未登录Pembrolizumab microgravity crystallization experimentationPembrolizumab微重力结晶实验
Reichert, Paul; Prosise, Winifred; Fischmann, Thierry O.; Scapin, Giovanna; Narasimhan, Chakravarthy; Spinale, April; Polniak, Ray; Yang, Xiaoyu; Walsh, Erika; Patel, Daya; Benjamin, Wendy; Welch, Johnathan; Simmons, Denarra; Strickland, Corey
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收藏Discovery of Novel 3,3-Disubstituted Piperidines as Orally Bioavailable, Potent, and Efficacious HDM2-p53 Inhibitors
Bogen, Stephane L.; Pan, Weidong; Gibeau, Craig R.; Lahue, Brian R.; Ma, Yao; Nair, Latha G.; Seigel, Elise; Shipps, Gerald W., Jr.; Tian, Yuan; Wang, Yaolin; Lin, Yinghui; Liu, Ming; Liu, Suxing; Mirza, Asra; Wang, Xiaoying; Lipar, Philip; Seidel-Dugan, Cynthia; Hicklin, Daniel J.; Bishop, W. Robert; Rindgen, Diane; Nomeir, Amin; Prosise, Winifred; Reichert, Paul; Scapin, Giovanna; Strickland, Corey; Doll, Ronald J.
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收藏Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core
Yu, Tao; Tagat, Jayaram R.; Kerekes, Angela D.; Doll, Ronald J.; Zhang, Yonglian; Xiao, Yushi; Esposite, Sara; Belanger, David B.; Curran, Patrick J.; Mandal, Amit K.; Siddiqui, M. Arshad; Shih, Neng-Yang; Basso, Andrea D.; Liu, Ming; Gray, Kimberly; Tevar, Seema; Jones, Jennifer; Lee, Suining; Liang, Lianzhu; Ponery, Samad; Smith, Elizabeth B.; Hruza, Alan; Voigt, Johannes; Ramanathan, Lata; Prosise, Winifred; Hu, Mengwei
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收藏Discovery of the HCVNS3/4A protease inhibitor (1R,5S)-N-[3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[2(S)-[[[(1,1-dimethylethyl)amino]carbonyl]amino]-3,3-dimethyl-1-oxobutyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexan-2(S)-carboxamide (Sch 503034) II.: Key steps in structure-based optimization
Prongay, Andrew J.; Guo, Zhuyan; Yao, Nanhua; Pichardo, John; Fischmann, Thierry; Strickland, Corey; Myers, Joseph, Jr.; Weber, Patricia C.; Beyer, Brian M.; Ingram, Richard; Hong, Zhi; Prosise, Winifred W.; Ramanathan, Lata; Taremi, S. Shane; Yarosh-Tomaine, Taisa; Zhang, Rumin; Senior, Mary; Yang, Rong-Sheng; Malcolm, Bruce; Arasappan, Ashok; Bennett, Frank; Bogen, Stephane L.; Chen, Kevin; Jao, Edwin; Liu, Yi-Tsung; Lovey, Raymond G.; Saksena, Anil K.; Venkatraman, Srikanth; Girijavallabhan, Viyyoor; Njoroge, F. George; Madison, Vincent
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