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收藏Discovery of MAP855, an Efficacious and Selective MEK1/2 Inhibitor with an ATP-Competitive Mode of Action
Poddutoori, Ramulu; Aardalen, Kimberly; Aithal, Kiran; Barahagar, Sanjeev Surendranath; Belliappa, Charamanna; Bock, Mark; Chelur, Shekar; Gerken, Andrea; Gopinath, Sreevalsam; Gruenenfelder, Bjoern; Kiffe, Michael; Krishnaswami, Maithreyi; Langowski, John; Madapa, Sudharshan; Narayanan, Kishore; Pandit, Chetan; Panigrahi, Sunil Kumar; Perrone, Mark; Potakamuri, Ravi Kumar; Ramachandra, Murali; Ramanathan, Anuradha; Ramos, Rita; Sager, Emine; Samajdar, Susanta; Subramanya, Hosahalli S.; Thimmasandra, Devaraja Seethappa; Venetsanakos, Eleni; Mobitz, Henrik
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收藏Bardet-Biedl syndrome proteins regulate intracellular signaling and neuronal function in patient-specific iPSC-derived neurons
Wang, Liheng; Liu, Yang; Stratigopoulos, George; Panigrahi, Sunil; Sui, Lina; Zhang, Yiying; Leduc, Charles A.; Glover, Hannah J.; De Rosa, Maria Caterina; Burnett, Lisa C.; Williams, Damian J.; Shang, Linshan; Goland, Robin; Tsang, Stephen H.; Wardlaw, Sharon; Egli, Dieter; Zheng, Deyou; Doege, Claudia A.; Leibel, Rudolph L.
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收藏Selective Vulnerability to Pyrimidine Starvation in Hematologic Malignancies Revealed by AG-636, a Novel Clinical-Stage Inhibitor of Dihydroorotate Dehydrogenase
McDonald, Gabrielle; Chubukov, Victor; Coco, John; Truskowski, Kevin; Narayanaswamy, Rohini; Choe, Sung; Steadman, Mya; Artin, Erin; Padyana, Anil K.; Jin, Lei; Ronseaux, Sebastien; Locuson, Charles; Fan, Zi-Peng; Erdmann, Tabea; Mann, Alan; Hayes, Sebastian; Fletcher, Mark; Nellore, Kavitha; Rao, Siva Sanjeeva; Subramanya, Hosahalli; Reddy, K. Satish; Panigrahi, Sunil K.; Antony, Thomas; Gopinath, Sreevalsam; Sui, Zhihua; Nagaraja, Nelamangala; Dang, Lenny; Lenz, Georg; Hurov, Jonathan; Biller, Scott A.; Murtie, Josh; Marks, Kevin M.; Ulanet, Danielle B.
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收藏Increased Cerebrospinal Fluid Amyloid-β During Sleep Deprivation in Healthy Middle-Aged Adults Is Not Due to Stress or Circadian Disruption健康中年人睡眠剥夺期间脑脊液淀粉样蛋白-β 的增加不是由于压力或昼夜节律中断
Blattner, Margaret S.; Panigrahi, Sunil K.; Toedebusch, Cristina D.; Hicks, Terry J.; McLeland, Jennifer S.; Banks, Ian R.; Schaibley, Claire; Ovod, Vitaliy; Mawuenyega, Kwasi G.; Bateman, Randall J.; Wardlaw, Sharon L.; Lucey, Brendan P.
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收藏Preclinical evaluation of pharmacokinetics, pharmacodynamics and efficacy of the dual CD73-A2AR Inhibitors
Chikkanna, Dinesh; Narayanan, Kishore; Panigrahi, Sunil; Priyadarshini, Garima; Goyal, Megha; Mani, Jiju; Samiulla, D. S.; Dadhania, Sagar; Aravind, A. B.; Daginakatte, Girish; Anthony, Thomas; Nellore, Kavitha; Samajdar, Susanta; Ramachandra, Murali
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收藏Selective PPARδ Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD) (vol 9, pg 935, 2018)
Lagu, Bharat; Kluge, Arthur F.; Tozzo, Effie; Fredenburg, Ross; Bell, Eric L.; Goddeeris, Matthew M.; Dwyer, Peter; Basinski, Andrew; Senaiar, Ramesh S.; Jaleel, Mahaboobi; Tiwari, Nirbhay Kumar; Panigrahi, Sunil K.; Krishnamurthy, Narasimha Rao; Takahashi, Taisuke; Patane, Michael A.
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收藏Selective PPARδ Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD)
Lagu, Bharat; Kluge, Arthur F.; Tozzo, Effie; Fredenburg, Ross; Bell, Eric L.; Goddeeris, Matthew M.; Dwyer, Peter; Basinski, Andrew; Senaiar, Ramesh S.; Jaleel, Mahaboobi; Tiwari, Nirbhay Kumar; Panigrahi, Sunil K.; Krishnamurthy, Narasimha Rao; Takahashi, Taisuke; Patane, Michael A.
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收藏Preclinical In vivo evaluation of efficacy, pharmacokinetics and pharmacodynamics of novel PRMT5 inhibitors in multiple tumor models
Chikkanna, Dinesh; Panigrahi, Sunil Kumar; Rajagopalan, Sujatha; Sammeta, Srinivasa Raju; Chawla, Darshan; Pavithra, S.; Samiulla, D. S.; Prasanna, Angelene; Chand, Priyabrata; Aithal, Kiran; Marri, Sai Sudheer; Kumar, Naveen; Ganipisetty, Srinivasa Rao; Mutyala, Raju; Rao, Kasieswara; Antony, Thomas; Daginakatte, Girish; Lakshminarasimhan, Anirudha; Mohan, R.; Narasihmarao, K.; Chelur, Shekar; Pandit, Chetan; Samajdar, Susanta; Ramachandra, Murali
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收藏Novel inhibitors of protein arginine methyltransferase 5 (PRMT5) for the treatment of solid tumors
Chikkanna, Dinesh; Panigrahi, Sunil Kumar; Rajagopalan, Sujatha; Sammeta, Srinivasa Raju; Lakshminarasimhan, Anirudha; Mohan, R.; Narasihmarao, K.; Chawla, Darshan; Bhat, Harsha; Kasturi, Venkateswarlu; Samiulla, D. S.; Prasanna, Angelene; Aithal, Kiran; Chand, Priyabrata Chand; Kumar, Naveen; Marri, Sai Sudheer; Ganipisetty, Srinivasa Rao; Rao, Kasieswara N.; Mutyala, Raju; Neerukattu, Nageswara Rao; Nithesh, K.; Amin, Ramya; Gorade, Priyanka Machhindra; Antony, Thomas; Daginakatte, Girish; Chelur, Shekar; Pandit, Chetan; Samajdar, Susanta; Ramachandra, Murali
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