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Identification and Optimization of a Ligand-Efficient Benzoazepinone Bromodomain and Extra Terminal (BET) Family Acetyl-Lysine Mimetic into the Oral Candidate Quality Molecule I-BET432 Humphreys, Philip G.; Anderson, Niall A.; Bamborough, Paul; Baxter, Andrew; Chung, Chun-wa; Cookson, Rosa; Craggs, Peter D.; Dalton, Toryn; Fournier, Julie C. L.; Gordon, Laurie J.; Gray, Heather F.; Gray, Matthew W.; Gregory, Richard; Hirst, David J.; Jamieson, Craig; Jones, Katherine L.; Kessedjian, Hripsimee; Lugo, David; McGonagle, Grant; Patel, Vipulkumar K.; Patten, Christopher; Poole, Darren L.; Prinjha, Rab K.; Ramirez-Molina, Cesar; Rioja, Inmaculada; Seal, Gail; Stafford, Kayleigh A. J.; Shah, Rishi R.; Tape, Daniel; Theodoulou, Natalie H.; Tomlinson, Laura; Ukuser, Sabri; Wall, Ian D.; Wellaway, Natalie; White, Gemma 分享 收藏
Cancer-associated fibroblasts require proline synthesis by PYCR1 for the deposition of pro-tumorigenic extracellular matrix (vol 4, pg 639, 2022) Kay, Emily J.; Paterson, Karla; Riera-Domingo, Carla; Sumpton, David; Dabritz, J. Henry M.; Tardito, Saverio; Boldrini, Claudia; Hernandez-Fernaud, Juan R.; Athineos, Dimitris; Dhayade, Sandeep; Stepanova, Ekaterina; Gjerga, Enio; Neilson, Lisa J.; Lilla, Sergio; Hedley, Ann; Koulouras, Grigorios; McGregor, Grace; Jamieson, Craig; Johnson, Radia Marie; Park, Morag; Kirschner, Kristina; Miller, Crispin; Kamphorst, Jurre J.; Loayza-Puch, Fabricio; Saez-Rodriguez, Julio; Mazzone, Massimiliano; Blyth, Karen; Zagnoni, Michele; Zanivan, Sara 分享 收藏
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Cancer-associated fibroblasts require proline synthesis by PYCR1 for the deposition of pro-tumorigenic extracellular matrix 癌症相关的成纤维细胞需要PYCR1合成脯氨酸以沉积促肿瘤发生的细胞外基质 Kay, Emily J.; Paterson, Karla; Riero-Domingo, Carla; Sumpton, David; Dabritz, J. Henry M.; Tardito, Saverio; Boldrini, Claudia; Hernandez-Fernaud, Juan R.; Athineos, Dimitris; Dhayade, Sandeep; Stepanova, Ekaterina; Gjerga, Enio; Neilson, Lisa J.; Lilla, Sergio; Hedley, Ann; Koulouras, Grigorios; McGregor, Grace; Jamieson, Craig; Johnson, Radia Marie; Park, Morag; Kirschner, Kristina; Miller, Crispin; Kamphorst, Jurre J.; Loayza-Puch, Fabricio; Saez-Rodriguez, Julio; Mazzone, Massimiliano; Blyth, Karen; Zagnoni, Michele; Zanivan, Sara 分享 收藏
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Design and Development of a Macrocyclic Series Targeting Phosphoinositide 3-Kinase δ Spencer, Jonathan A.; Baldwin, Ian R.; Barton, Nick; Chung, Chun-Wa; Convery, Maire A.; Edwards, Christopher D.; Jamieson, Craig; Mallett, David N.; Rowedder, James E.; Rowland, Paul; Thomas, Daniel A.; Hardy, Charlotte J. 分享 收藏