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George D. Hartman

merck & company

52H指数
284论文数
9.8K被引数
收录论文 69
发表时间
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Antiviral Activity, Safety, and Pharmacokinetics of Capsid Assembly Modulator NVR 3-778 in Patients with Chronic HBV Infection
err2019-04-01
err114
errOAAI
errYuen, Man Fung; Gane, Edward J.; Kim, Dong Joon; Weilert, Frank; Chan, Henry Lik Yuen; Lalezari, Jacob; Hwang, Seong Gyu; Tuan Nguyen; Flores, Osvaldo; Hartman, George; Liaw, Sandy; Lenz, Oliver; Kakuda, Thomas N.; Talloen, Willem; Schwabe, Christian; Klumpp, Klaus; Brown, Nathaniel
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Preclinical Characterization of NVR 3-778, a First-in-Class Capsid Assembly Modulator against Hepatitis B Virus
err2019-01-01
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errLam, Angela M.; Espiritu, Christine; Vogel, Robert; Ren, Suping; Lau, Vincent; Kelly, Mollie; Kuduk, Scott D.; Hartman, George D.; Flores, Osvaldo A.; Klumpp, Klaus
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MK-7622: A First-in-Class M1 Positive Allosteric Modulator Development Candidate
err2018-04-30
err28
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errBeshore, Douglas C.; Di Marco, Christina N.; Chang, Ronald K.; Greshock, Thomas J.; Ma, Lei; Wittmann, Marion; Seager, Matthew A.; Koeplinger, Kenneth A.; Thompson, Charles D.; Fuerst, Joy; Hartman, George D.; Bilodeau, Mark T.; Ray, William J.; Kuduk, Scott D.
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Hepatitis B Virus Capsid Assembly Modulators, but Not Nucleoside Analogs, Inhibit the Production of Extracellular Pregenomic RNA and Spliced RNA Variants
err2017-08-01
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errLam, Angela M.; Ren, Suping; Espiritu, Christine; Kelly, Mollie; Lau, Vincent; Zheng, Lingjie; Hartman, George D.; Flores, Osvaldo A.; Klumpp, Klaus
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NVR 3-778, A FIRST-IN-CLASS HBVCORE INHIBITOR, ALONE AND IN COMBINATION WITH PEG-INTERFERON (PEGIFN), IN TREATMENT-NAIVE HBEAG-POSITIVE PATIENTS: EARLY REDUCTIONS IN HBV DNA AND HBEAG
err2016-01-01
err45
PREAI
errYuen, M-F.; Kim, D. J.; Weilert, F.; Chan, H. L-Y.; Lalezari, J. P.; Hwang, S. G.; Nguyen, T.; Liaw, S.; Brown, N.; Klumpp, K.; Flores, O.; Hartman, G.; Gane, E.
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High-resolution crystal structure of a hepatitis B virus replication inhibitor bound to the viral core protein与病毒核心蛋白结合的乙型肝炎病毒复制抑制剂的高分辨率晶体结构
err2015-11-23
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errKlumpp, Klaus; Lam, Angela M.; Lukacs, Christine; Vogel, Robert; Ren, Suping; Espiritu, Christine; Baydo, Ruth; Atkins, Kateri; Abendroth, Jan; Liao, Guochun; Efimov, Andrey; Hartman, George; Flores, Osvaldo A.
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An allosteric Akt inhibitor effectively blocks Akt signaling and tumor growth with only transient effects on glucose and insulin levels in vivo
err2014-10-27
err58
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errCherrin, Craig; Haskell, Kathleen; Howell, Bonnie; Jones, Raymond; Leander, Karen; Robinson, Ronald; Watkins, Aubrey; Bilodeau, Mark; Hoffman, Jacob; Sanderson, Philip; Hartman, George; Mahan, Elizabeth; Prueksantanont, Thomayant; Jiang, Guoqiang; She, Qing-Bai; Rosen, Neal; Sepp-Lorenzino, Laura; Defeo-Jones, Deborah; Huber, Hans E.
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Discovery of Naphthyl-Fused 5-Membered Lactams as a New Class of M1 Positive Allosteric Modulators
err2014-02-26
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errYang, Zhi-Qiang; Shu, Youheng; Ma, Lei; Wittmann, Marion; Ray, William J.; Seager, Matthew A.; Koeplinger, Kenneth A.; Thompson, Charles D.; Hartman, George D.; Bilodeau, Mark T.; Kuduk, Scott D.
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Discovery of 5-Chloro-N-[( 5,6-dimethoxypyridin-2-yl)methyl]-2,2′:5′,3-terpyridine-3′-carboxamide (MK-1064): A Selective Orexin 2 Receptor Antagonist (2-SORA) for the Treatment of Insomnia
err2013-12-27
err78
PREAI
errRoecker, Anthony J.; Mercer, Swati P.; Schreier, John D.; Cox, Christopher D.; Fraley, Mark E.; Steen, Justin T.; Lemaire, Wei; Bruno, Joseph G.; Harrell, C. Meacham; Garson, Susan L.; Gotter, Anthony L.; Fox, Steven V.; Stevens, Joanne; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, Tamara D.; Cui, Donghui; Stellabott, Joyce; Hartman, George D.; Young, Steven D.; Winrow, Christopher J.; Renger, John J.; Coleman, Paul J.
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Identification of Amides as Carboxylic Acid Surrogates for Quinolizidinone-Based M1 Positive Allosteric Modulators
err2012-10-18
err22
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errKuduk, Scott D.; Chang, Ronald K.; Greshock, Thomas J.; Ray, William J.; Ma, Lei; Wittmann, Marion; Seager, Matthew A.; Koeplinger, Kenneth A.; Thompson, Charles D.; Hartman, George D.; Bilodeau, Mark T.
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Discovery of [(2R,5R)-5-{[(5-Fluoropyridin-2-yl)oxy]methyl}-2-methylpiperidin-1-yl][5-methyl-2-(pyrimidin-2-yl)phenyl]methanone (MK-6096): A Dual Orexin Receptor Antagonist with Potent Sleep-Promoting Properties
err2012-02-03
err121
PREAI
errColeman, Paul J.; Schreier, John D.; Cox, Christopher D.; Breslin, Michael J.; Whitman, David B.; Bogusky, Michael J.; McGaughey, Georgia B.; Bednar, Rodney A.; Lemaire, Wei; Doran, Scott M.; Fox, Steven V.; Garson, Susan L.; Gotter, Anthony L.; Harrell, C. Meacham; Reiss, Duane R.; Cabalu, Tamara D.; Cui, Donghui; Prueksaritanont, Thomayant; Stevens, Joanne; Tannenbaum, Pamela L.; Ball, Richard G.; Stellabott, Joyce; Young, Steven D.; Hartman, George D.; Winrow, Christopher J.; Renger, John J.
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Discovery of selective glucocorticoid receptor modulator MK-5932
err2011-12-01
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PREAI
errBungard, Christopher J.; Hartman, George D.; Manikowski, Jesse J.; Perkins, James J.; Bai, Chang; Brandish, Philip E.; Euler, Danielle H.; Hershey, James C.; Schmidt, Azriel; Fang, Yulin; Norcross, Ryan T.; Rushmore, Tom H.; Thompson, Charles D.; Meissner, Robert S.
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Discovery of a Selective Allosteric M1 Receptor Modulator with Suitable Development Properties Based on a Quinolizidinone Carboxylic Acid Scaffold
err2011-06-17
err60
PREAI
errKuduk, Scott D.; Chang, Ronald K.; Di Marco, Christina N.; Pitts, Daniel R.; Greshock, Thomas J.; Ma, Lei; Wittmann, Marion; Seager, Matthew A.; Koeplinger, Kenneth A.; Thompson, Charles D.; Hartman, George D.; Bilodeau, Mark T.; Rays, William J.
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Synthesis and Evaluation of 5-Fluoro-2-aryloxazolo[5,4-b]pyridines as β-Amyloid PET Ligands and Identification of MK-3328
err2011-04-18
err14
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errHarrison, Scott T.; Mulhearn, James; Wolkenberg, Scott E.; Miller, Patricia J.; O'Malley, Stacey S.; Zeng, Zhizhen; Williams, David L., Jr.; Hostetler, Eric D.; Sanabria-Bohorquez, Sandra; Gammage, Linda; Fan, Hong; Sur, Cyrille; Culberson, J. Christopher; Hargreaves, Richard J.; Cook, Jacquelynn J.; Hartman, George D.; Barrow, James C.
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Design, Synthesis, and Evaluation of Novel 3,6-Diaryl-4-aminoalkoxyquinolines as Selective Agonists of Somatostatin Receptor Subtype 2
err2011-03-11
err55
PREAI
errWolkenberg, Scott E.; Zhao, Zhijian; Thut, Catherine; Maxwell, Jill W.; McDonald, Terrence P.; Kinose, Fumi; Reilly, Michael; Lindsley, Craig W.; Hartman, George D.
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Short-Acting T-Type Calcium Channel Antagonists Significantly Modify Sleep Architecture in Rodents短效T型钙通道拮抗剂可显着改变啮齿动物的睡眠结构
err2010-08-24
err21
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errYang, Zhi-Qiang; Schlegel, Kelly-Ann S.; Shu, Youheng; Reger, Thomas S.; Cube, Rowena; Mattern, Christa; Coleman, Paul J.; Small, Jim; Hartman, George D.; Ballard, Jeanine; Tang, Cuyue; Kuo, Yuhsin; Prueksaritanont, Thomayant; Nuss, Cindy E.; Doran, Scott; Fox, Steve V.; Garson, Susan L.; Li, Yuxing; Kraus, Richard L.; Uebele, Victor N.; Taylor, Adekemi B.; Zeng, Wei; Fang, Wei; Chavez-Eng, Cynthia; Troyer, Matthew D.; Luk, Julie Ann; Laethem, Tine; Cook, William O.; Renger, John J.; Barrow, James C.
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Discovery of Oxazolobenzimidazoles as Positive Allosteric Modulators for the mGluR2 Receptor
err2010-07-12
err41
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errGarbaccio, Robert M.; Brnardic, Edward J.; Fraley, Mark E.; Hartman, George D.; Hutson, Pete H.; O'Brien, Julie A.; Magliaro, Brian C.; Uslaner, Jason M.; Huszar, Sarah L.; Fillgrove, Kerry L.; Small, James H.; Tang, Cuyue; Kuo, Yuhsin; Jacobson, Marlene A.
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