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杨财广 封面图

杨财广 (Cai‐Guang Yang)

chinese academy of sciences

44H指数
155论文数
9.5K被引数
收录论文 79
发表时间
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Development of Orally Bioavailable FTO Inhibitors with Potent Antileukemia Efficacy开发具有强效抗白血病活性的口服生物利用度FTO抑制剂
err2025-06-28
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PREAI
errTeng Yang; Ze Dong; Rong Du; Yiqing Wang; Lu Liu; Yangyang Xue; Xi Zhang; Yonggang Liao; Jianhua Gan; Xiaoxuan Yu; Yue Huang; Cai-Guang Yang
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Development of 3-arylaminothiophenic-2-carboxylic acid derivatives as new FTO inhibitors showing potent antileukemia activities
err2025-05-01
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PREAI
errZhang, Deyan; Liu, Lu; Li, Ming; Hu, Xinyi; Zhang, Xi; Xia, Wenyang; Wang, Zhen; Song, Xiaomin; Huang, Yue; Dong, Ze; Yang, Cai-Guang
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Structure-Based Development of a Covalent Inhibitor Targeting Streptococcus Pyogenes over Staphylococcus Aureus Sortase A
err2025-03-01
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PREAI
errZhou, Hailing; Yuan, Ziqi; Guan, Xiang-Na; Yue, Chuan; Wu, Wei; Lan, Lefu; Gan, Jianhua; Zhang, Tao; Yang, Cai-Guang
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Integrative study of lung cancer adeno-to-squamous transition in EGFR TKI resistance identifies RAPGEF3 as a therapeutic target
err2024-11-07
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errWang, Hua; Tang, Shijie; Wu, Qibiao; He, Yayi; Zhu, Weikang; Xie, Xinyun; Qin, Zhen; Wang, Xue; Zhou, Shiyu; Yao, Shun; Xu, Xiaoling; Guo, Chenchen; Tong, Xinyuan; Han, Shuo; Chou, Yueh-Hung; Wang, Yong; Wong, Kwok-Kin; Yang, Cai-Guang; Chen, Luonan; Hu, Liang; Ji, Hongbin
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Synthesis and antibacterial activities of heterocyclic ring-fused 20 (S)-protopanaxadiol derivatives
err2024-10-01
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PREAI
errZhang, De-Jie; Yuan, Zi-Qi; Yue, Yan-Xin; Zhang, Min; Wu, Wen-Juan; Yang, Cai-Guang; Qiu, Wen-Wei
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Expeditious Synthesis of Gwanakoside A and the Chloronaphthol Glycoside Congeners
err2024-03-20
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PREAI
errCheng, Yuting; Xia, Yan; Yuan, Ziqi; Li, Haotian; Wang, Jing; Wang, Yingjie; Yang, Cai-Guang; Yu, Biao
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Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent Staphylococcus aureus Sortase A Inhibitors
err2024-01-03
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PREAI
errYue, Chuan; Yuan, Ziqi; Xu, Guobin; Guan, Xiang-Na; Wei, Bingyan; Yao, Hequan; Yang, Cai-Guang; Zhang, Tao
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A covalent compound selectively inhibits RNA demethylase ALKBH5 rather than FTO
err2024-01-01
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errLai, Gan-Qiang; Li, Yali; Zhu, Heping; Zhang, Tao; Gao, Jing; Zhou, Hu; Yang, Cai-Guang
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Ascorbic Acid Reprograms Epigenome and Epitranscriptome by Reducing Fe(III) in the Catalytic Cycle of Dioxygenases
err2023-12-15
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PREAI
errHe, Weizhi; Yin, Xiaotong; Xu, Chu; Liu, Xiangyue; Huang, Yue; Yang, Caiguang; Xu, Yanhui; Hu, Lulu
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Selective activator of human ClpP triggers cell cycle arrest to inhibit lung squamous cell carcinoma
err2023-11-03
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errOAAI
errZhou, Lin-Lin; Zhang, Tao; Xue, Yun; Yue, Chuan; Pan, Yihui; Wang, Pengyu; Yang, Teng; Li, Meixia; Zhou, Hu; Ding, Kan; Gan, Jianhua; Ji, Hongbin; Yang, Cai-Guang
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Rational Design of RNA Demethylase FTO Inhibitors with Enhanced Antileukemia Drug-Like Properties
err2023-07-07
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PREAI
errXiao, Pan; Duan, Zongliang; Liu, Zeyu; Chen, Liang; Zhang, Deyan; Liu, Lu; Zhou, Chen; Gan, Jianhua; Dong, Ze; Yang, Cai-Guang
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Multi-omics for COVID-19: driving development of therapeutics and vaccines
err2023-05-30
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errOAAI
errGuo, Mengyu; Xiong, Muya; Peng, Jinying; Guan, Tong; Su, Haixia; Huang, Yanyi; Yang, Cai-Guang; Li, Yang; Boraschi, Diana; Pillaiyar, Thanigaimalai; Wang, Guanbo; Yi, Chengqi; Xu, Yechun; Chen, Chunying
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研究方向

基于化学遗传学的原创新药发现研究靶向RNA表观遗传的化学探针与靶标成药性研究小分子靶向性干预线粒体蛋白质稳态抗肿瘤新类型抗生素以及运用“非抗生素效应”抗耐药菌感染