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收藏Highlights from the Mech'cheM 2025 conference: New forces in Mechanochemistry, Montpellier, France, June 4-6, 2025Mech'cheM 2025 会议亮点:机械化学中的新力量,法国蒙彼利埃,2025年6月4日至6日
Bantreil, Xavier; Giani, Olivia; Monconduit, Laure; Petry, Nicolas; Pinaud, Julien; Roy, Beatrice; Lamaty, Frederic
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收藏5-HT6 receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivatives
Drop, Marcin; Koczurkiewicz-Adamczyk, Paulina; Bento, Ophelie; Pietrus, Wojciech; Satala, Grzegorz; Blicharz-Futera, Klaudia; Canale, Vittorio; Grychowska, Katarzyna; Bantreil, Xavier; Pekala, Elzbieta; Kurczab, Rafal; Bojarski, Andrzej J.; Chaumont-Dubel, Severine; Marin, Philippe; Lamaty, Frederic; Zajdel, Pawe l
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收藏Multistep Mechanochemical Synthesis of PZ-1190, a Multitarget Antipsychotic Agent
Canale, Vittorio; Kaminski, Michal; Trybala, Wojciech; Abram, Michal; Marciniec, Krzysztof; Bantreil, Xavier; Lamaty, Frederic; Parkitna, Jan Rodriguez; Zajdel, Pawel
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收藏Superiority of the Triple-Acting 5-HT6R/5-HT3R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT6R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats
Grychowska, Katarzyna; Lopez-Sanchez, Uriel; Vitalis, Mathieu; Canet, Geoffrey; Satala, Grzegorz; Olejarz-Maciej, Agnieszka; Golebiowska, Joanna; Kurczab, Rafal; Pietrus, Wojciech; Kubacka, Monika; Moreau, Christophe; Walczak, Maria; Blicharz-Futera, Klaudia; Bantreil, Xavier; Subra, Gilles; Bojarski, Andrzej J.; Lamaty, Frederic; Becamel, Carine; Zussy, Charleine; Chaumont-Dubel, Severine; Popik, Piotr; Nury, Hugues; Marin, Philippe; Givalois, Laurent; Zajdel, Pawel
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收藏Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT6 and D3R Affinity in the 1H-Pyrrolo[3,2-c]quinoline Series
Grychowska, Katarzyna; Pietrus, Wojciech; Kulawik, Ludmila; Bento, Ophelie; Satala, Grzegorz; Bantreil, Xavier; Lamaty, Frederic; Bojarski, Andrzej J.; Golebiowska, Joanna; Nikiforuk, Agnieszka; Marin, Philippe; Chaumont-Dubel, Severine; Kurczab, Rafal; Zajdel, Pawel
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收藏Advances in synthesis: general discussion
Angerhofer, Alexander; Balaz, Matej; Balema, Viktor; Belenguer, Ana M.; Blair, Richard G.; Boldyreva, Elena; Bolm, Carsten; Borchardt, Lars; Braunschweig, Adam B.; Browne, Duncan L.; Craig, Stephen; El Wenni, Lamis; Emmerling, Franziska; Ferguson, Michael; Fiore, Cecilia; Friscic, Tomislav; Fukushima, Kimichika; Garcia, Felipe; Gonnet, Lori; Gratz, Sven; Hernandez, Rafael A. R.; Ito, Hajime; James, Stuart L.; Karabiyikli, Deniz; Kim, Jeung Gon; Kubota, Koji; Lamaty, Frederic; Lampronti, Giulio, I; Leitch, Jamie; Lukin, Stipe; Mack, James; Maini, Lucia; Mohamed, Sharmarke; Moores, Audrey; Nagapudi, Karthik; Puccetti, Francesco; Tian, Mi; Yu, Qian
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收藏Kinetics and basic understanding: general discussion
Angerhofer, Alexander; Auvray, Thomas; Balema, Viktor; Balaz, Matej; Batteas, James D.; Blair, Richard G.; Boldyreva, Elena; Bolm, Carsten; Borchardt, Lars; Borchers, Tristan H.; Braunschweig, Adam B.; Browne, Duncan L.; Carpick, Robert W.; Ciaccia, Maria; Craig, Stephen; Emmerling, Franziska; Ferguson, Michael; Fiore, Cecilia; Friscic, Tomislav; Gratz, Sven; Halasz, Ivan; Hamzehpoor, Ehsan; Ito, Hajime; James, Stuart; Kim, Jeung Gon; Lamaty, Frederic; Lampronti, Giulio, I; Laurencin, Danielle; Leitch, Jamie; Lu, Erli; Lukin, Stipe; Mack, James; Maini, Lucia; Martini, Ashlie; Mazzeo, Paolo P.; Michalchuk, Adam A. L.; Mittelette, Sebastien; Mohamed, Sharmarke; Moores, Audrey; Mortera-Carbonell, Aldo de Jesus; Nagapudi, Karthik; Niidu, Allan; Puccetti, Francesco; Stahorsky, Martin; Vugrin, Leonarda
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收藏Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 H-pyrrolo-[3,2-c] quinolines
Grychowska, Katarzyna; Olejarz-Maciej, Agnieszka; Blicharz, Klaudia; Pietrus, Wojciech; Karcz, Tadeusz; Kurczab, Rafal; Koczurkiewicz, Paulina; Doroz-Plonka, Agata; Latacz, Gniewomir; Keeri, Abdul Raheem; Piska, Kamil; Satala, Grzegorz; Pegiel, Joanna; Trybala, Wojciech; Jastrzebska-Wiesek, Magdalena; Bojarski, Andrzej J.; Lamaty, Frederic; Partyka, Anna; Walczak, Maria; Krawczyk, Martyna; Malikowska-Racia, Natalia; Popik, Piotr; Zajdel, Pawel
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