahu; Gilbert, Adam M.; Brown, Matthew F.; Calabrese, Matthew F.
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Novel Methods for Prioritizing Close-In Analogs from Structure-Activity Relationship Matrices
err2017-07-13
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PREAI
errZhang, Liying; Johnson, Kjell; Starr, Jeremy; Milbank, Jared; Kuhn, Andrew M.; Poss, Christopher; Stanton, Robert V.; Shanmugasundaram, Veerabahu
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Markov modeling reveals novel intracellular modulation of the human TREK-2 selectivity filter
err2017-04-04
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errOAAI
errHarrigan, Matthew P.; McKiernan, Keri A.; Shanmugasundaram, Veerabahu; Denny, Rajiah Aldrin; Pande, Vijay S.
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Evaluation and Characterization of Trk Kinase Inhibitors for the Treatment of Pain: Reliable Binding Affinity Predictions from Theory and Computation
err2017-04-04
err32
errOAAI
errWan, Shunzhou; Bhati, Agastya P.; Skerratt, Sarah; Omoto, Kiyoyuki; Shanmugasundaram, Veerabahu; Bagal, Sharan K.; Coveney, Peter V.
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Collaborating to improve the use of free-energy and other quantitative methods in drug discovery
err2016-12-24
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PREAI
errSherborne, Bradley; Shanmugasundaram, Veerabahu; Cheng, Alan C.; Christ, Clara D.; DesJarlais, Renee L.; Duca, Jose S.; Lewis, Richard A.; Loughney, Deborah A.; Manas, Eric S.; McGaughey, Georgia B.; Peishoff, Catherine E.; van Vlijmen, Herman
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Molecular Basis for Inhibition of the Na+/Citrate Transporter NaCT (SLC13A5) by Dicarboxylate Inhibitors
err2016-12-01
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errOAAI
errPajor, Ana M.; de Oliveira, Cesar A.; Song, Kun; Huard, Kim; Shanmugasundaram, Veerabahu; Erion, Derek M.
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Discovery of a Selective Covalent Inhibitor of Lysophospholipase-like 1 (LYPLAL1) as a Tool to Evaluate the Role of this Serine Hydrolase in Metabolism
err2016-07-19
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errOAAI
errAhn, Kay; Boehm, Markus; Brown, Matthew F.; Calloway, Jessica; Che, Ye; Chen, Jinshan; Fennell, Kimberly F.; Geoghegan, Kieran F.; Gilbert, Adam M.; Gutierrez, Jemy A.; Kalgutkar, Amit S.; Lanba, Adhiraj; Limberalds, Chris; Magee, Thomas V.; O'Doherty, Inish; Oliver, Robert; Pabst, Brandon; Pandit, Jayvardhan; Parris, Kevin; Pfefferkorn, Jeffrey A.; Rolph, Timothy P.; Patel, Rushi; Schuff, Brandon; Shanmugasundaram, Veerabahu; Starr, Jeremy T.; Varghese, Alison H.; Vera, Nicholas B.; Vernochet, Cecile; Yan, Jiangli
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Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging
err2016-06-29
err75
errOAAI
errLiang, Steven H.; Chen, Jinshan Michael; Normandin, Marc D.; Chang, Jeanne S.; Chang, George C.; Taylor, Christine K.; Trapa, Patrick; Plummer, Mark S.; Para, Kimberly S.; Conn, Edward L.; Lopresti-Morrow, Lori; Lanyon, Lorraine F.; Cook, James M.; Richter, Karl E. G.; Nolan, Charlie E.; Schachter, Joel B.; Janat, Fouad; Che, Ye; Shanmugasundaram, Veerabahu; Lefker, Bruce A.; Enerson, Bradley E.; Livni, Elijahu; Wang, Lu; Guehl, Nicolas J.; Patnaik, Debasis; Wagner, Florence F.; Perlis, Roy; Holson, Edward B.; Haggarty, Stephen J.; El Fakhri, Georges; Kurumbail, Ravi G.; Vasdev, Neil
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