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Potent and Selective Human Constitutive Androstane Receptor Activator DL5055 Facilitates Cyclophosphamide-Based Chemotherapies 强效且选择性的 Constitutive Androstane Receptor 人体激活剂 DL5055 促进基于环磷酰胺的化疗 Liang, Dongdong; Li, Linhao; Ai, Yong; Li, Zhihui; Hedrich, William D.; Sakamuru, Srilatha; Lynch, Caitlin; Yu, Wenbo; Watts-Ouattara, Ismael; Heyward, Scott; Xia, Menghang; Mackerell Jr, Alexander D.; Wang, Hongbing; Xue, Fengtian 分享 收藏
SARS-CoV-2 ORF3a Protein as a Therapeutic Target against COVID-19 and Long-Term Post-Infection Effects Zhang, Jiantao; Hom, Kellie; Zhang, Chenyu; Nasr, Mohamed; Gerzanich, Volodymyr; Zhang, Yanjin; Tang, Qiyi; Xue, Fengtian; Simard, J. Marc; Zhao, Richard Y. 分享 收藏
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A small-molecule inhibitor and degrader of the RNF5 ubiquitin ligase Ruan, Jingjing; Liang, Dongdong; Yan, Wenjing; Zhong, Yongwang; Talley, Daniel C.; Rai, Ganesha; Tao, Dingyin; LeClair, Christopher A.; Simeonov, Anton; Zhang, Yinghua; Chen, Feihu; Quinney, Nancy L.; Boyles, Susan E.; Cholon, Deborah M.; Gentzsch, Martina; Henderson, Mark J.; Xue, Fengtian; Fang, Shengyun 分享 收藏
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Targeting CAR and Nrf2 improves cyclophosphamide bioactivation while reducing doxorubicin-induced cardiotoxicity in triple-negative breast cancer treatment Stern, Sydney; Liang, Dongdong; Li, Linhao; Kurian, Ritika; Lynch, Caitlin; Sakamuru, Srilatha; Heyward, Scott; Zhang, Junran; Kareem, Kafayat Ajoke; Chun, Young Wook; Huang, Ruili; Xia, Menghang; Hong, Charles C.; Xue, Fengtian; Wang, Hongbing 分享 收藏
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Profiling the Tox21 Chemical Collection for Acetylcholinesterase Inhibition Li, Shuaizhang; Zhao, Jinghua; Huang, Ruili; Travers, Jameson; Klumpp-Thomas, Carleen; Yu, Wenbo; MacKerell, Alexander D., Jr.; Sakamuru, Srilatha; Ooka, Masato; Xue, Fengtian; Sipes, Nisha S.; Hsieh, Jui-Hua; Ryan, Kristen; Simeonov, Anton; Santillo, Michael F.; Xia, Menghang 分享 收藏
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Pyrazole-4-Carboxamide (YW2065): A Therapeutic Candidate for Colorectal Cancer via Dual Activities of Wnt/β-Catenin Signaling Inhibition and AMP-Activated Protein Kinase (AMPK) Activation Yang, Wei; Li, Yingjun; Ai, Yong; Obianom, Obinna N.; Guo, Dong; Yang, Hong; Sakamuru, Srilatha; Xia, Menghang; Shu, Yan; Xue, Fengtian 分享 收藏
Human constitutive androstane receptor agonist DL5016: A novel sensitizer for cyclophosphamide-based chemotherapies Liang, Dongdong; Li, Linhao; Lynch, Caitlin; Mackowiak, Bryan; Hedrich, William D.; Ai, Yong; Yin, Yue; Heyward, Scott; Xia, Menghang; Wang, Hongbing; Xue, Fengtian 分享 收藏
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BCL6 Inhibitor-Mediated Downregulation of Phosphorylated SAMHD1 and T Cell Activation Are Associated with Decreased HIV Infection and Reactivation Cai, Yanhui; Abdel-Mohsen, Mohamed; Tomescu, Costin; Xue, Fengtian; Wu, Guoxin; Howell, Bonnie J.; Ai, Yong; Sun, Jie; Azzoni, Livio; Le Coz, Carole; Romberg, Neil; Montaner, Luis J. 分享 收藏