未登录In vitro and in vivo characterization of novel MAT2A allosteric inhibitors
Pei, Zhonghua; Alam, Muzaffar; Bhola, Neil; Cleary, Leah; Drummond, Jake; Fisher, Marcus; Fleury, Melissa; Garcia, Candy; Givmanesh, Atieh; Xin Linghu; McSpadden, Ethan; Mounir, Zineb; Neilan, Claire; Newby, Zach; Perumal, Senthil; Steel, Richard; Sutton, James; Vaidya, Kedar; Wagle, Marie-Claire; Wang, Jianhong; Yao, Bing; Lackner, Mark; Dillon, Michael P.
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收藏Mat2A Inhibitors decrease growth, increase senescence and p53 stability in MTAP-deleted cancer cells
Bhola, Neil; Givmanesh, Atieh; Wagle, Marie-Claire; Garcia, Candy; Vaidya, Kedar; Cleary, Leah; Pei, Zhonghua; Lackner, Mark; Mounir, Zineb
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收藏PARG inhibitors exhibit synthetic lethality with XRCC1 deficiency and a cellular mechanism of action that is distinct from PARP inhibition
Martin, Leenus; Cheng, Tzuling; James, Dominic I.; Begum, Habiba; Smith, Kate M.; Jordan, Allan; Waddell, Ian; Vaidya, Kedar; Fischer, Marcus; Yao, Bing; Drummond, Jason; Cleary, Leah; Martinez, Ruben; Sutton, James; Ravindran, Nandini; Joseph, James; Venetsanakos, Eleni; Dillon, Michael; Hager, Jeffrey H.; Belmont, Lisa D.
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