未登录Superior Efficacy of a Combined Epigenetic Therapy against Human Mantle Cell Lymphoma Cells (vol 18, pg 6227, 2012)
Fiskus, Warren; Rao, Rekha; Balusu, Ramesh; Ganguly, Siddhartha; Tao, Jianguo; Sotomayor, Eduardo; Mudunuru, Uma; Smith, Jacqueline E.; Hembruff, Stacey L.; Atadja, Peter; Marquez, Victor E.; Bhalla, Kapil
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收藏Discovery of Potent Small-Molecule Inhibitors of WDR5-MYC Interaction
Ding, Jian; Li, Guo; Liu, Hejun; Liu, Lulu; Lin, Ying; Gao, Jingyan; Zhou, Guoqiang; Shen, Lingling; Zhao, Mengxi; Yu, Yanyan; Guo, Weihui; Hommel, Ulrich; Ottl, Johannes; Blank, Jutta; Aubin, Nicola; Wei, Yi; He, Hu; Sage, David R.; Atadja, Peter W.; Li, En; Jain, Rishi K.; Tallarico, John A.; Canham, Stephen M.; Chiang, Ying-Ling; Wang, He
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收藏Discovery of the Clinical Candidate MAK683: An EED-Directed, Allosteric, and Selective PRC2 Inhibitor for the Treatment of Advanced Malignancies
Huang, Ying; Sendzik, Martin; Zhang, Jeff; Gao, Zhenting; Sun, Yongfeng; Wang, Long; Gu, Justin; Zhao, Kehao; Yu, Zhengtian; Zhang, Lijun; Zhang, Qiong; Blanz, Joachim; Chen, Zijun; Dubost, Valerie; Fang, Douglas; Feng, Lijian; Fu, Xingnian; Kiffe, Michael; Li, Ling; Luo, Fangjun; Luo, Xiao; Mi, Yuan; Mistry, Prakash; Pearson, David; Piaia, Alessandro; Scheufler, Clemens; Terranova, Remi; Weiss, Andreas; Zeng, Jue; Zhang, Hailong; Zhang, Jiangwei; Zhao, Mengxi; Dillon, Michael P.; Jeay, Sebastien; Qi, Wei; Moggs, Jonathan; Pissot-Soldermann, Carole; Li, En; Atadja, Peter; Lingel, Andreas; Oyang, Counde
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收藏Role of CAAT/Enhancer Binding Protein Homologous Protein in Panobinostat-mediated Potentiation of Bortezomib-induced Lethal Endoplasmic Reticulum Stress in Mantle Cell Lymphoma Cells (Expression of Concern of Vol 16, Pg 4742, 2010)
Rao, Rekha; Nalluri, Srilatha; Fiskus, Warren; Savoie, Andrew; Buckley, Kathleen M.; Ha, Kyungsoo; Balusu, Ramesh; Joshi, Atul; Coothankandaswamy, Veena; Tao, Jianguo; Sotomayor, Eduardo; Atadja, Peter; Bhalla, Kapil N.
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收藏Discovery of Potent and Selective Allosteric Inhibitors of Protein Arginine Methyltransferase 3 (PRMT3)蛋白质精氨酸甲基转移酶3 (PRMT3) 的有效和选择性变构抑制剂的发现
Kaniskan, H. Umit; Eram, Mohammad S.; Zhao, Kehao; Szewczyk, Magdalena M.; Yang, Xiaobao; Schmidt, Keith; Luo, Xiao; Xiao, Sean; Dai, Miao; He, Feng; Zang, Irene; Lin, Ying; Li, Fengling; Dobrovetsky, Elena; Smil, David; Min, Sun-Joon; Lin-Jones, Jennifer; Schapira, Matthieu; Atadja, Peter; Li, En; Barsyte-Lovejoy, Dalia; Arrowsmith, Cheryl H.; Brown, Peter J.; Liu, Feng; Yu, Zhengtian; Vedadi, Masoud; Jin, Jian
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收藏FXR1 regulates transcription and is required for tumor growth in TP53 homozygous deletion human cancers
Fan, Yichao; Yue, Jiao; Xiao, Mengtao; Han Han-Zhang; Wang, Yao Vickie; Ma, Chun; Deng, Zhilin; Li, Yingxiang; Yu, Yanyan; Wang, Xinghao; Niu, Shen; Hua, Youjia; Weng, Zhiping; Atadja, Peter; Li, En; Xiang, Bin
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收藏An allosteric PRC2 inhibitor targeting the H3K27me3 binding pocket of EED
Qi, Wei; Zhao, Kehao; Gu, Justin; Huang, Ying; Wang, Youzhen; Zhang, Hailong; Zhang, Man; Zhang, Jeff; Yu, Zhengtian; Li, Ling; Teng, Lin; Chuai, Shannon; Zhang, Chao; Zhao, Mengxi; Chan, HoMan; Chen, Zijun; Fang, Douglas; Qi, Fei; Feng, Leying; Feng, Lijian; Gao, Yuan; Ge, Hui; Ge, Xinjian; Lingel, Andreas; Li, Guobin; Lin, Ying; Liu, Yueqin; Luo, Fangjun; Shi, Minlong; Wang, Long; Wang, Zhaofu; Yu, Yanyan; Zeng, Jue; Zeng, Chenhui; Zhang, Lijun; Zhang, Qiong; Zhou, Shaolian; Oyang, Counde; Atadja, Peter; Li, En
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收藏HDAC Inhibitor Panobinostat Engages Host Innate Immune Defenses to Promote the Tumoricidal Effects of Trastuzumab in HER2+ TumorsHDAC抑制剂Panobinostat参与宿主先天免疫防御,以促进曲妥珠单抗在HER2肿瘤中的杀肿瘤作用
Medon, Mikolaj; Vidacs, Eva; Vervoort, Stephin J.; Li, Jason; Jenkins, Misty R.; Ramsbottom, Kelly M.; Trapani, Joseph A.; Smyth, Mark J.; Darcy, Phillip K.; Atadja, Peter W.; Henderson, Michael A.; Johnstone, Ricky W.; Haynes, Nicole M.
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收藏Discovery of First-in-Class, Potent, and Orally Bioavailable Embryonic Ectoderm Development (EED) Inhibitor with Robust Anticancer Efficacy
Huang, Ying; Zhang, Jeff; Yu, Zhengtian; Zhang, Hailong; Wang, Youzhen; Lingel, Andreas; Qi, Wei; Gu, Justin; Zhao, Kehao; Shultz, Michael D.; Wang, Long; Fu, Xingian; Sun, Yongfeng; Zhang, Qiong; Jiang, Xiangqing; Zhang, Jiangwei; Zhang, Chunye; Li, Ling; Zeng, Jue; Feng, Lijian; Zhang, Chao; Liu, Yueqin; Zhang, Man; Zhang, Lijun; Zhao, Mengxi; Gao, Zhenting; Liu, Xianghui; Fang, Douglas; Guo, Haibing; Mi, Yuan; Gabriel, Tobias; Dillon, Michael P.; Atadja, Peter; Oyang, Counde
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收藏An allosteric PRC2 inhibitor targeting the H3K27me3 binding pocket of EED
Qi, Wei; Zhao, Kehao; Gu, Justin; Huang, Ying; Wang, Youzhen; Zhang, Hailong; Zhang, Man; Zhang, Jeff; Yu, Zhengtian; Li, Ling; Teng, Lin; Chuai, Shannon; Zhang, Chao; Zhao, Mengxi; Chan, Homan; Chen, Zijun; Fang, Douglas; Fei, Qi; Feng, Leying; Feng, Lijian; Gao, Yuan; Ge, Hui; Ge, Xinjian; Li, Guobin; Lingel, Andreas; Lin, Ying; Liu, Yueqin; Luo, Fangjun; Shi, Minlong; Wang, Long; Wang, Zhaofu; Yu, Yanyan; Zeng, Jue; Zeng, Chenhui; Zhang, Lijun; Zhang, Qiong; Zhou, Shaolian; Oyang, Counde; Atadja, Peter; Li, En
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收藏Histone Demethylase LSD1 Promotes Adipocyte Differentiation through Repressing Wnt Signaling
Chen, Yan; Kim, Jeesun; Zhang, Ruipeng; Yang, Xiaoqin; Zhang, Yong; Fang, Jianwu; Chen, Zhui; Teng, Lin; Chen, Xiaowei; Ge, Hui; Atadja, Peter; Li, En; Chen, Taiping; Qi, Wei
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收藏RETRACTION: Histone deacetylase inhibitors activate NF-κB in human leukemia cells through an ATM/NEMO-related pathway (Retraction of vol 285, pg 10064, 2010)
Rosato, Roberto R.; Kolla, Sarah S.; Hock, Stefanie K.; Almenara, Jorge A.; Patel, Ankita; Amin, Sanjay; Atadja, Peter; Fisher, Paul B.; Dent, Paul; Grant, Steven
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收藏High-throughput screening using patient-derived tumor xenografts to predict clinical trial drug response使用患者来源的肿瘤异种移植物进行高通量筛选以预测临床试验药物反应
Gao, Hui; Korn, Joshua M.; Ferretti, Stephane; Monahan, John E.; Wang, Youzhen; Singh, Mallika; Zhang, Chao; Schnell, Christian; Yang, Guizhi; Zhang, Yun; Balbin, O. Alejandro; Barbe, Stephanie; Cai, Hongbo; Casey, Fergal; Chatterjee, Susmita; Chiang, Derek Y.; Chuai, Shannon; Cogan, Shawn M.; Collins, Scott D.; Dammassa, Ernesta; Ebel, Nicolas; Embry, Millicent; Green, John; Kauffmann, Audrey; Kowa, Colleen; Leary, Rebecca J.; Lehar, Joseph; Liang, Ying; Loo, Alice; Lorenzana, Edward; McDonald, E. Robert, III; McLaughlin, Margaret E.; Merkin, Jason; Meyer, Ronald; Naylor, Tara L.; Patawaran, Montesa; Reddy, Anupama; Roeelli, Claudia; Ruddy, David A.; Salangsang, Fernando; Santacroce, Francesca; Singh, Angad P.; Tang, Yan; Tinetto, Walter; Tobler, Sonja; Velazquez, Roberto; Venkatesan, Kavitha; Von Arx, Fabian; Wang, Hui Qin; Wang, Zongyao; Wiesmann, Marion; Wyss, Daniel; Xu, Fiona; Bitter, Hans; Atadja, Peter; Lees, Emma; Hofmann, Francesco; Li, En; Keen, Nicholas; Cozens, Robert; Jensen, Michael Rugaard; Pryer, Nancy K.; Williams, Juliet A.; Sellers, William R.
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收藏Histone methyltransferase SETDB1 regulates liver cancer cell growth through methylation of p53
Fei, Qi; Shang, Ke; Zhang, Jianhua; Chuai, Shannon; Kong, Desheng; Zhou, Tianlun; Fu, Shijun; Liang, Ying; Li, Chong; Chen, Zhi; Zhao, Yuan; Yu, Zhengtian; Huang, Zheng; Hu, Min; Ying, Haiyan; Chen, Zhui; Zhang, Yun; Xing, Feng; Zhu, Jidong; Xu, Haiyan; Zhao, Kehao; Lu, Chris; Atadja, Peter; Xiao, Zhi-Xiong; Li, En; Shou, Jianyong
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收藏SETDB1 modulates PRC2 activity at developmental genes independently of H3K9 trimethylation in mouse ES cells
Fei, Qi; Yang, Xiaoqin; Jiang, Hua; Wang, Qian; Yu, Yanyan; Yu, Yiling; Yi, Wei; Zhou, Shaolian; Chen, Taiping; Lu, Chris; Atadja, Peter; Liu, Xiaole Shirley; Li, En; Zhang, Yong; Shou, Jianyong
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收藏A Potent, Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 3 (PRMT3)蛋白质精氨酸甲基转移酶3 (PRMT3) 的有效,选择性和细胞活性变构抑制剂
Kaniskan, H. Uemit; Szewczyk, Magdalena M.; Yu, Zhengtian; Eram, Mohammad S.; Yang, Xiaobao; Schmidt, Keith; Luo, Xiao; Dai, Miao; He, Feng; Zang, Irene; Lin, Ying; Kennedy, Steven; Li, Fengling; Dobrovetsky, Elena; Dong, Aiping; Smil, David; Min, Sun-Joon; Landon, Melissa; Lin-Jones, Jennifer; Huang, Xi-Ping; Roth, Bryan L.; Schapira, Matthieu; Atadja, Peter; Barsyte-Lovejoy, Dalia; Arrowsmith, Cheryl H.; Brown, Peter J.; Zhao, Kehao; Jin, Jian; Vedadi, Masoud
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