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收藏Structural determinants of the catalytic mechanism of Plasmodium CCT, a key enzyme of malaria lipid biosynthesis
Guca, Ewelina; Nagy, Gergely N.; Hajdu, Fanni; Marton, Livia; Izrael, Richard; Hoh, Francois; Yang, Yinshan; Vial, Henri; Vertessy, Beata G.; Guichou, Jean-Francois; Cerdan, Rachel
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收藏High Accumulation and In Vivo Recycling of the New Antimalarial Albitiazolium Lead to Rapid Parasite Death
Wein, Sharon; Taudon, Nicolas; Maynadier, Marjorie; van Ba, Christophe Tran; Margout, Delphine; Bordat, Yann; Fraisse, Laurent; Wengelnik, Kai; Cerdan, Rachel; Bressolle-Gomeni, Francoise; Vial, Henri J.
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收藏Hydroxyl Ketone-Based Histone Deacetylase Inhibitors To Gain Insight into Class I HDAC Selectivity versus That of HDAC6
Traore, Mohamed D. M.; Zwick, Vincent; Simoes-Pires, Claudia A.; Nurisso, Alessandra; Issa, Mark; Cuendet, Muriel; Maynadier, Marjorie; Wein, Sharon; Vial, Henri; Jamet, Helene; Wong, Yung-Sing
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收藏SC83288 is a clinical development candidate for the treatment of severe malaria (vol 8, 14193, 2017)
Pegoraro, Stefano; Duffey, Maelle; Otto, Thomas D.; Wang, Yulin; Rosemann, Roman; Baumgartner, Roland; Fehler, Stefanie K.; Lucantoni, Leonardo; Avery, Vicky M.; Moreno-Sabater, Alicia; Mazier, Dominique; Vial, Henri J.; Strobl, Stefan; Sanchez, Cecilia P.; Lanzer, Michael
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收藏SC83288 is a clinical development candidate for the treatment of severe malaria
Pegoraro, Stefano; Duffey, Maelle; Otto, Thomas D.; Wang, Yulin; Roesemann, Roman; Baumgartner, Roland; Fehler, Stefanie K.; Lucantoni, Leonardo; Avery, Vicky M.; Moreno-Sabater, Alicia; Mazier, Dominique; Vial, Henri J.; Strobl, Stefan; Sanchez, Cecilia P.; Lanzer, Michael
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收藏Synthesis of an Uncharged Tetra-cyclopeptide Acting as a Transmennbrane Carrier: Enhanced Cellular and Nuclear Uptake
Hilario, Flaviane Francisco; Traore, Mohamed Dit Mady; Zwick, Vincent; Berry, Laurence; Simoes-Pires, Claudia A.; Cuendet, Muriel; Fantozzi, Nicolas; de Freitas, Rossimiriam Pereira; Maynadier, Marjorie; Wein, Sharon; Vial, Henri; Wong, Yung-Sing
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收藏Composite Aromatic Boxes for Enzymatic Transformations of Quaternary Ammonium Substrates (vol 53, pg 13471, 2014)
Nagy, Gergely N.; Marton, Livia; Contet, Alicia; Ozohanics, Oliver; Ardelean, Laura-Mihaela; Revesz, Agnes; Vekey, Karoly; Irimie, Florin Dan; Vial, Henri; Cerdan, Rachel; Vertessy, Beata G.
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收藏Composite Aromatic Boxes for Enzymatic Transformations of Quaternary Ammonium Substrates
Nagy, Gergely N.; Marton, Livia; Contet, Alicia; Ozohanics, Oliver; Ardelean, Laura-Mihaela; Revesz, Agnes; Vekey, Karoly; Irimie, Florin Dan; Vial, Henri; Cerdan, Rachel; Vertessy, Beata G.
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收藏Discovery of Compounds Blocking the Proliferation of Toxoplasma gondii and Plasmodium falciparum in a Chemical Space Based on Piperidinyl-Benzimidazolone Analogs
Saidani, Nadia; Botte, Cyrille Y.; Deligny, Michael; Bonneau, Anne-Laure; Reader, Janette; Lasselin, Ronald; Merer, Goulven; Niepceron, Alisson; Brossier, Fabien; Cintrat, Jean-Christophe; Rousseau, Bernard; Birkholtz, Lyn-Marie; Cesbron-Delauw, Marie-France; Dubremetz, Jean-Franois; Mercier, Corinne; Vial, Henri; Lopez, Roman; Marechala, Eric
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收藏Evolutionary and mechanistic insights into substrate and product accommodation of CTP:phosphocholine cytidylyltransferase from Plasmodiumfalciparum
Nagy, Gergely N.; Marton, Livia; Kramos, Balazs; Olah, Julianna; Revesz, Agnes; Vekey, Karoly; Delsuc, Frederic; Hunyadi-Gulyas, Eva; Medzihradszky, Katalin F.; Lavigne, Marina; Vial, Henri; Cerdan, Rachel; Vertessy, Beata G.
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收藏Flexible Synthesis and Evaluation of Diverse Anti-Apicomplexa Cyclic Peptides
Traore, Mariam; Mietton, Flore; Maubon, Daniele; Peuchmaur, Marine; Hilario, Flaviane Francisco; de Freitas, Rossimiriam Pereira; Bougdour, Alexandre; Curt, Aurelie; Maynadier, Marjorie; Vial, Henri; Pelloux, Herve; Hakimi, Mohamed-Ali; Wong, Yung-Sing
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收藏Biochemical characterization of Plasmodium falciparum CTP:phosphoethanolamine cytidylyltransferase shows that only one of the two cytidylyltransferase domains is active
Maheshwari, Sweta; Lavigne, Marina; Contet, Alicia; Alberge, Blandine; Pihan, Emilie; Kocken, Clemens; Wengelnik, Kai; Douguet, Dominique; Vial, Henri; Cerdan, Rachel
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收藏New Bis-thiazolium Analogues as Potential Antimalarial Agents: Design, Synthesis, and Biological Evaluation
Caldarelli, Sergio A.; El Fangour, Siham; Wein, Sharon; van Ba, Christophe Tran; Perigaud, Christian; Pellet, Alain; Vial, Henri J.; Peyrottes, Suzanne
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收藏Antimalarial and anticancer activities of artemisinin-quinoline hybrid-dimers and pharmacokinetic properties in mice青蒿素-喹啉杂化二聚体的抗疟和抗癌活性及其在小鼠中的药代动力学特性
Lombard, Marli C.; N'Da, David D.; Breytenbach, Jaco C.; Kolesnikova, Natasha I.; Van Ba, Christophe Tran; Wein, Sharon; Norman, Jennifer; Denti, Paolo; Vial, Henri; Wiesner, Lubbe
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