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收藏Design, synthesis and biological evaluation of (E)-4-(2-((1H-indol-5-yl) methylene) hydrazineyl)-5,6,7,8-tetrahydropyrido [4′,3′:4,5] thieno[2,3-d] pyrimidine derivatives as Arf1-GEFs inhibitors for the treatment of colon cancer(E)-4-(2-((1H-吲哚-5-基)亚甲基)肼基)-5,6,7,8-四氢吡啶并[4',3':4,5]噻吩并[2,3-d]嘧啶衍生物的设计、合成及生物评价:作为Arf1-GEFs抑制剂用于结肠癌的治疗
Ning Li; Chenfei Luo; Yufan Liu; Shaoliang Duan; Xuan Wang; Hua Cheng; Dengqi Xue; Yuetong Wang; Wei Li; Steven X. Hou; Liming Shao
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收藏Design, synthesis, and structure-activity relationship of 5,7-dimethylbenzo [d]thiazoles as novel Kv7.2/7.3 activators with antiepileptic effects5,7-二甲基苯并[d]噻唑的设计、合成及其作为具有抗癫痫作用的Kv7.2/7.3激活剂的构效关系
Zhang, Denggao; Xiang, Wei; Liu, Jie; Li, Wei; Qiao, Zhen; Wang, Kewei; Shao, Liming
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收藏Discovery of an Ortho-Substituted N-Cyclopropylmethyl-7α-phenyl-6,14-endoethano-tetrahydronorthebaine Derivative as a Selective and Potent Kappa Opioid Receptor Agonist with Subsided Sedative Effect
Li, Zixiang; Ye, Rufeng; He, Qian; Lu, Jiashuo; Sun, Yanting; Sun, Xiujian; Tang, Siyuan; Hu, Shuyang; Chai, Jingrui; Kong, Linghui; Liu, Xiaoning; Chen, Jing; Fang, Yun; Lan, Yingjie; Xie, Qiong; Liu, Jinggen; Shao, Liming; Fu, Wei; Wang, Yujun; Li, Wei
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收藏Synthesis of easily-modified and useful dibenzo-[b,d]azepines by palladium(ii)-catalyzed cyclization/addition with a green solvent
Cheng, Hua; Liu, Rongqi; Fang, Shengyang; Li, Zixiang; Zhang, Denggao; Zhang, Xi; Chen, Wenfei; Chen, Huixin; Kang, Leyi; Wang, Juan; Xu, Yulong; Song, Shaoli; Shao, Liming
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收藏Reversal of subtype-selectivity and function by the introduction of a para-benzamidyl substituent to N-cyclopropylmethyl nornepenthone
Kong, Linghui; Ning, Kuan; Liu, Xiao; Lu, Jiashuo; Chen, Baiyu; Ye, Rongrong; Li, Zixiang; Jiang, Shuang; Tang, Siyuan; Chai, Jing-Rui; Fang, Yun; Lan, Yingjie; Mai, Xiaobo; Xie, Qiong; Liu, Jinggen; Shao, Liming; Fu, Wei; Wang, Yujun; Li, Wei
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收藏Design, synthesis, and biological evaluation of acyl sulfonamide derivatives with spiro cycles as NaV1.7 inhibitors for antinociception
Ouyang, Xiangshuo; Su, Min; Xue, Dengqi; Dong, Liying; Niu, Heling; Li, Wei; Liu, Yani; Wang, KeWei; Shao, Liming
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