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John Xue

AbbVie

16H指数
48论文数
5.4K被引数
收录论文 18
发表时间
Compelling colorings: A generalization of the dominator chromatic number
err2022-09-01
err2
errOAAI
errBachstein, Anna; Goddard, Wayne; Henning, Michael A.; Xue, John
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Hexavalent TRAIL Fusion Protein Eftozanermin Alfa Optimally Clusters Apoptosis-Inducing TRAIL Receptors to Induce On-Target Antitumor Activity in Solid Tumors
err2021-03-09
err29
errOAAI
errPhillips, Darren C.; Buchanan, Fritz G.; Cheng, Dong; Solomon, Larry R.; Xiao, Yu; Xue, John; Tahir, Stephen K.; Smith, Morey L.; Zhang, Haichao; Widomski, Deborah; Abraham, Vivek C.; Xu, Nan; Liu, Zhihong; Zhou, Li; DiGiammarino, Enrico; Lu, Xin; Rudra-Ganguly, Nandini; Trela, Bruce; Morgan-Lappe, Susan E.
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Discovery of A-1331852, a First-in-Class, Potent, and Orally-Bioavailable BCL-XL Inhibitor
err2020-03-30
err93
errOAAI
errWang, Le; Doherty, George A.; Judd, Andrew S.; Tao, Zhi-Fu; Hansen, T. Matthew; Frey, Robin R.; Song, Xiaohong; Bruncko, Milan; Kunzer, Aaron R.; Wang, Xilu; Wendt, Michael D.; Flygare, John A.; Catron, Nathaniel D.; Judge, Russell A.; Park, Chang H.; Shekhar, Shashank; Phillips, Darren C.; Nimmer, Paul; Smith, Morey L.; Tahir, Stephen K.; Xiao, Yu; Xue, John; Zhang, Haichao; Le, Phuong N.; Mitten, Michael J.; Boghaert, Erwin R.; Gao, Wenqing; Kovar, Peter; Choo, Edna F.; Diaz, Dolores; Fairbrother, Wayne J.; Elmore, Steven W.; Sampath, Deepak; Leverson, Joel D.; Souers, Andrew James
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A novel CDK9 inhibitor increases the efficacy of venetoclax (ABT-199) in multiple models of hematologic malignancies
errLEUKEMIA
IF13.4
err2019-12-11
err61
errOAAI
errPhillips, Darren C.; Jin, Sha; Gregory, Gareth P.; Zhang, Qi; Xue, John; Zhao, Xiaoxian; Chen, Jun; Tong, Yunsong; Zhang, Haichao; Smith, Morey; Tahir, Stephen K.; Clark, Rick F.; Penning, Thomas D.; Devlin, Jennifer R.; Shortt, Jake; Hsi, Eric D.; Albert, Daniel H.; Konopleva, Marina; Johnstone, Ricky W.; Leverson, Joel D.; Souers, Andrew J.
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Genomic analysis and selective small molecule inhibition identifies BCL-XL as a critical survival factor in a subset of colorectal cancer
err2015-07-02
err47
errOAAI
errZhang, Haichao; Xue, John; Hessler, Paul; Tahir, Stephen K.; Chen, Jun; Jin, Sha; Souers, Andrew J.; Leverson, Joel D.; Lam, Lloyd T.
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Structure-Guided Design of a Series of MCL-1 Inhibitors with High Affinity and Selectivity (vol 58, pg 2180, 2015)
err2015-05-01
err5
PREAI
errBruncko, Milan; Wang, Le; Sheppard, George S.; Phillips, Darren C.; Tahir, Stephen K.; Xue, John; Erickson, Scott; Fidanze, Steve; Fry, Elizabeth; Hasvold, Lisa; Jenkins, Gary J.; Jin, Sha; Judge, Russell A.; Kovar, Peter J.; Madar, David; Nimmer, Paul; Park, Chang; Petros, Andrew M.; Rosenberg, Saul H.; Smith, Morey L.; Song, Xiaohong; Sun, Chaohong; Tao, Zhi-Fu; Wang, Xilu; Xiao, Yu; Zhang, Haichao; Tse, Chris; Leverson, Joel D.; Elmore, Steven W.; Souers, Andrew J.
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Exploiting selective BCL-2 family inhibitors to dissect cell survival dependencies and define improved strategies for cancer therapy
err2015-03-18
err474
PREAI
errLeverson, Joel D.; Phillips, Darren C.; Mitten, Michael J.; Boghaert, Erwin R.; Diaz, Dolores; Tahir, Stephen K.; Belmont, Lisa D.; Nimmer, Paul; Xiao, Yu; Ma, Xiaoju Max; Lowes, Kym N.; Kovar, Peter; Chen, Jun; Jin, Sha; Smith, Morey; Xue, John; Zhang, Haichao; Oleksijew, Anatol; Magoc, Terrance J.; Vaidya, Kedar S.; Albert, Daniel H.; Tarrant, Jacqueline M.; La, Nghi; Wang, Le; Tao, Zhi-Fu; Wendt, Michael D.; Sampath, Deepak; Rosenberg, Saul H.; Tse, Chris; Huang, David C. S.; Fairbrother, Wayne J.; Elmore, Steven W.; Souers, Andrew J.
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Structure-Guided Design of a Series of MCL-1 Inhibitors with High Affinity and Selectivity
err2015-02-26
err158
PREAI
errBruncko, Milan; Wang, Le; Sheppard, George S.; Phillips, Darren C.; Tahir, Stephen K.; Xue, John; Erickson, Scott; Fidanze, Steve; Fry, Elizabeth; Hasvold, Lisa; Jenkins, Gary J.; Jin, Sha; Judge, Russell A.; Kovar, Peter J.; Madar, David; Nimmer, Paul; Park, Chang; Petros, Andrew M.; Rosenberg, Saul H.; Smith, Morey L.; Song, Xiaohong; Sun, Chaohong; Tao, Zhi-Fu; Wang, Xilu; Xiao, Yu; Zhang, Haichao; Tse, Chris; Leverson, Joel D.; Elmore, Steven W.; Souers, Andrew J.
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Potent and selective small-molecule MCL-1 inhibitors demonstrate on-target cancer cell killing activity as single agents and in combination with ABT-263 (navitoclax)
err2015-01-15
err431
errOAAI
errLeverson, J. D.; Zhang, H.; Chen, J.; Tahir, S. K.; Phillips, D. C.; Xue, J.; Nimmer, P.; Jin, S.; Smith, M.; Xiao, Y.; Kovar, P.; Tanaka, A.; Bruncko, M.; Sheppard, G. S.; Wang, L.; Gierke, S.; Kategaya, L.; Anderson, D. J.; Wong, C.; Eastham-Anderson, J.; Ludlam, M. J. C.; Sampath, D.; Fairbrother, W. J.; Wertz, I.; Rosenberg, S. H.; Tse, C.; Elmore, S. W.; Souers, A. J.
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Colorectal cancer cell lines with high BCL-XL and low MCL-1 expression are sensitive to a potent and selective BCL-XL inhibitor
err2014-10-01
err2
PREAI
errLam, Lloyd T.; Zhang, Haichao; Xue, John; Hessler, Paul; Tahir, Stephen K.; Chen, Jun; Jin, Sha; Souers, Andrew J.; Leverson, Joel D.
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Discovery of a Potent and Selective BCL-XL Inhibitor with in Vivo Activity
err2014-09-08
err286
errOAAI
errTao, Zhi-Fu; Hasvold, Lisa; Wang, Le; Wang, Xilu; Petros, Andrew M.; Park, Chang H.; Boghaert, Erwin R.; Catron, Nathaniel D.; Chen, Jun; Colman, Peter M.; Czabotar, Peter E.; Deshayes, Kurt; Fairbrother, Wayne J.; Flygare, John A.; Hymowitz, Sarah G.; Jin, Sha; Judge, Russell A.; Koehler, Michael F. T.; Kovar, Peter J.; Lessene, Guillaume; Mitten, Michael J.; Ndubaku, Chudi O.; Nimmer, Paul; Purkey, Hans E.; Oleksijew, Anatol; Phillips, Darren C.; Sleebs, Brad E.; Smith, Brian J.; Smith, Morey L.; Tahir, Stephen K.; Watson, Keith G.; Xiao, Yu; Xue, John; Zhang, Haichao; Zobel, Kerry; Rosenberg, Saul H.; Tse, Chris; Leverson, Joel D.; Elmore, Steven W.; Souers, Andrew J.
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ABT-199, a potent and selective BCL-2 inhibitor, achieves antitumor activity while sparing platelets
err2013-01-06
err2.6K
PREAI
errSouers, Andrew J.; Leverson, Joel D.; Boghaert, Erwin R.; Ackler, Scott L.; Catron, Nathaniel D.; Chen, Jun; Dayton, Brian D.; Ding, Hong; Enschede, Sari H.; Fairbrother, Wayne J.; Huang, David C. S.; Hymowitz, Sarah G.; Jin, Sha; Khaw, Seong Lin; Kovar, Peter J.; Lam, Lloyd T.; Lee, Jackie; Maecker, Heather L.; Marsh, Kennan C.; Mason, Kylie D.; Mitten, Michael J.; Nimmer, Paul M.; Oleksijew, Anatol; Park, Chang H.; Park, Cheol-Min; Phillips, Darren C.; Roberts, Andrew W.; Sampath, Deepak; Seymour, John F.; Smith, Morey L.; Sullivan, Gerard M.; Tahir, Stephen K.; Tse, Chris; Wendt, Michael D.; Xiao, Yu; Xue, John C.; Zhang, Haichao; Humerickhouse, Rod A.; Rosenberg, Saul H.; Elmore, Steven W.
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Design, synthesis, and biological activity of 5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one-based potent and selective Chk-1 inhibitors
err2007-07-21
err49
PREAI
errWang, Le; Sullivan, Gerard M.; Hexamer, Laura A.; Hasvold, Lisa A.; Thalji, Reema; Przytulinska, Magdalena; Tao, Zhi-Fu; Li, Gaoquan; Chen, Zehan; Xiao, Zhan; Gu, Wen-Zhen; Xue, John; Bui, Mai-Ha; Merta, Philip; Kovar, Peter; Bouska, Jennifer J.; Zhang, Haiying; Park, Chang; Stewart, Kent D.; Sham, Hing L.; Sowin, Thomas J.; Rosenberg, Saul H.; Lin, Nan-Horng
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Selective Chk1 inhibitors differentially sensitize p53-deficient cancer cells to cancer therapeutics
err2006-10-26
err126
errOAAI
errChen, Zehan; Xiao, Zhan; Gul, Wen-zhen; Xue, John; Bui, Mai H.; Kovar, Peter; Li, Gaoquan; Wang, Gary; Tao, Zhi-Fu; Tong, Yunsong; Lin, Nan-Horng; Sham, Hing L.; Wang, Jean Y. J.; Sowin, Thomas J.; Rosenberg, Saul H.; Zhang, Haiying
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Novel indication for cancer therapy: Chk1 inhibition sensitizes tumor cells to antimitotics
err2005-04-18
err48
PREAI
errXiao, Z; Xue, J; Semizarov, D; Sowin, TJ; Rosenberg, SH; Zhang, HY
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A novel mechanism of checkpoint abrogation conferred by Chk1 downregulation
err2004-12-20
err99
PREAI
errXiao, Z; Xue, J; Sowin, TJ; Rosenberg, SH; Zhang, HY
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