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Discovery and Early Optimization of 1H-Indole-2-carboxamides with Anti-Trypanosoma cruzi Activity 1H-吲哚-2-甲酰胺类化合物的发现及其抗克氏锥虫活性初探 de Oliveira, Ramon G.; Cruz, Luiza R.; Dessoy, Marco A.; Koovits, Paul J.; dos Santos, Deborah A.; de Oliveira, Luiz F. N.; Ferreira, Rafael A.; Mollo, Maria C.; Lee, Eun; Duarte, Simone M.; Krogh, Renata; Ferreira, Leonardo L. G.; Chelucci, Rafael C.; Dichiara, Maria; Simpson, Quillon J.; Feltrin, Clarissa; da Silva, Adriana C.; dos Santos, Benedito M.; Broering, Milena F.; Pollastri, Michael P.; Ferrins, Lori; Moraes, Carolina B.; Andricopulo, Adriano D.; Kratz, Jadel M.; Sjo, Peter; Mowbray, Charles E.; Dias, Luiz C. 分享 收藏
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Identification of Substituted 4-Aminocinnolines as Broad-Spectrum Antiparasitic Agents Spaulding, Andrew; Sharma, Amrita; Giardini, Miriam A.; Hoffman, Benjamin; Bernatchez, Jean A.; Mccall, Laura-Isobel; Calvet, Claudia M.; Ackermann, Jasmin; Souza, Julia M.; Thomas, Diane; Millard, Caroline C.; Devine, William G.; Singh, Baljinder; Silva, Everton M.; Leed, Susan E.; Roncal, Norma E.; Penn, Erica C.; Erath, Jessey; Kumar, Gaurav; Sepulveda, Yadira; Garcia, Arnold; Rodriguez, Ana; El-Sakkary, Nelly; Sciotti, Richard J.; Campbell, Robert F.; Momper, Jeremiah D.; Mckerrow, James H.; Caffrey, Conor R.; Siqueira-Neto, Jair L.; Pollastri, Michael P.; Mensa-Wilmot, Kojo; Ferrins, Lori 分享 收藏
Heterocyclic core modifications in trypanosomacidal 2-[(phenylheteroaryl)ethyl]ureas Toynton, Arthur; Ferrins, Lori; Newson, Harriet L.; Sykes, Melissa L.; Varghese, Swapna; Nguyen, Nghi; Russell, Stephanie; Rahmani, Raphael; Cheang, Jeremy; Flematti, Gavin R.; Skelton, Brian W.; Zulfiqar, Bilal; Avery, Vicky M.; Baell, Jonathan B.; Piggott, Matthew J. 分享 收藏
Pharmacophore Identification and Structure-Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei Ferrins, Lori; Diaz, Rosario; Cordon-Obras, Carlos; Rojas-Barros, Domingo; Quotadamo, Antonio; Oehme, Daniel P.; Ceballos-Perez, Gloria; Swaminathan, Uma; Perez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Garcia-Hernandez, Raquel; Gomez-Linan, Claudia; Saura, Andreu; Ruiz-Perez, Luis Miguel; Gamarro, Francisco; Martinez-Martinez, Maria Santos; Manzano, Pilar; Gonzalez-Pacanowska, Dolores; Navarro, Miguel; Pollastri, Michael P. 分享 收藏
Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus 开源抗生素: 简单的二芳基咪唑对耐甲氧西林金黄色葡萄球菌有效 Klug, Dana M.; Tse, Edwin G.; Silva, Daniel G.; Cao, Yafeng; Charman, Susan A.; Chauhan, Jyoti; Crighton, Elly; Dichiara, Maria; Drake, Chris; Drewry, David; da Silva Emery, Flavio; Ferrins, Lori; Graves, Lee; Hopkins, Emily; Kresina, Thomas A. C.; Lorente-Macias, Alvaro; Perry, Benjamin; Phipps, Richard; Quiroga, Bruno; Quotadamo, Antonio; Sabatino, Giada N.; Sama, Anthony; Schatzlein, Andreas; Simpson, Quillon J.; Steele, Jonathan; Shanu-Wilson, Julia; Sjo, Peter; Stapleton, Paul; Swain, Christopher J.; Vaideanu, Alexandra; Xie, Huanxu; Zuercher, William; Todd, Matthew H. 分享 收藏
Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes (vol 14, 1149145, 2023) Ferrins, Lori; Buskes, Melissa J.; Kapteyn, Madison M.; Engels, Hannah N.; Enos, Suzanne E.; Lu, Chenyang; Klug, Dana M.; Singh, Baljinder; Quotadamo, Antonio; Bachovchin, Kelly; Tear, Westley F.; Spaulding, Andrew E.; Forbes, Katherine C.; Bag, Seema; Rivers, Mitch; Leblanc, Catherine; Burchfield, Erin; Armand, Jeremy R.; Diaz-Gonzalez, Rosario; Ceballos-Perez, Gloria; Garcia-Hernandez, Raquel; Perez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Gomez-Linan, Claudia; Ruiz-Perez, Luis Miguel; Gamarro, Francisco; Gonzalez-Pacanowska, Dolores; Navarro, Miguel; Mensa-Wilmot, Kojo; Pollastri, Michael P.; Kyle, Dennis E.; Rice, Christopher A. 分享 收藏
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Structure-Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis Dichiara, Maria; Simpson, Quillon J.; Quotadamo, Antonio; Jalani, Hitesh B.; Huang, Anson X.; Millard, Caroline C.; Klug, Dana M.; Tse, Edwin G.; Todd, Matthew H.; Silva, Daniel Gedder; Emery, Flavio da Silva; Carlson, J. Eric; Zheng, Shao-Liang; Vleminckx, Margot; Matheeussen, An; Caljon, Guy; Pollastri, Michael P.; Sjo, Peter; Perry, Benjamin; Ferrins, Lori 分享 收藏
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