未登录Dual A2A/A2B Adenosine Receptor Antagonist M1069 Counteracts Immunosuppressive Mechanisms of Adenosine and Reduces Tumor Growth In Vivo
Schiemann, Kai; Belousova, Natalya; Matevossian, Armine; Nallaparaju, Kalyan C.; Kradjian, Giorgio; Pandya, Meghana; Chen, Zhouxiang; Aral, Esengul; Krauel, Eva-Maria; Petrova, Elissaveta; Boesler, Carsten; Kitzing, Thomas; Lecomte, Marc; Wagner, Christian; Blayo, Anne Laure; Schann, Stephan; Huck, Bayard; Moisan, Jacques; Zaynagetdinov, Rinat
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收藏Discovery of quinazoline HPK1 inhibitors with high cellular potency
Toure, Momar; Johnson, Theresa; Li, Bin; Schmidt, Ralf; Ma, Hong; Neagu, Constantin; Lopez, Andrea Unzue; Wang, Yanping; Guler, Satenig; Xiao, YuFang; Henkes, Renate; Ho, Kevin; Zhang, Susan; Chu, Chia Lin; Gundra, Uma Mahesh; Porichis, Filippos; Li, Long; Maurer, Christine Katharina; Fang, Zhizhou; Musil, Djordje; DiPoto, Maria; Friis, Emily; Jones, Reinaldo; Jones, Christopher; Cummings, James; Chekler, Eugene; Tanzer, Eva Maria; Huck, Bayard; Sherer, Brian
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收藏Selective Wee1 Inhibitors Led to Antitumor Activity In Vitro and Correlated with Myelosuppression选择性Wee1抑制剂导致体外抗肿瘤活性并与骨髓抑制相关
Guler, Satenig; DiPoto, Maria C.; Crespo, Alejandro; Caldwell, Richard; Doerfel, Benjamin; Grossmann, Nina; Ho, Kevin; Huck, Bayard; Jones, Christopher C., V; Lan, Ruoxi; Musil, Djordje; Potnick, Justin; Schilke, Heike; Sherer, Brian; Simon, Stephanie; Sirrenberg, Christian; Zhang, Zhuo; Liu-Bujalski, Lesley
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收藏Identification of Clinical Candidate M2698, a Dual p70S6K and Akt Inhibitor, for Treatment of PAM Pathway-Altered Cancers
DeSelm, Lizbeth; Huck, Bayard; Lan, Ruoxi; Neagu, Constantin; Potnick, Justin; Xiao, Yufang; Chen, Xiaoling; Jones, Reinaldo; Richardson, Thomas E.; Heasley, Brian H.; Haxell, Thomas; Moore, Joseph; Tian, Hui; Georgi, Katrin; Rohdich, Felix; Sutton, Amanda; Johnson, Theresa; Mochalkin, Igor; Jackson, Jennifer; Lin, Jing; Crowley, Lindsey; Machl, Andreas; Clark, Anderson; Wilker, Erik; Sherer, Brian; Goutopoulos, Andreas
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收藏Discovery of Evobrutinib: An Oral, Potent, and Highly Selective, Covalent Bruton's Tyrosine Kinase (BTK) Inhibitor for the Treatment of Immunological Diseases
Caldwell, Richard D.; Qiu, Hui; Askew, Ben C.; Bender, Andrew T.; Brugger, Nadia; Camps, Montserrat; Dhanabal, Mohanraj; Dutt, Vikram; Eichhorn, Thomas; Gardberg, Anna S.; Goutopoulos, Andreas; Grenningloh, Roland; Head, Jared; Healey, Brian; Hodous, Brian L.; Huck, Bayard R.; Johnson, Theresa L.; Jones, Christopher; Jones, Reinaldo C.; Mochalkin, Igor; Morandi, Federica; Ngan Nguyen; Meyring, Michael; Potnick, Justin R.; Santos, Dusica Cvetinovic; Schmidt, Ralf; Sherer, Brian; Shutes, Adam; Urbahns, Klaus; Follis, Ariele Viacava; Wegener, Ansgar A.; Zimmerli, Simone C.; Liu-Bujalski, Lesley
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收藏Antitumor activity of M8891, a potent and reversible inhibitor of methionine aminopeptidase 2
Friese-Hamim, Manja; Bogatyrova, Olga; Ortiz, Maria J.; Wienke, Dirk; Heinrich, Timo; Rohdich, Felix; Duecker, Klaus; Schultes, Christoph; Huck, Bayard; Zenke, Frank T.; Blaukat, Andree
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收藏A FIRST IN HUMAN, DOSE ESCALATION TRIAL OF MSC2363318A-A DUAL P70S6K/AKT INHIBITOR, FOR PATIENTS WITH ADVANCED MALIGNANCIES
Tsimberidou, A. M.; Verschraegen, C.; Heestand, G.; Kaleta, R.; Scheuenpflug, J.; Huck, B.; Weise, A.; Kurzrock, R.
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收藏Evaluation of p70S6K/Akt inhibitor MSC2363318A in patient derived xenograft (PDX) models of breast cancer
Huck, Bayard R.; Tian, H.; Syed, Sakeena; Lin, Jing; Ma, Jianguo; Clark, Anderson; Kaleta, Remiguisz; Machl, Andreas; Wilker, Erik; Lecomte, Marc
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收藏Identification of brain penetrant p70S6K/Akt inhibitor MSC2363318A.
Huck, Bayard R.; Machl, Andreas; Wilker, Erik; Tian, Hui; Syed, Sakeena; Lin, Jing; Ma, Jianguo; Clark, Anderson; Waterhouse, Roseann; Kaleta, Remiguisz; Micu, Alina; Soughley, Lynne; Li, Long; Groll, Karin; Kroesser, Sonja; Beier, Frank; Hering, Ursula; Lecomte, Marc; Wichert, Katrin; D'Antonio, Mauro; Di Eugenio, Paolo
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