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Jean‐Philippe Pin

university of bonn

93H指数
440论文数
3.5W被引数
收录论文 180
发表时间
EDNRB-dependent endothelin signaling reduces proliferation and promotes proneural-to-mesenchymal transition in gliomasEDNRB依赖的内皮素信号减少胶质瘤的增殖并促进前神经向间充质转变
err2026-04-23
err0
errOAAI
errDonovan Pineau; Leonor Garcia; Hugo Arnold; Antonija Hanžek; Maialen Arrieta; Laurent R Gauthier; Christine Granotier-Beckers; François D Boussin; Amaury Herbet; Marie Hautière; Valentin Asei-Ceschino; Clémentin Jacques; Laura Brard; Thomas Harnois; Valérie Coronas; Bruno Constantin; Aurélien Chatelier; Jean Chemin; Serge Urbach; Martial Seveno; Szimonetta Hideg; Chantal Ripoll; Kasandra Aguilar-Cázarez; Min Zheng; Guo-Hao Huang; Sheng-Qing Lv; Lei Zhang; Philippe Rondard; Laurent Prezeau; Jean-Philippe Pin; Hugues Duffau; Luc Bauchet; Valérie Rigau; Franck Denat; Charles Truillet; Didier Boquet; Jean-Philippe Hugnot
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Divergent Roles of mGlu2 and mGlu3 Receptors in Amyloid-β Production and Cognitive Dysfunctions in Alzheimer's DiseasemGlu2和mGlu3受体在阿尔茨海默病中淀粉样蛋白-β产生和认知功能障碍中的不同作用
err2026-04-14
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errOAAI
errPierre-André Lafon; Mireille Elodie Tsitokana; Ugo Guy Alenda; Yen-Ling Lian; Clémentine Eva Philibert; Mathieu Oosterlaken; Marta Cimadevila; Gaëlle Dudon; Jessica Monnic; Salomé Roux; Julie Bessié; Séverine Diem; Franck Vandermoere; Laurent Prézeau; Patrick Chames; Julie Kniazeff; Sylvie Claeysen; Anaïs Menny; Jean-Philippe Pin; Véronique Perrier; Jianfeng Liu; Philippe Rondard
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Multi-faceted roles of β-arrestins in G protein-coupled receptor endocytosisΒ-抑制蛋白在g蛋白偶联受体内吞中的多方面作用
err2025-12-11
err0
errOAAI
errJunke Liu; Li Xue; Magalie A. Ravier; Floriane Eshak; Francine C. Acher; Anne Goupil-Lamy; Marta Cimadevila; Julia Drube; Carsten Hoffmann; Asuka Inoue; Eric Trinquet; Elodie Dupuis; Laurent Prézeau; Jean-Philippe Pin; Philippe Rondard
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The Concise Guide to PHARMACOLOGY 2025/26: G protein-coupled receptors《简明药理学指南2025/26:G蛋白偶联受体》
err2025-12-01
err29
errOAAI
errAlexander, Stephen P. H.; Davenport, Anthony P.; Kelly, Eamonn; Gibb, Alasdair J.; Mathie, Alistair A.; Peach, Chloe J.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Southan, Christopher; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George R.; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bennett, Kirstie A.; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria A.; Bonaventure, Pascal; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Brown, Andrew J.; Burnstock, Geoffrey; Busnelli, Marta; Calo, Girolamo; Caruso, Vanni; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Christopoulos, Arthur; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dautzenberg, Frank M.; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Dubocovich, Margarita L.; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Forsman, Huamei Fu; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gbahou, Florence; Gerard, Craig; Gershengorn, Marvin; Glass, Michelle; Gloriam, David E.; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gruber, Christian; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hartman, Deborah S.; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Heitman, Laura; Herr, Deron R.; Hollenberg, Morley D.; Holliday, Nicholas D.; Holst, Birgitte; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; IJzerman, Adriaan P.; Inagami, Tadashi; Insel, Paul A.; Jacobson, Kenneth A.; Jacobson, Laura H.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kinsolving, Julia; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Laishram, Luxmichan; Langenhan, Tobias; Langmead, Christopher J.; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Leurs, Rob; Li, Xaria X.; Liebscher, Ines; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet J.; Malfacini, Davide; Manning, Maurice; Marangon, Davide; Martemyanov, Kirill; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Neubig, Richard R.; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Perry-Hauser, Nicole; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Qin, Helena Chengxue; Quinn, Mark; Raffaele, Stefano; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Buzon, Alejandro Romeral; Rondard, Philippe; Rosenkilde, Mette M.; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Scholz, Nicole; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Shukla, Arun K.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Smith, Nicola J.; Staeubert, Claudia; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David M.; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Verbalis, Joseph G.; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Wu, Huixian; Yang, Cheng; Yao, Chengcan; Ye, Richard D.; Zaidman, Nathan
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Nanobodies: a new paradigm for brain disorder therapies纳米抗体:治疗脑部疾病的一种新范式
err2025-11-05
err0
PREAI
errPierre-André Lafon; Laurent Prézeau; Jean-Philippe Pin; Philippe Rondard
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Structural characterization of five functional states of metabotropic glutamate receptor 8代谢型谷氨酸受体8五种功能状态的结构表征
err2025-09-18
err0
PREAI
errJie Zhao; Yue Deng; Zheng Xu; Chanjuan Xu; Chang Zhao; Ziyan Li; Hui Sun; Xiaowen Tian; Yuxuan Song; Marta Cimadevila; Heli Wang; Yuxuan Liu; Xiaoyu Zhang; Yiyang Chen; Suyue Sun; Xihao Yong; Lantian Su; Yixiao He; Yi Zhong; Hao Yang; Jean-Philippe Pin; Wei Yan; Zhenhua Shao; Jianfeng Liu
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Non-canonical internalization mechanisms of mGlu receptorsmGlu受体的非经典内化机制
err2025-07-30
err0
errOAAI
errMarta Cimadevila; Junke Liu; Damien Maurel; Isabelle Brabet; Marine Hoscar; Julia Drube; Carsten Hoffmann; Asuka Inoue; Philippe Rondard; Pierre-André Lafon; Laurent Prézeau; Jean-Philippe Pin
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Nanobody therapy rescues behavioural deficits of NMDA receptor hypofunction纳米抗体疗法可挽救NMDA受体功能减退的行为缺陷
errNature
IF48.5
err2025-07-23
err0
errOAAI
errMathieu Oosterlaken; Angelina Rogliardo; Tatiana Lipina; Pierre-André Lafon; Mireille Elodie Tsitokana; Mathilde Keck; Héloïse Cahuzac; Pierre Prieu-Sérandon; Séverine Diem; Cécile Derieux; Célia Camberlin; Chrystel Lafont; Damien Meyer; Patrick Chames; Franck Vandermoere; Philippe Marin; Laurent Prézeau; Denis Servent; Ali Salahpour; Amy J. Ramsey; Carine Bécamel; Jean-Philippe Pin; Julie Kniazeff; Philippe Rondard
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Triple Labeling Resolves a GPCR Intermediate State by Using Three-Color Single Molecule FRET三重标记利用三色单分子FRET解析GPCR的中间状态
err2025-05-15
err0
errOAAI
errBonhomme, Leo; Bilgen, Ecenaz; Clerte, Caroline; Pin, Jean-Philippe; Rondard, Philippe; Margeat, Emmanuel; Lamb, Don C.; Quast, Robert B.
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A modular click ligand-directed approach to label endogenous dopamine D1 receptors in live cells一种模块化的点击配体定向方法用于标记活细胞内源性多巴胺D1受体
err2025-04-11
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errOAAI
errGomez-Santacana, Xavier; Boutonnet, Marin; Martinez-Juves, Carles; Cimadevila, Marta; Catena, Juanlo; Moutin, Enora; Roux, Thomas; Trinquet, Eric; Lamarque, Laurent; Perroy, Julie; Prezeau, Laurent; Zwier, Jurriaan M.; Pin, Jean-Philippe; Llebaria, Amadeu
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Structural basis of orientated asymmetry in a mGlu heterodimer
err2024-11-28
err0
errOAAI
errHuang, Weizhu; Jin, Nan; Guo, Jia; Shen, Cangsong; Xu, Chanjuan; Xi, Kun; Bonhomme, Leo; Quast, Robert B.; Shen, Dan-Dan; Qin, Jiao; Liu, Yi-Ru; Song, Yuxuan; Gao, Yang; Margeat, Emmanuel; Rondard, Philippe; Pin, Jean-Philippe; Zhang, Yan; Liu, Jianfeng
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Novel Inhibitory Site Revealed by XAP044 Mode of Action on the Metabotropic Glutamate 7 Receptor Venus Flytrap Domain
err2024-05-01
err2
PREAI
errCristiano, Nunzia; Cabaye, Alexandre; Brabet, Isabelle; Glatthar, Ralf; Tora, Amelie; Goudet, Cyril; Bertrand, Hugues-Olivier; Goupil-Lamy, Anne; Flor, Peter J.; Pin, Jean-Philippe; McCort-Tranchepain, Isabelle; Acher, Francine C.
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Absence of calcium-sensing receptor basal activity due to inter-subunit disulfide bridges
err2024-04-25
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errOAAI
errMa, Shumin; Yin, Xueliang; Pin, Jean-Philippe; Rondard, Philippe; Yi, Ping; Liu, Jianfeng
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Specific pharmacological and Gi/o protein responses of some native GPCRs in neurons
err2024-03-05
err4
errOAAI
errXu, Chanjuan; Zhou, Yiwei; Liu, Yuxuan; Lin, Li; Liu, Peng; Wang, Xiaomei; Xu, Zhengyuan; Pin, Jean-Philippe; Rondard, Philippe; Liu, Jianfeng
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Epitope Identification of an mGlu5 Receptor Nanobody Using Physics-Based Molecular Modeling and Deep Learning Techniques
err2024-02-29
err4
PREAI
errEshak, Floriane; Pion, Leo; Scholler, Pauline; Nevoltris, Damien; Chames, Patrick; Rondard, Philippe; Pin, Jean-Philippe; Acher, Francine C.; Goupil-Lamy, Anne
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Synthesis and pharmacological characterization of conformationally restricted 2-amino-Adipic acid analogs and carboxycyclopropyl glycines as selective metabotropic glutamate 2 receptor agonists
err2024-02-01
err1
errOAAI
errStaudt, Markus; Liu, Na; Malhaire, Fanny; Doroudian, Yasaman; Prezeau, Laurent; Renard, Emma; Hasanpour, Zahra; Pin, Jean-Philippe; Bunch, Lennart
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TrkB receptor interacts with mGlu2 receptor and mediates antipsychotic- like effects of mGlu2 receptor activation in the mouse
err2024-01-26
err3
errOAAI
errPhilibert, Clementine Eva; Disdier, Candice; Lafon, Pierre-Andre; Bouyssou, Alexandre; Oosterlaken, Mathieu; Galant, Sonya; Pizzoccaro, Anne; Tuduri, Pola; Ster, Jeanne; Liu, Jianfeng; Kniazeff, Julie; Pin, Jean-Philippe; Rondard, Philippe; Marin, Philippe; Vandermoere, Franck
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Design, Synthesis, Pharmacology, and In Silico Studies of (1S,2S,3S)-2-((S)-Amino(carboxy)methyl)-3-(carboxymethyl)cyclopropane-1-carboxylic Acid (LBG30300): A Picomolar Potency Subtype-Selective mGlu2 Receptor Agonist
err2024-01-03
err2
PREAI
errLiu, Na; Eshak, Floriane; Malhaire, Fanny; Brabet, Isabelle; Prezeau, Laurent; Renard, Emma; Pin, Jean-Philippe; Acher, Francine C.; Staudt, Markus; Bunch, Lennart
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The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors药理学2023/24简明指南: g蛋白偶联受体
err2023-12-20
err149
errOAAI
errAlexander, Stephen P. H.; Christopoulos, Arthur; Davenport, Anthony P.; Kelly, Eamonn; Mathie, Alistair A.; Peters, John A.; Veale, Emma L.; Armstrong, Jane F.; Faccenda, Elena; Harding, Simon D.; Davies, Jamie A.; Abbracchio, Maria Pia; Abraham, George; Agoulnik, Alexander; Alexander, Wayne; Al-hosaini, Khaled; Back, Magnus; Baker, Jillian G.; Barnes, Nicholas M.; Bathgate, Ross; Beaulieu, Jean-Martin; Beck-Sickinger, Annette G.; Behrens, Maik; Bernstein, Kenneth E.; Bettler, Bernhard; Birdsall, Nigel J. M.; Blaho, Victoria; Boulay, Francois; Bousquet, Corinne; Brauner-Osborne, Hans; Burnstock, Geoffrey; Calo, Girolamo; Castano, Justo P.; Catt, Kevin J.; Ceruti, Stefania; Chazot, Paul; Chiang, Nan; Chini, Bice; Chun, Jerold; Cianciulli, Antonia; Civelli, Olivier; Clapp, Lucie H.; Couture, Rejean; Cox, Helen M.; Csaba, Zsolt; Dahlgren, Claes; Dent, Gordon; Douglas, Steven D.; Dournaud, Pascal; Eguchi, Satoru; Escher, Emanuel; Filardo, Edward J.; Fong, Tung; Fumagalli, Marta; Gainetdinov, Raul R.; Garelja, Michael L.; de Gasparo, Marc; Gerard, Craig; Gershengorn, Marvin; Gobeil, Fernand; Goodfriend, Theodore L.; Goudet, Cyril; Gratz, Lukas; Gregory, Karen J.; Gundlach, Andrew L.; Hamann, Jorg; Hanson, Julien; Hauger, Richard L.; Hay, Debbie L.; Heinemann, Akos; Herr, Deron; Hollenberg, Morley D.; Holliday, Nicholas D.; Horiuchi, Mastgugu; Hoyer, Daniel; Hunyady, Laszlo; Husain, Ahsan; Ijzerman, Adriaan P.; Inagami, Tadashi; Jacobson, Kenneth A.; Jensen, Robert T.; Jockers, Ralf; Jonnalagadda, Deepa; Karnik, Sadashiva; Kaupmann, Klemens; Kemp, Jacqueline; Kennedy, Charles; Kihara, Yasuyuki; Kitazawa, Takio; Kozielewicz, Pawel; Kreienkamp, Hans-Juergen; Kukkonen, Jyrki P.; Langenhan, Tobias; Larhammar, Dan; Leach, Katie; Lecca, Davide; Lee, John D.; Leeman, Susan E.; Leprince, Jerome; Li, Xaria X.; Lolait, Stephen J.; Lupp, Amelie; Macrae, Robyn; Maguire, Janet; Malfacini, Davide; Mazella, Jean; McArdle, Craig A.; Melmed, Shlomo; Michel, Martin C.; Miller, Laurence J.; Mitolo, Vincenzo; Mouillac, Bernard; Mueller, Christa E.; Murphy, Philip M.; Nahon, Jean-Louis; Ngo, Tony; Norel, Xavier; Nyimanu, Duuamene; O'Carroll, Anne-Marie; Offermanns, Stefan; Panaro, Maria Antonietta; Parmentier, Marc; Pertwee, Roger G.; Pin, Jean-Philippe; Prossnitz, Eric R.; Quinn, Mark; Ramachandran, Rithwik; Ray, Manisha; Reinscheid, Rainer K.; Rondard, Philippe; Rovati, G. Enrico; Ruzza, Chiara; Sanger, Gareth J.; Schoeneberg, Torsten; Schulte, Gunnar; Schulz, Stefan; Segaloff, Deborah L.; Serhan, Charles N.; Singh, Khuraijam Dhanachandra; Smith, Craig M.; Stoddart, Leigh A.; Sugimoto, Yukihiko; Summers, Roger; Tan, Valerie P.; Thal, David; Thomas, Walter (Wally); Timmermans, Pieter B. M. W. M.; Tirupula, Kalyan; Toll, Lawrence; Tulipano, Giovanni; Unal, Hamiyet; Unger, Thomas; Valant, Celine; Vanderheyden, Patrick; Vaudry, David; Vaudry, Hubert; Vilardaga, Jean-Pierre; Walker, Christopher S.; Wang, Ji Ming; Ward, Donald T.; Wester, Hans-Juergen; Willars, Gary B.; Williams, Tom Lloyd; Woodruff, Trent M.; Yao, Chengcan; Ye, Richard D.
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Different EGF-induced receptor dimer conformations for signaling and internalization
err2023-12-10
err0
errOAAI
errHaubrich, Jordi; Zwier, Jurriaan M.; Charrier-Savournin, Fabienne; Prezeau, Laurent; Pin, Jean-Philippe
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