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Robert A. Reamer

merck & company

49H指数
401论文数
7.8K被引数
收录论文 95
发表时间
Practical Asymmetric Synthesis of a Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonist Ubrogepant
err2017-11-02
err29
PREAI
errYasuda, Nobuyoshi; Cleator, Ed; Kosjek, Birgit; Yin, Jianguo; Xiang, Bangping; Chen, Frank; Kuo, Shen-Chun; Belyk, Kevin; Mullens, Peter R.; Goodyear, Adrian; Edwards, John S.; Bishop, Brian; Ceglia, Scott; Belardi, Justin; Tan, Lushi; Song, Zhiguo J.; DiMichele, Lisa; Reamer, Robert; Cabiro, Fabien L.; Tang, Weng Lin; Liu, Guiquan
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Asymmetric Formal Synthesis of the Long-Acting DPP-4 Inhibitor Omarigliptin
err2017-08-14
err19
errOAAI
errPeng, Feng; Chen, Yonggang; Chen, Cheng-yi; Dormer, Peter G.; Kassim, Amude; McLaughlin, Mark; Reamer, Robert A.; Sherer, Edward C.; Song, Zhiguo J.; Tan, Lushi; Tudge, Matthew T.; Wan, Baoqiang; Chung, John Y. L.
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Enantioselective Synthesis of 4′-Ethynyl-2-fluoro-2′-deoxyadenosine (EFdA) via Enzymatic Desymmetrization
err2017-02-06
err51
PREAI
errMcLaughlin, Mark; Kong, Jongrock; Belyk, Kevin M.; Chen, Billy; Gibson, Andrew W.; Keen, Stephen P.; Lieberman, David R.; Milczek, Erika M.; Moore, Jeffrey C.; Murray, David; Peng, Feng; Qi, Ji; Reamer, Robert A.; Song, Zhiguo J.; Tan, Lushi; Wang, Lin; Williams, Michael J.
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Promotion of a Ti-Mediated Mannich Reaction by a Proton Source
err2015-12-21
err1
PREAI
errLimanto, John; Yoshikawa, Naoki; Reamer, Robert A.; Tan, Lushi; Brunskill, Andrew; Reibarkh, Mikhail
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Careful Navigation of the Crystallographic Landscape of MK-8970: A Racemic Acetal Carbonate Prodrug of Raltegravir
err2015-06-19
err1
PREAI
errTsou, Nancy; Shultz, C. Scott; Andreani, Teresa; Ball, Richard G.; Brunskill, Andrew; Balsells, Jaume; Cohen, Ryan D.; DaSilva, Jimmy; Li, Jing; Reamer, Robert A.; Ruiz, Manuel de Lera; Variankaval, Narayan; Varsolona, Richard J.; Yasuda, Nobuyoshi; York, Gregory
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N-Boc Deprotection and Isolation Method for Water-Soluble Zwitterionic Compounds
err2014-11-18
err21
PREAI
errLiu, Zhijian; Yasuda, Nobuyoshi; Simeone, Michael; Reamer, Robert A.
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Unusual Pyrimidine Participation: Efficient Stereoselective Synthesis of Potent Dual Orexin Receptor Antagonist MK-6096
err2014-11-03
err15
PREAI
errChung, John Y. L.; Zhong, Yong-Li; Maloney, Kevin M.; Reamer, Robert A.; Moore, Jeffrey C.; Strotman, Hallena; Kalinin, Alexei; Feng, Ronnie; Strotman, Neil A.; Xiang, Bangping; Yasuda, Nobuyoshi
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Discovery and Application of Doubly Quaternized Cinchona-Alkaloid-Based Phase-Transfer Catalysts
err2014-06-24
err71
PREAI
errXiang, Bangping; Belyk, Kevin M.; Reamer, Robert A.; Yasuda, Nobuyoshi
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Enantioselective Synthesis of an HCV NS5a Antagonist
err2014-04-11
err63
PREAI
errMangion, Ian K.; Chen, Cheng-yi; Li, Hongmei; Maligres, Peter; Chen, Yonggang; Christensen, Melodie; Cohen, Ryan; Jeon, Ingyu; Klapars, Artis; Krska, Shane; Hoa Nguyen; Reamer, Robert A.; Sherry, Benjamin D.; Zavialov, Ilia
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Practical Asymmetric Synthesis of a Chiral Piperazinone Derivative
err2013-07-31
err26
PREAI
errMcLaughlin, Mark; Belyk, Kevin; Chen, Cheng-yi; Xin Linghu; Jun Pan; Gang Qian; Reamer, Robert A.; Xu, Yingju
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Synthesis of α-Hydroxyacetophenones
err2012-05-22
err15
PREAI
errMcLaughlin, Mark; Belyk, Kevin M.; Qian, Gang; Reamer, Robert A.; Chen, Cheng-yi
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Synthesis of Antifungal Glucan Synthase Inhibitors from Enfumafungin
err2012-03-28
err20
PREAI
errZhong, Yong-Li; Gauthier, Donald R., Jr.; Shi, Yao-Jun; McLaughlin, Mark; Chung, John Y. L.; Dagneau, Philippe; Marcune, Benjamin; Krska, Shane W.; Ball, Richard G.; Reamer, Robert A.; Yasuda, Nobuyoshi
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Synthesis of Vaniprevir (MK-7009): Lactamization To Prepare a 22-Membered Macrocycle (vol 76, pg 7804, 2011)
err2011-10-19
err3
errOAAI
errSong, Zhiguo J.; Tellers, David M.; Journet, Michel; Kuethe, Jeffrey T.; Lieberman, David; Humphrey, Guy; Zhang, Fei; Peng, Zhihui; Waters, Marjorie S.; Zewge, Daniel; Nolting, Andrew; Zhao, Dalian; Reamer, Robert A.; Dormer, Peter G.; Belyk, Kevin M.; Davies, Ian W.; Devine, Paul N.; Tschaen, David M.
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Synthesis of Vaniprevir (MK-7009): Lactamization To Prepare a 22-Membered Macrocycle
err2011-08-31
err52
PREAI
errSong, Zhiguo J.; Tellers, David M.; Journet, Michel; Kuethe, Jeffrey T.; Lieberman, David; Humphrey, Guy; Zhang, Fei; Peng, Zhihui; Waters, Marjorie S.; Zewge, Daniel; Nolting, Andrew; Zhao, Dalian; Reamer, Robert A.; Dormer, Peter G.; Belyk, Kevin M.; Davies, Ian W.; Devine, Paul N.; Tschaen, David M.
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Reaction Development and Mechanistic Study of a Ruthenium Catalyzed Intramolecular Asymmetric Reductive Amination en Route to the Dual Orexin Inhibitor Suvorexant (MK-4305)
err2011-05-11
err99
PREAI
errStrotman, Neil A.; Baxter, Carl A.; Brands, Karel M. J.; Cleator, Ed; Krska, Shane W.; Reamer, Robert A.; Wallace, Debra J.; Wright, Timothy J.
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The First Large-Scale Synthesis of MK-4305: A Dual Orexin Receptor Antagonist for the Treatment of Sleep Disorder
err2011-03-04
err114
PREAI
errBaxter, Carl A.; Cleator, Ed; Brands, Karel M. J.; Edwards, John S.; Reamer, Robert A.; Sheen, Faye J.; Stewart, Gavin W.; Strotman, Neil A.; Wallace, Debra J.
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Development of a Second-Generation, Highly Efficient Manufacturing Route for the HIV Integrase Inhibitor Raltegravir Potassium
err2010-11-16
err49
PREAI
errHumphrey, Guy R.; Pye, Philip J.; Zhong, Yong-Li; Angelaud, Remy; Askin, David; Belyk, Kevin M.; Maligres, Peter E.; Mancheno, Danny E.; Miller, Ross A.; Reamer, Robert A.; Weissman, Steven A.
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Practical Synthesis of Functionalized 1,5-Disubstituted 1,2,4-Triazole Derivatives
err2010-11-16
err34
PREAI
errXu, Yingju; McLaughlin, Mark; Bolton, Emily N.; Reamer, Robert A.
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A General Method for the Synthesis of 3,5-Diarylcyclopentenones via Friedel-Crafts Acylation of Vinyl Chlorides
err2009-06-01
err18
PREAI
errXu, Yingju; McLaughlin, Mark; Chen, Cheng-yi; Reamer, Robert A.; Dormer, Peter G.; Davies, Ian W.
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