未登录Growing a single suspended perfect protein crystal in a fully noncontact manner
Wu, Zi-Qing; Liu, Yong-Ming; Cheng, Qing-Di; Li, Chen-Yuan; Liu, Ya-Li; Ge, Wan-Yi; Falke, Sven; Brognaro, Hevila; Chen, Jing-Jie; Zhou, Huan; Shang, Peng; He, Jian-Hua; Betzel, Christian; Yin, Da-Chuan
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收藏Time-resolved crystallography of boric acid binding to the active site serine of the β-lactamase CTX-M-14 and subsequent 1,2-diol esterification
Prester, Andreas; Perbandt, Markus; Galchenkova, Marina; Oberthuer, Dominik; Werner, Nadine; Henkel, Alessandra; Maracke, Julia; Yefanov, Oleksandr; Hakanpaeae, Johanna; Pompidor, Guillaume; Meyer, Jan; Chapman, Henry; Aepfelbacher, Martin; Hinrichs, Winfried; Rohde, Holger; Betzel, Christian
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收藏SARS-CoV-2 Mpro responds to oxidation by forming disulfide and NOS/SONOS bonds
Reinke, Patrick Y. A.; Schubert, Robin; Oberthuer, Dominik; Galchenkova, Marina; Mashhour, Aida Rahmani; Guenther, Sebastian; Chretien, Anais; Round, Adam; Seychell, Brandon Charles; Norton-Baker, Brenna; Kim, Chan; Schmidt, Christina; Koua, Faisal H. M.; Tolstikova, Alexandra; Ewert, Wiebke; Murillo, Gisel Esperanza Pena; Mills, Grant; Kirkwood, Henry; Brognaro, Hevila; Han, Huijong; Koliyadu, Jayanath; Schulz, Joachim; Bielecki, Johan; Lieske, Julia; Maracke, Julia; Knoska, Juraj; Lorenzen, Kristina; Brings, Lea; Sikorski, Marcin; Kloos, Marco; Vakili, Mohammad; Vagovic, Patrik; Middendorf, Philipp; de Wijn, Raphael; Bean, Richard; Letrun, Romain; Han, Seonghyun; Falke, Sven; Geng, Tian; Sato, Tokushi; Srinivasan, Vasundara; Kim, Yoonhee; Yefanov, Oleksandr M.; Gelisio, Luca; Beck, Tobias; Dore, Andrew S.; Mancuso, Adrian P.; Betzel, Christian; Bajt, Sasa; Redecke, Lars; Chapman, Henry N.; Meents, Alke; Turk, Dusan; Hinrichs, Winfried; Lane, Thomas J.
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收藏Controlling the size, shape, and stability of SeNPs by bromelain: Improved antioxidant, anti-bacterial and anti-cancer activities
Bibi, Surriya; Munawar, Aisha; Ishaq, Muhammad Waqas; Zaman, Fakhar; Abid, Muhammad; Rafi, Ali; Saeed, Ahsan; Akrem, Ahmad; Schubert, Robin; Aftab, Usman; Ali, Syed Abid; Betzel, Christian; Khan, Irfan Ullah
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收藏Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections
Reinke, Patrick Y. A.; de Souza, Edmarcia Elisa; Guenther, Sebastian; Falke, Sven; Lieske, Julia; Ewert, Wiebke; Loboda, Jure; Herrmann, Alexander; Mashhour, Aida Rahmani; Karnicar, Katarina; Usenik, Aleksandra; Lindic, Natasa; Sekirnik, Andreja; Botosso, Viviane Fongaro; Santelli, Glaucia Maria Machado; Kapronezai, Josana; de Araujo, Marcelo Valdemir; Silva-Pereira, Taiana Taina; de Souza Filho, Antonio Francisco; Tavares, Mariana Silva; Florez-Alvarez, Lizdany; de Oliveira, Danielle Bruna Leal; Durigon, Edison Luiz; Giaretta, Paula Roberta; Heinemann, Marcos Bryan; Hauser, Maurice; Seychell, Brandon; Boehler, Hendrik; Rut, Wioletta; Drag, Marcin; Beck, Tobias; Cox, Russell; Chapman, Henry N.; Betzel, Christian; Brehm, Wolfgang; Hinrichs, Winfried; Ebert, Gregor; Latham, Sharissa L.; de Sa Guimaraes, Ana Marcia; Turk, Dusan; Wrenger, Carsten; Meents, Alke
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收藏CogiTx1: A novel subtilisin A inhibitor isolated from the sea anemone Condylactis gigantea belonging to the defensin 4 protein family
Rojas, Laritza; Cabrera-Munoz, Aymara; Espinosa, Luis A.; Montane, Sergi; Alvarez-Lajonchere, Luis; Mojarena, Jesus D.; Moya, Galina; Lorenzo, Julia; Gonzalez, Luis J.; Betzel, Christian; Antigua, Maday Alonso-del-Rivero
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收藏Initiation and modulation of Tau protein phase separation by the drug suramin
Prince, Prabhu Rajaiah; Hochmair, Janine; Brognaro, Hevila; Gevorgyan, Susanna; Franck, Maximilian; Schubert, Robin; Lorenzen, Kristina; Yazici, Selin; Mandelkow, Eckhard; Wegmann, Susanne; Betzel, Christian
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收藏Intrinsically disordered plant protein PARCL colocalizes with RNA in phase-separated condensates whose formation can be regulated by mutating the PLD
Ostendorp, Anna; Ostendorp, Steffen; Zhou, Yuan; Chaudron, Zoe; Wolffram, Lukas; Rombi, Khadija; von Pein, Linn; Falke, Sven; Jeffries, Cy M.; Svergun, Dmitri I.; Betzel, Christian; Morris, Richard J.; Kragler, Friedrich; Kehr, Julia
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收藏Comparative Study to Characterise the Pharmaceutical Potential of Synthesised Snake Venom Bradykinin-Potentiating Peptides In Vivo
Munawar, Aisha; Zaman, Fakhar; Ishaq, Muhammad Waqas; Hassan, Khwaja Ali; Masood, Saima; Ali, Zahid; Majeed, Khalid Abdul; Akrem, Ahmed; Ali, Syed Abid; Betzel, Christian
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收藏Comprehensive Structural and Functional Characterization of a Seed γ-thionin as a Potent Bioactive Molecule Against Fungal Pathogens and Insect Pests
Khaliq, Binish; Abdalla, Mohnad; Mehmood, Sohaib; Saeed, Ahsan; Munawar, Aisha; Saeed, Muhammad Qamar; Saeed, Qamar; Ibrahim, Muhammad; Ali, Zahid; Hussain, Saber; Eltayb, Wafa Ali; Betzel, Christian; Akrem, Ahmed
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收藏Antiviral activity of natural phenolic compounds in complex at an allosteric site of SARS-CoV-2 papain-like protease
Srinivasan, Vasundara; Brognaro, Hevila; Prabhu, Prince R.; de Souza, Edmarcia Elisa; Guenther, Sebastian; Reinke, Patrick Y. A.; Lane, Thomas J.; Ginn, Helen; Han, Huijong; Ewert, Wiebke; Sprenger, Janina; Koua, Faisal H. M.; Falke, Sven; Werner, Nadine; Andaleeb, Hina; Ullah, Najeeb; Franca, Bruno Alves; Wang, Mengying; Barra, Angelica Luana C.; Perbandt, Markus; Schwinzer, Martin; Schmidt, Christina; Brings, Lea; Lorenzen, Kristina; Schubert, Robin; Guaragna Machado, Rafael Rahal; Candido, Erika Donizette; Leal Oliveira, Danielle Bruna; Durigon, Edison Luiz; Niebling, Stephan; Garcia, Angelica Struve; Yefanov, Oleksandr; Lieske, Julia; Gelisio, Luca; Domaracky, Martin; Middendorf, Philipp; Groessler, Michael; Trost, Fabian; Galchenkova, Marina; Mashhour, Aida Rahmani; Saouane, Sofiane; Hakanpaeae, Johanna; Wolf, Markus; Alai, Maria Garcia; Turk, Dusan; Pearson, Arwen R.; Chapman, Henry N.; Hinrichs, Winfried; Wrenger, Carsten; Meents, Alke; Betzel, Christian
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收藏Hydrazones and Thiosemicarbazones Targeting Protein-Protein-Interactions of SARS-CoV-2 Papain-like Protease
Ewert, Wiebke; Guenther, Sebastian; Miglioli, Francesca; Falke, Sven; Reinke, Patrick Y. A.; Niebling, Stephan; Guenther, Christian; Han, Huijong; Srinivasan, Vasundara; Brognaro, Hevila; Lieske, Julia; Lorenzen, Kristina; Garcia-Alai, Maria M.; Betzel, Christian; Carcelli, Mauro; Hinrichs, Winfried; Rogolino, Dominga; Meents, Alke
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收藏Molecular crowding and RNA synergize to promote phase separation, microtubule interaction, and seeding of Tau condensates
Hochmair, Janine; Exner, Christian; Franck, Maximilian; Dominguez-Baquero, Alvaro; Diez, Lisa; Brognaro, Hevila; Kraushar, Matthew L.; Mielke, Thorsten; Radbruch, Helena; Kaniyappan, Senthil; Falke, Sven; Mandelkow, Eckhard; Betzel, Christian; Wegmann, Susanne
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收藏Eruca sativa seed napin structural insights and thorough functional characterization
Khaliq, Binish; Falke, Sven; Saeed, Qamar; Bilal, Muhammad; Munawar, Aisha; Ali, Arslan; Baermann, Gunnar; Athar, Habib-ur-Rehman; Mahmood, Seema; Betzel, Christian; Ali, Qurban; Akrem, Ahmed
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