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Novel indole-sulfonamide hybrids as α-amylase and α-glucosidase inhibitors: a rational approach combining enzyme kinetics and in silico analysis 新型吲哚-磺酰胺类杂合物作为α-淀粉酶和α-葡萄糖苷酶抑制剂:一种结合酶动力学和计算机模拟分析的合理方法 Taha, Muhammad; Rahim, Fazal; Zada, Hussan; Chigurupati, Sridevi; Imran, Syahrul; Nawaz, Muhammad; Khan, Khalid Mohammed; Ali, Muhammad; Shah, Syed Adnan Ali; Felemban, Shatha Ghazi; Venugopal, Vijayan; Uddin, Nizam 分享 收藏
Synthesis, biological evaluation, molecular dynamic and docking study of benzimidazole analogues as potent acetylcholinesterase and butyrylcholinesterase inhibitors Taha, Muhammad; Rahim, Fazal; Rehman, Hafiz Ur; Imran, Syahrul; Uddin, Nizam; Khan, Khalid Mohammed; Shah, Syed Adnan Ali; Shehzad, Adeeb 分享 收藏
Synthesis, enzyme inhibitory kinetics, & computational studies of N-(substituted phenyl)-(5-(3,4-dichlorobenzyl)-4-(4-chlorophenyl)-4H-1,2,4-triazol-3-ylthio)methylbenzamides: As potent alkaline phosphatase inhibitors Zeb, Aurang; Siddiqui, Sabahat Zahra; Abbasi, Muhammad Athar; Aziz-ur-Rehman; Shah, Syed Adnan Ali; Imran, Syahrul; Raza, Hussain; Kim, Song Ja; Parveen, Riffat; Abbas, Ghazanfar 分享 收藏
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Synthesis of benzimidazole derivatives and their antiglycation, antioxidant, antiurease and molecular docking study 苯并咪唑衍生物的合成及其抗糖基化、抗氧化、抗脲酶和分子对接研究 Taha, Muhammad; Rahim, Fazal; Adalath, Bushra; Imran, Syahrul; Khan, Khalid Mohammed; Shah, Syed Adnan Ali; Uddin, Nizam; Nawaz, Muhammad; Break, Mohammed Khaled Bin; Magam, Sami M.; Alqarni, Saad 分享 收藏
New piperidinyl heterocyclic azoles acquired through Li(I)-catalyzed reactions: Anti-enzymatic, ADME and computational studies Hamid, Sujhla; Amjad, Hira; Abbasi, Muhammad Athar; Siddiqui, Sabahat Zahra; Ashraf, Muhammad; Iqbal, Javed; Farhan, Muhammad; Rasool, Shahid; Shah, Syed Adnan Ali; Imran, Syahrul; Rehman, Muhammad Tjammal; Aziz-ur-Rehman 分享 收藏
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The b-carboline analogs as a potent inhibitor for Alzheimer's Disease, molecular docking and dynamics simulation study Taha, Muhammad; Rahim, Fazal; Khan, Azmat Ali; Adalat, Bushra; Imran, Syahrul; Alshehri, Jamilah M.; Ahmad, Asrar; Khan, Khalid Mohammed; Shah, Syed Adnan Ali; Uddin, Nizam 分享 收藏
Synthesis, in vitro evaluation and molecular docking studies of hybrid 4-quinolinyl bearing 1,3,4-thiadiazole-2-amine as a new inhibitor of ?-amylase and ?-glucosidase Taha, Muhammad; Khan, Aftab Ahmad; Rahim, Fazal; Hayat, Shawkat; Imran, Syahrul; Iqbal, Naveed; Uddin, Nizam; Khan, Khalid Mohammed; Anouar, El Hassane; Farooq, Rai Khalid; Nawaz, Muhammad; Shah, Syed Adnan Ali 分享 收藏
New pyrrolopyridine-based thiazolotriazoles as diabetics inhibitors: enzymatic kinetics and in silico study Taha, Muhammad; Rahim, Fazal; Hayat, Shawkat; Chigurupati, Sridevi; Khand, Khalid Mohammed; Imran, Syahrul; Ali Shah, Syed Adnan; Uddin, Nizam; Felemban, Shatha Ghazi; Venugopal, Vijayan 分享 收藏
In vitro and in silico assessment of bioactivity properties and pharmacokinetic studies of new 3,5-disubstituted-1,2,4-triazoles Amjad, Hira; Abbasi, Muhammad Athar; Siddiqui, Sabahat Zahra; Iqbal, Javed; Rasool, Shahid; Ashraf, Muhammad; Hussain, Safdar; Shah, Syed Adnan Ali; Imran, Syahrul; Shahid, Muhammad; Rasool, Arslan; Rehman, Muhammad Tjammal; ur Rehman, Aziz 分享 收藏
Benzoxazole based thiazole hybrid analogs: Synthesis, in vitro cholinesterase inhibition, and molecular docking studies Hussain, Rafaqat; Rahim, Fazal; Rehman, Wajid; Shah, Syed Adnan Ali; Khan, Shoaib; Khan, Imran; Rasheed, Liaqat; Imran, Syahrul; Wadood, Abdul; Abdellattif, Magda H. 分享 收藏
Discovering biological efficacy of new thiadiazole as effective inhibitors of urease, glycation, and (DPPH) scavengers: Biochemical and in silico study Taha, Muhammad; Imran, Syahrul; Rahim, Fazal; Uddin, Nizam; Iqbal, Naveed; Khan, Khalid Mohammed; Farooq, Rai Khalid; Alomari, Munther; Islam, Imadul; Algheribe, Shatha 分享 收藏
Bio-Oriented Synthesis and Molecular Docking Studies of 1,2,4-Triazole Based Derivatives as Potential Anti-Cancer Agents against HepG2 Cell Line Akhter, Naheed; Batool, Sidra; Khan, Samreen Gul; Rasool, Nasir; Anjum, Fozia; Rasul, Azhar; Adem, Sevki; Mahmood, Sadaf; Rehman, Aziz Ur; Nisa, Mehr Un; Razzaq, Zainib; Christensen, Jorn B.; Abourehab, Mohammed A. S.; Shah, Syed Adnan Ali; Imran, Syahrul 分享 收藏
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Synthesis of new 1,2-disubstituted benzimidazole analogs as potent inhibitors of β-Glucuronidase and in silico study Taha, Muhammad; Khan, Aftab Ahmad; Rahim, Fazal; Imran, Syahrul; Salahuddin, Mohammed; Uddin, Nizam; Khan, Khalid Mohammed; Shah, Syed Adnan Ali; Zafar, Ameeduzzafar; Zakaria, Zainul Amiruddin 分享 收藏