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B

B. A. Kashemirov

David Geffen School of Medicine at UCLA

H指数:28

被引数:2,691

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教育背景

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工作经历

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荣誉奖项

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Humanized Candida and NanoBiT Assays Expedite Discovery of Bdf1 Bromodomain Inhibitors With Antifungal Potential

人源化念珠菌和NanoBiT分析加速具有抗真菌潜力的Bdf1溴域抑制剂的开发

ADVANCED SCIENCE

IF14.1

2025-01-160

OAAI

Uridine Bisphosphonates Differentiate Phosphoglycosyl Transferase Superfamilies

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

IF15.6

2024-01-250

OA

Synthesis and anti-cancer potential of potent peripheral MAOA inhibitors designed to limit blood:brain penetration

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2023-09-016

OAAI

Microwave-Accelerated McKenna Synthesis of Phosphonic Acids: An Investigation

IF4.6

2023-04-152

OAAI

Toward more potent imidazopyridine inhibitors of Candida albicans Bdf1: Modeling the role of structural waters in selective ligand binding

JOURNAL OF COMPUTATIONAL CHEMISTRY

IF4.8

2022-10-032

OAAI

Fluorescent risedronate analogue 800CW-pRIS improves tooth extraction-associated abnormal wound healing in zoledronate-treated mice

COMMUNICATIONS MEDICINE

IF6.3

2022-09-052

OAAI

A Novel Small Molecule Neurotrophin-3 Analogue Promotes Inner Ear Neurite Outgrowth and Synaptogenesis In vitro

FRONTIERS IN CELLULAR NEUROSCIENCE

IF4

2021-07-1512

OAAI

Design and Synthesis of Cathepsin-K-Activated Osteoadsorptive Fluorogenic Sentinel (OFS) Probes for Detecting Early Osteoclastic Bone Resorption in a Multiple Myeloma Mouse Model

BIOCONJUGATE CHEMISTRY

IF3.9

2021-05-0614

OAAI

Paradoxical androgen receptor regulation by small molecule enantiomers

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

IF9.1

2021-03-190

OAAI

Completing the β,γ-CXY-dNTP Stereochemical Probe Toolkit: Synthetic Access to the dCTP Diastereomers and 31P and 19F NMR Correlations with Absolute Configurations

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2020-10-308

PREAI

Paradoxical androgen receptor regulation by small molecule enantiomers

CANCER RESEARCH

IF16.6

2020-08-150

PRE

A pre-catalytic non-covalent step governs DNA polymerase β fidelity

NUCLEIC ACIDS RESEARCH

IF13.1

2019-11-1611

OAAI

Bisphosphonate-Linked TrkB Agonist: Cochlea-Targeted Delivery of a Neurotrophic Agent as a Strategy for the Treatment of Hearing Loss

BIOCONJUGATE CHEMISTRY

IF3.9

2018-02-2722

OAAI

Selective BET bromodomain inhibition as an antifungal therapeutic strategy

NATURE COMMUNICATIONS

IF15.7

2017-05-1838

OAAI

Fluorescent Bisphosphonate and Carboxyphosphonate Probes: A Versatile Imaging Toolkit for Applications in Bone Biology and Biomedicine

BIOCONJUGATE CHEMISTRY

IF3.9

2015-12-0848

OA

5′-β,γ-CHF-ATP Diastereomers: Synthesis and Fluorine-Mediated Selective Binding by c-Src Protein Kinase

ORGANIC LETTERS

IF5

2015-03-1715

OAAI

Real-Time Intravital Imaging Establishes Tumor-Associated Macrophages as the Extraskeletal Target of Bisphosphonate Action in Cancer

CANCER DISCOVERY

IF33.3

2015-01-11121

OAAI

Small Molecule Inhibition of SAMHD1 dNTPase by Tetramer Destabilization

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

IF15.6

2014-07-0838

OAAI

On the Observation of Discrete Fluorine NMR Spectra for Uridine 5′-β,γ-Fluoromethylenetriphosphate Diastereonners at Basic pH

JOURNAL OF ORGANIC CHEMISTRY

IF3.6

2014-05-128

OAAI

β,γ-CHF- and β,γ-CHCl-dGTP Diastereomers: Synthesis, Discrete 31P NMR Signatures, and Absolute Configurations of New Stereochemical Probes for DNA Polymerases

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

IF15.6

2012-05-1837

OAAI