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Pavel K. Mykhailiuk

enamine ltd

48H指数
557论文数
8.2K被引数
收录论文 95
发表时间
Bench-Stable α-Fluoroamines: Synthesis, Properties, and Application in Medicinal Chemistry台架稳定的α-氟代胺:合成、性质及其在药物化学中的应用
err2026-10-07
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PREAI
errVadym Levterov; Oleh Shablykin; Oleksandr Stashkevych; Volodymyr Kokhalskyi; Vadym Konashuk; Iryna Sadkova; Olha Shevchuk; Petro Borysko; Henry S. Rzepa; Pavel K. Mykhailiuk
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A Safe Approach to meta-Fluorinated Pyridines一种制备间氟化吡啶的安全方法
err2026-06-16
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PREAI
errOleksandra Rushchak; Vadym Sham; Bohdan Dansberg; Andrii Kysil; Tetyana Yegorova; Pavel K. Mykhailiuk
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O-Vinylhydroxylamines for De Novo Pyrrole Synthesis乙烯基羟胺用于从头吡咯合成
err2026-05-23
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errOAAI
errCharlotte Randolph; Oleksandr Buravov; Zachary Grimm; Pavel K. Mykhailiuk; László Kürti
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Replacement of the Piperidine Ring with Aza-Spirocycles Reduces Cardiotoxicity of the Local Anesthetic Drug Bupivacaine将哌啶环替换为氮杂螺环可降低局部麻醉药布比卡因的心脏毒性
err2026-05-08
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PREAI
errAlexander A. Kirichok; Yevhenii Vaiser; Irina Shton; Olexandr Tarasov; Maria Sokolenko; Dmytro Lesyk; Liana Dmytrovska; Kseniia Khrenova; Anatoly Soloviev; Sergey Tishkin; Petro Borysko; Yuliia Holota; Nadiia Diyuk; Valentyn Chigrinov; Tetyana Yegorova; Dmitry Granat; Pavel K. Mykhailiuk; Vladimir Kubyshkin; Iryna Pishel
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Direct α-C−H Heteroarylation of Unprotected Primary Amines未保护伯胺的直接α-C−H杂芳基化
err2026-05-06
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errOAAI
errGeorge D. Johnson; Stephanie A. Corio; James D. Grayson; Joshua D. Tibbetts; George Ballantyne; Qiao Cao; Hannah E. Askey; Joseph J. Bell-Tyrer; Oleksandr P. Datsenko; Mark A. Graham; Pavel K. Mykhailiuk; Jennifer S. Hirschi; Alexander J. Cresswell
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Mechanistically Guided Functionalization of α; α-Disubstituted Alkenyl Amides Enabled by a Conformationally Flexible Directing Auxiliary基于构象灵活的导向辅基指导的α,α-双取代烯基酰胺的功能化
err2026-02-20
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PREAI
errAl Vicente Riano D. Lisboa; Phornphan Yongpanich; Shijia Li; Ruchira Hariharan; Yilin Cao; Yang Gao; John A. Gurak Jr.; Pavel K. Mykhailiuk; Donna G. Blackmond; Peng Liu; Keary M. Engle
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A C1-Homologative Trifluoromethylation: Light-Driven Decarboxylative Trifluoroethylation of Carboxylic AcidsC1-Homologative的三氟甲基化: 光驱动的羧酸脱羧三氟乙基化
err2026-02-06
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PREAI
errFederico Belnome; Antonio Pulcinella; Stefano Bonciolini; Mattia Lepori; Oleksandr P. Datsenko; Zhen He; Matteo Gasparetto; Pavel K. Mykhailiuk; Bas de Bruin; Timothy Noël
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Asymmetric C-H Functionalization of Bicyclo[2.1.1]hexanes and Their 2-Oxa- and 2-Aza Derivatives via Rhodium Carbene Intermediates
err2026-01-01
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PREAI
errChen, Ziyi; Ly, Duc; Kanda, Yuzuru; Levterov, Vadym V.; Panasiuk, Yaroslav; Mykhailiuk, Pavel K.; Musaev, Djamaladdin G.; Davies, Huw M. L.
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Alkyl sulfonyl fluorides as ambiphiles in the stereoselective palladium(II)-catalysed cyclopropanation of unactivated alkenes烷基磺酰氟作为双亲试剂在非活化烯烃的立体选择性钯(II)催化环丙烷化反应中。
err2025-12-16
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errOAAI
errYilin Cao; Warabhorn Rodphon; Turki M. Alturaifi; Al Vicente Riano D. Lisboa; Zhouyang Ren; Job J. C. Struijs; Hui-Qi Ni; Taras Savchuk; Richard P. Loach; Shouliang Yang; Indrawan J. McAlpine; Donna G. Blackmond; Pavel K. Mykhailiuk; Peng Liu; K. Barry Sharpless; Keary M. Engle
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Ring-Expansion of Ketones with [1.1.1]Propellane
err2025-12-01
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PREAI
errKadam, Ganesh Arjun; Midya, Suparnak; Levchenko, Vitalina; Sham, Vadym; Mykhailiuk, Pavel K.; Hari, Durga Prasad
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Bicyclo[1.1.1]pentane Ketones via Friedel-Crafts Acylation
err2025-12-01
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PREAI
errUrbanska, Karolina; Ritterling, Freya; Twamley, Brendan; Cseh, Oliver; Levchenko, Vitalina; Ripenko, Vasyl; Mykhailiuk, Pavel K.; Senge, Mathias O.
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Glyoxylate Sulfonyl Hydrazone Enables a Scalable Approach to Reformatsky-Type Products from Aliphatic Alcohols via Photocatalytic HAT乙醛酸磺酰腙通过光催化氢原子转移实现了从脂肪醇制备 Reformatsky 型产物的一种可放大方法
err2025-12-01
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PREAI
errGasparetto, Matteo; Bonciolini, Stefano; Diprima, Damiano; Pulcinella, Antonio; Gabbey, Alexis L.; Datsenko, Oleksandr P.; Belnome, Federico; Schuurmans, Jasper H. A.; Mykhailiuk, Pavel K.; Noel, Timothy
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Triply convergent Ni-electrocatalytic assembly of 1,1-diaryl cyclobutanes, azetidines and oxetanes三重汇聚的Ni电催化组装1,1-二芳基环丁烷、氮杂环丁烷和氧杂环丁烷
err2025-11-11
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PREAI
errLuca Massaro; Philipp Neigenfind; Andrew Feng; Gannon Kuehn; Flynn C. Attard; Ava DeSanti; Michael R. Collins; Martin Bravo; Raymond K. Twumasi; Doris Chen; Philippe N. Bolduc; Michael Nicastri; Megan A. Emmanuel; Martins S. Oderinde; Maximilian D. Palkowitz; Xiaofan Zheng; Arianne C. Hunter; Kaid C. Harper; Chet C. Tyrol; Pavel K. Mykhailiuk; Yu Kawamata; Phil S. Baran
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Bicyclic Isosteres of Pyridine/Piperidine: From Synthesis to Applications吡啶/哌啶的双环类异构体:从合成到应用
err2025-09-22
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PREAI
errOleksandr Stashkevych; Volodymyr Kokhalskyi; Yevhenii Mynak; Vadym Levterov; Oleh Shablykin; Iryna Pishel; Pavel K. Mykhailiuk
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Angular Spirocyclic Azetidines: Synthesis, Characterization, and Evaluation in Drug Discovery
err2024-12-12
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errOAAI
errKirichok, Alexander A.; Tkachuk, Hennadii; Levchenko, Kostiantyn; Granat, Dmitry; Yegorova, Tetyana; Lesyk, Dmytro; Anisiforova, Anna; Holota, Yuliia; Zomchak, Viktoriia; Bodenchuk, Iryna; Kosach, Viktoriia; Borysko, Petro; Korzh, Rodion A.; Al-Maali, Galeb; Kubyshkin, Vladimir; Rzepa, Henry S.; Mykhailiuk, Pavel K.
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