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Identification of the Allosteric Binding Site for Thiazolopyrimidine on the C-Type Lectin Langerin 鉴定噻唑并嘧啶在C型凝集素Langerin上的变构结合位点 Zhang, Hengxi; Modenutti, Carlos; Nekkanti, Yelha Phani Kumar; Denis, Maxime; Bermejo, Iris A.; Lefebre, Jonathan; Che, Kateryna; Kim, Dongyoon; Kagelmacher, Marten; Kurzbach, Dennis; Nazare, Marc; Rademacher, Christoph 分享 收藏
Targeting undruggable carbohydrate recognition sites through focused fragment library design Shanina, Elena; Kuhaudomlarp, Sakonwan; Siebs, Eike; Fuchsberger, Felix F.; Denis, Maxime; da Silva Figueiredo Celestino Gomes, Priscila; Clausen, Mads H.; Seeberger, Peter H.; Rognan, Didier; Titz, Alexander; Imberty, Anne; Rademacher, Christoph 分享 收藏
Drug-like Inhibitors of DC-SIGN Based on a Quinolone Scaffold Zhang, Hengxi; Danek, Ondrej; Makarov, Dmytro; Radl, Stanislav; Kim, Dongyoon; Ledvinka, Jiri; Vychodilova, Kristyna; Hlavac, Jan; Lefebre, Jonathan; Denis, Maxime; Rademacher, Christoph; Menova, Petra 分享 收藏
Automated Laser-Transfer Synthesis of High-Density Microarrays for Infectious Disease Screening Paris, Grigori; Heidepriem, Jasmin; Tsouka, Alexandra; Liu, Yuxin; Mattes, Daniela S.; Pinzon Martin, Sandra; Dallabernardina, Pietro; Mende, Marco; Lindner, Celina; Wawrzinek, Robert; Rademacher, Christoph; Seeberger, Peter H.; Breitling, Frank; Bischoff, Frank Ralf; Wolf, Timo; Loeffler, Felix F. 分享 收藏
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A Remote Secondary Binding Pocket Promotes Heteromultivalent Targeting of DC-SIGN Wawrzinek, Robert; Wamhoff, Eike-Christian; Lefebre, Jonathan; Rentzsch, Mareike; Bachem, Gunnar; Domeniconi, Gary; Schulze, Jessica; Fuchsberger, Felix F.; Zhang, Hengxi; Modenutti, Carlos; Schnirch, Lennart; Marti, Marcelo A.; Schwardt, Oliver; Braeutigam, Maria; Guberman, Monica; Hauck, Dirk; Seeberger, Peter H.; Seitz, Oliver; Titz, Alexander; Ernst, Beat; Rademacher, Christoph 分享 收藏
Specific Protein Antigen Delivery to Human Langerhans Cells in Intact Skin Rentzsch, Mareike; Wawrzinek, Robert; Zelle-Rieser, Claudia; Strandt, Helen; Bellmann, Lydia; Fuchsberger, Felix F.; Schulze, Jessica; Busmann, Jil; Rademacher, Juliane; Sigl, Stephan; Del Frari, Barbara; Stoitzner, Patrizia; Rademacher, Christoph 分享 收藏
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Non-Carbohydrate Glycomimetics as Inhibitors of Calcium(II)-Binding Lectins 非碳水化合物模拟糖作为钙 (II) 结合凝集素的抑制剂 Kuhaudomlarp, Sakonwan; Siebs, Eike; Shanina, Elena; Topin, Jeremie; Joachim, Ines; Gomes, Priscila da Silva Figueiredo Celestino; Varrot, Annabelle; Rognan, Didier; Rademacher, Christoph; Imberty, Anne; Titz, Alexander 分享 收藏
Impact of Glycan Linkage to Staphylococcus aureus Wall Teichoic Acid on Langerin Recognition and Langerhans Cell Activation 糖链与金黄色葡萄球菌壁磷壁酸对朗格蛋白识别和朗格汉斯细胞活化的影响 Hendriks, Astrid; van Dalen, Rob; Ali, Sara; Gerlach, David; van der Marel, Gijsbert A.; Fuchsberger, Felix F.; Aerts, Piet C.; de Haas, Carla J. C.; Peschel, Andreas; Rademacher, Christoph; van Strijp, Jos A. G.; Codee, Jeroen D. C.; van Sorge, Nina M. 分享 收藏
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Notch-Mediated Generation of Monocyte-Derived Langerhans Cells: Phenotype and Function Bellmann, Lydia; Zelle-Rieser, Claudia; Milne, Paul; Resteu, Anastasia; Tripp, Christoph H.; Hermann-Kleiter, Natascha; Zaderer, Viktoria; Wilflingseder, Doris; Hoertnagl, Paul; Theochari, Maria; Schulze, Jessica; Rentzsch, Mareike; Del Frari, Barbara; Collin, Matthew; Rademacher, Christoph; Romani, Nikolaus; Stoitzner, Patrizia 分享 收藏
From Pyrazolones to Azaindoles: Evolution of Active-Site SHP2 Inhibitors Based on Scaffold Hopping and Bioisosteric Replacement Mostinski, Yelena; Heynen, Guus J. J. E.; Lopez-Alberca, Maria Pascual; Paul, Jerome; Miksche, Sandra; Radetzki, Silke; Schaller, David; Shanina, Elena; Seyffarth, Carola; Kolomeets, Yuliya; Ziebart, Nandor; de Schryver, Judith; Oestreich, Sylvia; Neuenschwander, Martin; Roske, Yvette; Heinemann, Udo; Rademacher, Christoph; Volkamer, Andrea; von Kries, Jens Peter; Birchmeier, Walter; Nazare, Marc 分享 收藏