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Thomas P. Roddy

bristol-myers squibb

36H指数
157论文数
5.2K被引数
收录论文 52
发表时间
ATV-1601 is a Potent and Selective Allosteric Inhibitor of AKT1-E17K and Shows Profound and Durable Regressions in AKT1-E17K-Driven Patient Derived Xenograft Models
err2024-10-01
err0
PREAI
errSchinzel, A. C.; Coffin, A.; Pham, T.; Brigham, B.; Iantosca, G.; Govindaraj, R.; LaPointe, J.; Prescott-Roy, J.; Church, D.; Murray, G.; Roddy, T.; Padyana, A. K.; Dorsch, M.; Sengupta, S.; Blanco, M. J.
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ACLY and ACSS2 link nutrient-dependent chromatin accessibility to CD8 T cell effector responses
err2024-08-16
err0
PREAI
errKaymak, Irem; Watson, McLane J.; Oswald, Brandon M.; Ma, Shixin; Johnson, Benjamin K.; Decamp, Lisa M.; Mabvakure, Batsirai M.; Luda, Katarzyna M.; Ma, Eric H.; Lau, Kin; Fu, Zhen; Muhire, Brejnev; Kitchen-Goosen, Susan M.; Vander Ark, Alexandra; Dahabieh, Michael S.; Samborska, Bozena; Vos, Matthew; Shen, Hui; Fan, Zi Peng; Roddy, Thomas P.; Kingsbury, Gillian A.; Sousa, Cristovao M.; Krawczyk, Connie M.; Williams, Kelsey S.; Sheldon, Ryan D.; Kaech, Susan M.; Roy, Dominic G.; Jones, Russell G.
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13C metabolite tracing reveals glutamine and acetate as critical in vivo fuels for CD8 T cells
err2024-05-31
err6
errOAAI
errMa, Eric H.; Dahabieh, Michael S.; Decamp, Lisa M.; Kaymak, Irem; Kitchen-Goosen, Susan M.; Oswald, Brandon M.; Longo, Joseph; Roy, Dominic G.; Verway, Mark J.; Johnson, Radia M.; Samborska, Bozena; Duimstra, Lauren R.; Scullion, Catherine A.; Steadman, Mya; Vos, Matthew; Roddy, Thomas P.; Krawczyk, Connie M.; Williams, Kelsey S.; Sheldon, Ryan D.; Jones, Russell G.
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Identifying functional allosteric binding sites using a systematic and scalable AMPS screening platform for drug discovery
err2023-12-01
err0
PREAI
errPadyana, Anil K.; Schinzel, Anna; Murray, Gordon; LaPointe, Joseph H.; Selmer, Kaitlyn; Truc Pham; Buskes, Melissa J.; Sengupta, Shomit; Blanco, Maria-Jesus; Roddy, Thomas; Dorsch, Marion
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Itaconate confers tolerance to late NLRP3 inflammasome activation
err2021-03-01
err144
errOAAI
errBambouskova, Monika; Potuckova, Lucie; Paulenda, Tomas; Kerndl, Martina; Mogilenko, Denis A.; Lizotte, Kate; Swain, Amanda; Hayes, Sebastian; Sheldon, Ryan D.; Kim, Hyeryun; Kapadnis, Unnati; Ellis, Abigail E.; Isaguirre, Christine; Burdess, Samantha; Laha, Anwesha; Amarasinghe, Gaya K.; Chubukov, Victor; Roddy, Thomas P.; Diamond, Michael S.; Jones, Russell G.; Simons, Donald M.; Artyomov, Maxim N.
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Rapid, Selective, and Sensitive Method for Semitargeted Discovery of Congeneric Natural Products by Liquid Chromatography Tandem Mass Spectrometry
err2021-02-01
err0
PREAI
errHerath, Kithsiri B.; Previs, Stephen F.; Roddy, Thomas P.; Attygalle, Athula B.; Gonzalez, Ignacio; Genilloud, Olga; Singh, Sheo B.
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Preclinical toxicology profile of squalene epoxidase inhibitors
err2020-08-01
err20
PREAI
errNagaraja, Raj; Olaharski, Andrew; Narayanaswamy, Rohini; Mahoney, Christopher; Pirman, David; Gross, Stefan; Roddy, Thomas P.; Popovici-Muller, Janeta; Smolen, Gromoslaw A.; Silverman, Lee
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Comparative evaluation of itaconate and its derivatives reveals divergent inflammasome and type I interferon regulation in macrophages
err2020-05-25
err200
errOAAI
errSwain, Amanda; Bambouskova, Monika; Kim, Hyeryun; Andhey, Prabhakar Sairam; Duncan, Dustin; Auclair, Karine; Chubukov, Victor; Simons, Donald M.; Roddy, Thomas P.; Stewart, Kelly M.; Artyomov, Maxim N.
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Methionine Metabolism Shapes T Helper Cell Responses through Regulation of Epigenetic Reprogramming蛋氨酸代谢通过调控表观遗传重编程塑造T辅助细胞反应
err2020-02-01
err208
errOAAI
errRoy, Dominic G.; Chen, Jocelyn; Mamane, Victoria; Ma, Eric H.; Muhire, Brejnev M.; Sheldon, Ryan D.; Shorstova, Tatiana; Koning, Rutger; Johnson, Radia M.; Esaulova, Ekaterina; Williams, Kelsey S.; Hayes, Sebastian; Steadman, Mya; Samborska, Bozena; Swain, Amanda; Daigneault, Audrey; Chubukov, Victor; Roddy, Thomas P.; Foulkes, William; Pospisilik, J. Andrew; Bourgeois-Daigneault, Marie-Claude; Artyomov, Maxim N.; Witcher, Michael; Krawczyk, Connie M.; Larochelle, Catherine; Jones, Russell G.
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Metabolic Profiling Using Stable Isotope Tracing Reveals Distinct Patterns of Glucose Utilization by Physiologically Activated CD8+ T Cells使用稳定同位素示踪的代谢分析揭示了生理激活的CD8 T细胞对葡萄糖利用的不同模式
errIMMUNITY
IF26.3
err2019-11-01
err447
errOAAI
errMa, Eric H.; Verway, Mark J.; Johnson, Radia M.; Roy, Dominic G.; Steadman, Mya; Hayes, Sebastian; Williams, Kelsey S.; Sheldon, Ryan D.; Samborska, Bozena; Kosinski, Penelope A.; Kim, Hyeryun; Griss, Takla; Faubert, Brandon; Condotta, Stephanie A.; Krawczyk, Connie M.; DeBerardinis, Ralph J.; Stewart, Kelly M.; Richer, Martin J.; Chubukov, Victor; Roddy, Thomas P.; Jones, Russell G.
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Inhibition of mutant IDH enzymes reduces production of 2-HG but does not restore wild type IDH activity in vitro or in vivo
err2019-07-01
err1
PREAI
errSellers, Katie; Sieger, Taryn; Ronseaux, Sebastien; Narayanaswamy, Rohini; Hudson, Christine; Roddy, Thomas; Nicolay, Brandon
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A chemical biology screen identifies a vulnerability of neuroendocrine cancer cells to SQLE inhibition化学生物学筛选确定了神经内分泌癌细胞对SQLE抑制的脆弱性
err2019-01-09
err66
errOAAI
errMahoney, Christopher E.; Pirman, David; Chubukov, Victor; Sleger, Taryn; Hayes, Sebastian; Fan, Zi Peng; Allen, Eric L.; Chen, Ying; Huang, Lingling; Liu, Meina; Zhang, Yingjia; McDonald, Gabrielle; Narayanaswamy, Rohini; Choe, Sung; Chen, Yue; Gross, Stefan; Cianchetta, Giovanni; Padyana, Anil K.; Murray, Stuart; Liu, Wei; Marks, Kevin M.; Murtie, Joshua; Dorsch, Marion; Jin, Shengfang; Nagaraja, Nelamangala; Biller, Scott A.; Roddy, Thomas; Popovici-Muller, Janeta; Smolen, Gromoslaw A.
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Relation of plasma ceramides to visceral adiposity, insulin resistance and the development of type 2 diabetes mellitus: the Dallas Heart Study
err2018-08-29
err67
errOAAI
errNeeland, Ian J.; Singh, Shruti; McGuire, Darren K.; Vega, Gloria L.; Roddy, Thomas; Reilly, Dermot F.; Castro-Perez, Jose; Kozlitina, Julia; Scherer, Philipp E.
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A chemical biology screen identifies a unique vulnerability of neuroendocrine cancer cells to SQLE inhibition化学生物学筛选确定了神经内分泌癌细胞对SQLE抑制的独特脆弱性
err2018-07-01
err0
PREAI
errMahoney, Christopher; Pirman, David; Chubukov, Victor; Sleger, Taryn; Padyana, Anil; Gross, Stefan; Hayes, Sebastian; Fan, Zi Peng; McDonald, Gabrielle; Chen, Yu; Murtie, Joshua; Cianchetta, Giovanni; Nagaraja, Raj; Narayanaswamy, Rohini; Choe, Sung; Murray, Stuart; Jin, Shengfang; Biller, Scott; Roddy, Thomas; Smolen, Gromoslaw A.
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Enhancing Studies of Pharmacodynamic Mechanisms via Measurements of Metabolic Flux: Fundamental Concepts and Guiding Principles for Using Stable Isotope Tracers
err2017-10-01
err10
errOAAI
errDaurio, Natalie A.; Wang, Sheng-Ping; Chen, Ying; Zhou, Haihong; McLaren, David G.; Roddy, Thomas P.; Johns, Douglas G.; Milot, Denise; Kasumov, Takhar; Erion, Mark D.; Kelley, David E.; Previs, Stephen F.
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CETP (Cholesteryl Ester Transfer Protein) Inhibition With Anacetrapib Decreases Production of Lipoprotein(a) in Mildly Hypercholesterolemic Subjects
err2017-09-01
err69
errOAAI
errThomas, Tiffany; Zhou, Haihong; Karmally, Wahida; Ramakrishnan, Rajasekhar; Holleran, Stephen; Liu, Yang; Jumes, Patricia; Wagner, John A.; Hubbard, Brian; Previs, Stephen F.; Roddy, Thomas; Johnson-Levonas, Amy O.; Gutstein, David E.; Marcovina, Santica M.; Rader, Daniel J.; Ginsberg, Henry N.; Millar, John S.; Reyes-Soffer, Gissette
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Plasma Levels of Risk-Variant APOL1 Do Not Associate with Renal Disease in a Population-Based Cohort
err2016-03-22
err59
errOAAI
errKozlitina, Julia; Zhou, Haihong; Brown, Patricia N.; Rohm, Rory J.; Pan, Yi; Ayanoglu, Gulesi; Du, Xiaoyan; Rimmer, Eric; Reilly, Dermot F.; Roddy, Thomas P.; Cully, Doris F.; Vogt, Thomas F.; Blom, Daniel; Hoek, Maarten
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Evaluation of CETP activity in vivo under non-steady-state conditions: influence of anacetrapib on HDL-TG flux
err2016-03-01
err12
errOAAI
errMcLaren, David G.; Previs, Stephen F.; Phair, Robert D.; Stout, Steven J.; Xie, Dan; Chen, Ying; Salituro, Gino M.; Xu, Suoyu S.; Castro-Perez, Jose M.; Opiteck, Gregory J.; Akinsanya, Karen O.; Cleary, Michele A.; Dansky, Hayes M.; Johns, Douglas G.; Roddy, Thomas P.
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Discovery of Novel Allosteric Non-Bisphosphonate Inhibitors of Farnesyl Pyrophosphate Synthase by Integrated Lead Finding
err2015-09-18
err28
errOAAI
errMarzinzik, Andreas L.; Amstutz, Rene; Bold, Guido; Bourgier, Emmanuelle; Cotesta, Simona; Glickman, J. Fraser; Goette, Marjo; Henry, Christelle; Lehmann, Sylvie; Hartwieg, J. Constanze D.; Ofner, Silvio; Pelle, Xavier; Roddy, Thomas P.; Rondeau, Jean-Michel; Stauffer, Frederic; Stout, Steven J.; Widmer, Armin; Zimmermann, Johann; Zoller, Thomas; Jahnke, Wolfgang
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