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Ronald J. Hill

University of Sydney

41H指数
280论文数
1.0W被引数
收录论文 43
发表时间
Preclinical development of TCR-modified T cell therapies against mutated KRAS针对突变型KRAS的TCR修饰T细胞疗法的临床前开发
err2024-09-01
err0
PREAI
errSalter, H.; Pase, L.; Brass, A.; Bashir, Z.; Casarrubea, D.; Cullerton, S. Virding; Dunst, J.; Horta, S.; Masia-Balague, M.; Lange, J.; Parrot, T.; Totomi, A.; Uchtenhagen, H.; Wang, S.; Hill, R.; Jarvis, R.
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Discovery of Reversible Covalent Bruton's Tyrosine Kinase InhibitorsPRN473 and PRN1008 (Rilzabrutinib)
err2022-03-18
err37
PREAI
errOwens, Timothy D.; Brameld, Ken A.; Verner, Erik J.; Ton, Tony; Li, Xiaoyan; Zhu, Jiang; Masjedizadeh, Mohammad R.; Bradshaw, J. Michael; Hill, Ronald J.; Tam, Danny; Bisconte, Angelina; Kim, Eun Ok; Francesco, Michelle; Xing, Yan; Shu, Jin; Karr, Dane; LaStant, Jacob; Finkle, David; Loewenstein, Natalie; Haberstock-Debic, Helena; Taylor, Michael J.; Nunn, Philip; Langrish, Claire L.; Goldstein, David M.
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Purification of an insect juvenile hormone receptor complex enables insights into its post-translational phosphorylation
err2021-12-01
err15
errOAAI
errJindra, Marek; McKinstry, William J.; Nebl, Thomas; Bittova, Lenka; Ren, Bin; Shaw, Jan; Phan, Tram; Lu, Louis; Low, Jason K. K.; Mackay, Joel P.; Sparrow, Lindsay G.; Lovrecz, George O.; Hill, Ronald J.
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Oncogenic activation of JAK3-STAT signaling confers clinical sensitivity to PRN371, a novel selective and potent JAK3 inhibitor, in natural killer/T-cell lymphoma
errLEUKEMIA
IF13.4
err2018-02-02
err46
errOAAI
errNairismagi, M. -L.; Gerritsen, M. E.; Li, Z. M.; Wijaya, G. C.; Chia, B. K. H.; Laurensia, Y.; Lim, J. Q.; Yeoh, K. W.; Yao, X. S.; Pang, W. L.; Bisconte, A.; Hill, R. J.; Bradshaw, J. M.; Huang, D.; Song, T. L. L.; Ng, C. C. Y.; Rajasegaran, V.; Tang, T.; Tang, Q. Q.; Xia, X. J.; Kang, T. B.; Teh, B. T.; Lim, S. T.; Ong, C. K.; Tan, J.
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PRN473, an inhibitor of Bruton's tyrosine kinase, inhibits neutrophil recruitment via inhibition of macrophage antigen-1 signalling
err2017-12-22
err23
errOAAI
errHerter, Jan M.; Margraf, Andreas; Volmering, Stephanie; Correia, Benedito Eduardo; Bradshaw, J. Michael; Bisconte, Angelina; Hill, Ronald J.; Langrish, Claire L.; Lowell, Clifford A.; Zarbock, Alexander
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The Irreversible Covalent Fibroblast Growth Factor Receptor Inhibitor PRN1371 Exhibits Sustained Inhibition of FGFR after Drug Clearance
err2017-12-03
err22
errOAAI
errVenetsanakos, Eleni; Brameld, Ken A.; Phan, Vernon T.; Verner, Erik; Owens, Timothy D.; Xing, Yan; Tam, Danny; LaStant, Jacob; Leung, Kwan; Karr, Dane E.; Hill, Ronald J.; Gerritsen, Mary E.; Goldstein, David M.; Funk, Jens Oliver; Bradshaw, J. Michael
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A Small Molecule Inhibitor of ITK and RLK Impairs Th1 Differentiation and Prevents Colitis Disease Progression
err2015-11-15
err31
errOAAI
errCho, Hyoung-Soo; Shin, Hyun Mu; Haberstock-Debic, Helena; Xing, Yan; Owens, Timothy D.; Funk, Jens Oliver; Hill, Ronald J.; Bradshaw, J. Michael; Berg, Leslie J.
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Genetic Evidence for Function of the bHLH-PAS Protein Gce/Met As a Juvenile Hormone Receptor
err2015-07-10
err190
errOAAI
errJindra, Marek; Uhlirova, Mirka; Charles, Jean-Philippe; Smykal, Vlastimil; Hill, Ronald J.
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PRECLINICAL CHARACTERIZATION OF PRN1008, A NOVEL REVERSIBLE COVALENT INHIBITOR OF BTK THAT SHOWS EFFICACY IN A RAT MODEL OF COLLAGEN-INDUCED ARTHRITIS
err2015-06-01
err10
PREAI
errHill, R. J.; Bradshaw, J. M.; Bisconte, A.; Tam, D.; Owens, T. D.; Brameld, K. A.; Smith, P. F.; Funk, J. O.; Goldstein, D. M.; Nunn, P. A.
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Prolonged and tunable residence time using reversible covalent kinase inhibitors
err2015-05-25
err355
errOAAI
errBradshaw, J. Michael; McFarland, Jesse M.; Paavilainen, Ville O.; Bisconte, Angelina; Tam, Danny; Phan, Vernon T.; Romanov, Sergei; Finkle, David; Shu, Jin; Patel, Vaishali; Ton, Tony; Li, Xiaoyan; Loughhead, David G.; Nunn, Philip A.; Karr, Dane E.; Gerritsen, Mary E.; Funk, Jens Oliver; Owens, Timothy D.; Verner, Erik; Brameld, Ken A.; Hill, Ronald J.; Goldstein, David M.; Taunton, Jack
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Targeting Interleukin-2-inducible T-cell Kinase (ITK) and Resting Lymphocyte Kinase (RLK) Using a Novel Covalent Inhibitor PRN694
err2015-03-01
err50
errOAAI
errZhong, Yiming; Dong, Shuai; Strattan, Ethan; Ren, Li; Butchar, Jonathan P.; Thornton, Kelsey; Mishra, Anjali; Porcu, Pierluigi; Bradshaw, J. Michael; Bisconte, Angelina; Owens, Timothy D.; Verner, Erik; Brameld, Ken A.; Funk, Jens Oliver; Hill, Ronald J.; Johnson, Amy J.; Dubovsky, Jason A.
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Structure-Based Drug Design of RN486, a Potent and Selective Bruton's Tyrosine Kinase (BTK) Inhibitor, for the Treatment of Rheumatoid Arthritis
err2014-04-16
err96
PREAI
errLou, Yan; Han, Xiaochun; Kuglstatter, Andreas; Kondru, Rama K.; Sweeney, Zachary K.; Soth, Michael; McIntosh, Joel; Litman, Renee; Suh, Judy; Kocer, Buelent; Davis, Dana; Park, Jaehyeon; Frauchiger, Sandra; Dewdney, Nolan; Zecic, Hasim; Taygerly, Joshua P.; Sarma, Keshab; Hong, Junbae; Hill, Ronald J.; Gabriel, Tobias; Goldstein, David M.; Owens, Timothy D.
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Ecdysone Receptors: From the Ashburner Model to Structural Biology
err2013-01-07
err129
PREAI
errHill, Ronald J.; Billas, Isabelle M. L.; Bonneton, Francois; Graham, Lloyd D.; Lawrence, Michael C.
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The nature of porosity in organic-rich mudstones of the Upper Jurassic Kimmeridge Clay Formation, North Sea, offshore United Kingdom
err2012-12-01
err353
PREAI
errFishman, Neil S.; Hackley, Paul C.; Lowers, Heather A.; Hill, Ronald J.; Egenhoff, Sven O.; Eberl, Dennis D.; Blum, Alex E.
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RN486, a Selective Bruton's Tyrosine Kinase Inhibitor, Abrogates Immune Hypersensitivity Responses and Arthritis in Rodents
err2012-04-01
err142
PREAI
errXu, Daigen; Kim, Yong; Postelnek, Jennifer; Minh Diem Vu; Hu, Dong-Qing; Liao, Cheng; Bradshaw, Mike; Hsu, Jonathan; Zhang, Jun; Pashine, Achal; Srinivasan, Dinesh; Woods, John; Levin, Anita; O'Mahony, Alison; Owens, Timothy D.; Lou, Yan; Hill, Ronald J.; Narula, Satwant; DeMartino, Julie; Fine, Jay S.
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Isoforms of the heteropteran Nezara viridula ecdysone receptor: protein characterisation, RH5992 insecticide binding and homology modelling
err2011-05-18
err10
PREAI
errTohidi-Esfahani, Donya; Lawrence, Michael C.; Graham, Lloyd D.; Hannan, Garry N.; Simpson, Ann M.; Hill, Ronald J.
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Discovery of 6-(2,4-Difluorophenoxy)-2[3-hydroxy-1-(2-hydroxyethyl)propylamino]-8-methyl-8H-pyrido[2,3-d]pyrimidin-7-one (Pamapimod) and 6-(2,4-Difluorophenoxy)-8-methyl-2-(tetrahydro-2H-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8H)-one (R1487) as Orally Bioavailable and Highly Selective Inhibitors of p38α Mitogen-Activated Protein Kinase
err2011-03-04
err60
PREAI
errGoldstein, David M.; Soth, Michael; Gabriel, Tobias; Dewdney, Nolan; Kuglstatter, Andreas; Arzeno, Humberto; Chen, Jeffrey; Bingenheimer, William; Dalrymple, Stacie A.; Dunn, James; Farrell, Robert; Frauchiger, Sandra; La Fargue, JoAnn; Ghate, Manjiri; Graves, Bradford; Hill, Ronald J.; Li, Fujun; Litman, Renee; Loe, Brad; McIntosh, Joel; McWeeney, Daniel; Papp, Eva; Park, Jaehyeon; Reese, Harlan F.; Roberts, Richard T.; Rotstein, David; Pablo, Bong San; Sarma, Keshab; Stahl, Martin; Sung, Man-Ling; Suttman, Rebecca T.; Sjogren, Eric B.; Tan, Yunchou; Trejo, Alejandra; Welch, Mary; Weller, Paul; Wong, Brian R.; Zecic, Hasim
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