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Bayard R. Huck

merck kgaa

17H指数
62论文数
1.3K被引数
收录论文 18
发表时间
Dual A2A/A2B Adenosine Receptor Antagonist M1069 Counteracts Immunosuppressive Mechanisms of Adenosine and Reduces Tumor Growth In Vivo
err2024-08-20
err0
PREAI
errSchiemann, Kai; Belousova, Natalya; Matevossian, Armine; Nallaparaju, Kalyan C.; Kradjian, Giorgio; Pandya, Meghana; Chen, Zhouxiang; Aral, Esengul; Krauel, Eva-Maria; Petrova, Elissaveta; Boesler, Carsten; Kitzing, Thomas; Lecomte, Marc; Wagner, Christian; Blayo, Anne Laure; Schann, Stephan; Huck, Bayard; Moisan, Jacques; Zaynagetdinov, Rinat
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Discovery of quinazoline HPK1 inhibitors with high cellular potency
err2023-09-01
err7
PREAI
errToure, Momar; Johnson, Theresa; Li, Bin; Schmidt, Ralf; Ma, Hong; Neagu, Constantin; Lopez, Andrea Unzue; Wang, Yanping; Guler, Satenig; Xiao, YuFang; Henkes, Renate; Ho, Kevin; Zhang, Susan; Chu, Chia Lin; Gundra, Uma Mahesh; Porichis, Filippos; Li, Long; Maurer, Christine Katharina; Fang, Zhizhou; Musil, Djordje; DiPoto, Maria; Friis, Emily; Jones, Reinaldo; Jones, Christopher; Cummings, James; Chekler, Eugene; Tanzer, Eva Maria; Huck, Bayard; Sherer, Brian
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Selective Wee1 Inhibitors Led to Antitumor Activity In Vitro and Correlated with Myelosuppression选择性Wee1抑制剂导致体外抗肿瘤活性并与骨髓抑制相关
err2023-04-07
err12
errOAAI
errGuler, Satenig; DiPoto, Maria C.; Crespo, Alejandro; Caldwell, Richard; Doerfel, Benjamin; Grossmann, Nina; Ho, Kevin; Huck, Bayard; Jones, Christopher C., V; Lan, Ruoxi; Musil, Djordje; Potnick, Justin; Schilke, Heike; Sherer, Brian; Simon, Stephanie; Sirrenberg, Christian; Zhang, Zhuo; Liu-Bujalski, Lesley
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Rules were made to be broken
err2023-01-01
err40
PREAI
errHartung, Ingo V.; Huck, Bayard R.; Crespo, Alejandro
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The expanding role for small molecules in immuno-oncology
err2022-08-18
err78
PREAI
errOffringa, Rienk; Kotzner, Lisa; Huck, Bayard; Urbahns, Klaus
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Identification of Clinical Candidate M2698, a Dual p70S6K and Akt Inhibitor, for Treatment of PAM Pathway-Altered Cancers
err2021-10-01
err5
PREAI
errDeSelm, Lizbeth; Huck, Bayard; Lan, Ruoxi; Neagu, Constantin; Potnick, Justin; Xiao, Yufang; Chen, Xiaoling; Jones, Reinaldo; Richardson, Thomas E.; Heasley, Brian H.; Haxell, Thomas; Moore, Joseph; Tian, Hui; Georgi, Katrin; Rohdich, Felix; Sutton, Amanda; Johnson, Theresa; Mochalkin, Igor; Jackson, Jennifer; Lin, Jing; Crowley, Lindsey; Machl, Andreas; Clark, Anderson; Wilker, Erik; Sherer, Brian; Goutopoulos, Andreas
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Discovery of Evobrutinib: An Oral, Potent, and Highly Selective, Covalent Bruton's Tyrosine Kinase (BTK) Inhibitor for the Treatment of Immunological Diseases
err2019-08-01
err104
errOAAI
errCaldwell, Richard D.; Qiu, Hui; Askew, Ben C.; Bender, Andrew T.; Brugger, Nadia; Camps, Montserrat; Dhanabal, Mohanraj; Dutt, Vikram; Eichhorn, Thomas; Gardberg, Anna S.; Goutopoulos, Andreas; Grenningloh, Roland; Head, Jared; Healey, Brian; Hodous, Brian L.; Huck, Bayard R.; Johnson, Theresa L.; Jones, Christopher; Jones, Reinaldo C.; Mochalkin, Igor; Morandi, Federica; Ngan Nguyen; Meyring, Michael; Potnick, Justin R.; Santos, Dusica Cvetinovic; Schmidt, Ralf; Sherer, Brian; Shutes, Adam; Urbahns, Klaus; Follis, Ariele Viacava; Wegener, Ansgar A.; Zimmerli, Simone C.; Liu-Bujalski, Lesley
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Antitumor activity of M8891, a potent and reversible inhibitor of methionine aminopeptidase 2
err2019-07-01
err2
PREAI
errFriese-Hamim, Manja; Bogatyrova, Olga; Ortiz, Maria J.; Wienke, Dirk; Heinrich, Timo; Rohdich, Felix; Duecker, Klaus; Schultes, Christoph; Huck, Bayard; Zenke, Frank T.; Blaukat, Andree
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A FIRST IN HUMAN, DOSE ESCALATION TRIAL OF MSC2363318A-A DUAL P70S6K/AKT INHIBITOR, FOR PATIENTS WITH ADVANCED MALIGNANCIES
err2015-03-01
err3
errOAAI
errTsimberidou, A. M.; Verschraegen, C.; Heestand, G.; Kaleta, R.; Scheuenpflug, J.; Huck, B.; Weise, A.; Kurzrock, R.
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Evaluation of p70S6K/Akt inhibitor MSC2363318A in patient derived xenograft (PDX) models of breast cancer
err2014-10-01
err1
PREAI
errHuck, Bayard R.; Tian, H.; Syed, Sakeena; Lin, Jing; Ma, Jianguo; Clark, Anderson; Kaleta, Remiguisz; Machl, Andreas; Wilker, Erik; Lecomte, Marc
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Identification of brain penetrant p70S6K/Akt inhibitor MSC2363318A.
err2013-11-01
err0
PREAI
errHuck, Bayard R.; Machl, Andreas; Wilker, Erik; Tian, Hui; Syed, Sakeena; Lin, Jing; Ma, Jianguo; Clark, Anderson; Waterhouse, Roseann; Kaleta, Remiguisz; Micu, Alina; Soughley, Lynne; Li, Long; Groll, Karin; Kroesser, Sonja; Beier, Frank; Hering, Ursula; Lecomte, Marc; Wichert, Katrin; D'Antonio, Mauro; Di Eugenio, Paolo
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Protein prosthesis:: A semisynthetic enzyme with a β-peptide reverse turn
err2002-06-22
err122
PREAI
errArnold, U; Hinderaker, MP; Nilsson, BL; Huck, BR; Gellman, SH; Raines, RT
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Stereochemical control of hairpin formation in β-peptides containing dinipecotic acid reverse turn segments
err2000-04-12
err145
PREAI
errChung, YJ; Huck, BR; Christianson, LA; Stanger, HE; Krauthäuser, S; Powell, DR; Gellman, SH
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