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收藏Preclinical characterization and phase I clinical trial of CT053PTSA targets MET, AXL, and VEGFR2 in patients with advanced solid tumors
Ma, Yu-Xiang; Liu, Fu-Rong; Zhang, Yang; Chen, Qun; Chen, Zhi-Qiang; Liu, Qian-Wen; Huang, Yan; Yang, Yun-Peng; Fang, Wen-Feng; Xi, Ning; Kang, Ning; Zhuang, Yu-Lei; Zhang, Qi; Jiang, Ying-Zhi; Zhang, Li; Zhao, Hong-Yun
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收藏A Class II small heat shock protein OsHsp18.0 plays positive roles in both biotic and abiotic defense responses in rice
Kuang, Jie; Liu, Jianzhong; Mei, Jun; Wang, Changchun; Hu, Haitao; Zhang, Yanjun; Sun, Meihao; Ning, Xi; Xiao, Langtao; Yang, Ling
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收藏Discovery of CT365, a highly potent inhibitor of PI3K and mTOR, for cancer treatment
Xi, Ning; Wu, Yanjun; Wang, Tingjin; Wang, Heng; Li, Zhiyong; Meng, Qingwei; Li, Jing; Wang, Zhaohe; Zhang, Yingjun
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收藏Structure-Based Design of Novel Class II c-Met Inhibitors: 2. SAR and Kinase Selectivity Profiles of the Pyrazolone Series
Liu, Longbin; Norman, Mark H.; Lee, Matthew; Xi, Ning; Siegmund, Aaron; Boezio, Alessandro A.; Booker, Shon; Choquette, Debbie; D'Angelo, Noel D.; Germain, Julie; Yang, Kevin; Yang, Yajing; Zhang, Yihong; Bellon, Steven F.; Whittington, Douglas A.; Harmange, Jean-Christophe; Dominguez, Celia; Kim, Tae-Seong; Dussault, Isabelle
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收藏Structure-Based Design of Novel Class II c-Met Inhibitors: 1. Identification of Pyrazolone-Based Derivatives
Norman, Mark H.; Liu, Longbin; Lee, Matthew; Xi, Ning; Fellows, Ingrid; D'Angelo, Noel D.; Dominguez, Celia; Rex, Karen; Bellon, Steven F.; Kim, Tae-Seong; Dussault, Isabelle
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收藏Discovery and Optimization of a Series of Benzothiazole Phosphoinositide 3-Kinase (PI3K)/Mammalian Target of Rapamycin (mTOR) Dual Inhibitors
D'Angelo, Noel D.; Kim, Tae-Seong; Andrews, Kristin; Booker, Shon K.; Caenepeel, Sean; Chen, Kui; D'Amico, Derin; Freeman, Dan; Jiang, Jian; Liu, Longbin; McCarter, John D.; Miguel, Tisha San; Mullady, Erin L.; Schrag, Michael; Subramanian, Raju; Tang, Jin; Wahl, Robert C.; Wang, Ling; Whittington, Douglas A.; Wu, Tian; Xi, Ning; Xu, Yang; Yakowec, Peter; Yang, Kevin; Zalameda, Leeanne P.; Zhang, Nancy; Hughes, Paul; Norman, Mark H.
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收藏Design, synthesis, and biological evaluation of potent c-Met inhibitors
D'Angelo, Noel D.; Bellon, Steven F.; Booker, Shon K.; Cheng, Yuan; Coxon, Angela; Dominguez, Celia; Fellows, Ingrid; Hoffman, Douglas; Hungate, Randall; Kaplan-Lefko, Paula; Lee, Matthew R.; Li, Chun; Liu, Longbin; Rainbeau, Elizabeth; Reider, Paul J.; Rex, Karen; Siegmund, Aaron; Sun, Yaxiong; Tasker, Andrew S.; Xi, Ning; Xu, Shimin; Yang, Yajing; Zhang, Yihong; Burgess, Teresa L.; Dussault, Isabelle; Kim, Tae-Seong
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收藏Discovery of a potent, selective, and orally bioavailable c-Met inhibitor:: 1-(2-Hydroxy-2-methylpropyl)-N-(5-(7-methoxyquinolin-4-yloxy)pyridin-2-yl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazole-4-carboxamide (AMG 458)
Liu, Longbin; Siegmund, Aaron; Xi, Ning; Kaplan-Lefko, Paula; Rex, Karen; Cheti, April; Lin, Jasmine; Moriguchi, Jodi; Berry, Loren; Huang, Liyue; Teffera, Yohannes; Yang, Yajing; Zhang, Yihong; Bellon, Steven F.; Lee, Matthew; Shimanovich, Roman; Bak, Annette; Dominguez, Celia; Norman, Mark H.; Harmange, Jean-Christophe; Dussault, Isabelle; Kimt, Tae-Seong
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收藏Design of potent, orally available antagonists of the transient receptor potential vanilloid 1.: Structure-activity relationships of 2-piperazin-1-yl-1H-benzimidazoles
Ognyanov, Vassil I.; Balan, Chenera; Bannon, Anthony W.; Bo, Yunxin; Dominguez, Celia; Fotsch, Christopher; Gore, Vijay K.; Klionsky, Lana; Ma, Vu V.; Qian, Yi-Xin; Tamir, Rami; Wang, Xianghong; Xi, Ning; Xu, Shimin; Zhu, Dawn; Gavva, Narender R.; Treanor, James J. S.; Norman, Mark H.
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