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Application of Lipophilic Prodrug Charge Masking Strategy to Obtain Novel, Potential Oxytocin Prodrugs 应用脂溶性前药电荷掩蔽策略以获得新型、潜在催产素前药 Gitlin-Domagalska, Agata; Olejnik, Anna; Ruczynski, Jaroslaw; Starego, Dominika; Ptaszynska, Natalia; Legowska, Anna; Debowski, Dawid; Gilon, Chaim; Rolka, Krzysztof 分享 收藏
Anti-Inflammatory Effects of Clarstatin, a Shared-Epitope-Antagonistic Cyclic Peptide, on Experimental Autoimmune Uveitis in Mice Merzbach, Shira; Schumacher-Klinger, Adi; Klazas, Michal; Hoffman, Amnon; Lazarovici, Philip; Gilon, Chaim; Nussbaum, Gabriel; Amer, Radgonde 分享 收藏
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Structure-Activity Relationship of Synthetic Linear KTS-Peptides Containing Meta-Aminobenzoic Acid as Antagonists of α1β1 Integrin with Anti-Angiogenic and Melanoma Anti-Tumor Activities Naamneh, Majdi Saleem; Momic, Tatjana; Klazas, Michal; Grosche, Julius; Eble, Johannes A.; Marcinkiewicz, Cezary; Khazanov, Netaly; Senderowitz, Hanoch; Hoffman, Amnon; Gilon, Chaim; Katzhendler, Jehoshua; Lazarovici, Philip 分享 收藏
Synthesis of Novel Arginine Building Blocks with Increased Lipophilicity Compatible with Solid-Phase Peptide Synthesis Glavas, Mladena; Gitlin-Domagalska, Agata; Ptaszynska, Natalia; Starego, Dominika; Freza, Sylwia; Debowski, Dawid; Helbik-Maciejewska, Aleksandra; Legowska, Anna; Gilon, Chaim; Rolka, Krzysztof 分享 收藏
PH-Binding Motif in PAR4 Oncogene: From Molecular Mechanism to Drug Design Nag, Jeetendra Kumar; Malka, Hodaya; Sedley, Shoshana; Appasamy, Priyanga; Rudina, Tatyana; Levi, Tgst; Hoffman, Amnon; Gilon, Chaim; Uziely, Beatrice; Bar-Shavit, Rachel 分享 收藏
Synthesis and Pharmacological Characterization of Visabron, a Backbone Cyclic Peptide Dual Antagonist of α4β1 (VLA-4)/α9β1 Integrin for Therapy of Multiple Sclerosis 用于治疗多发性硬化的 α4β1 (VLA-4)/α9β1整合素骨架环肽双拮抗剂Visabron的合成和药理表征 Gilon, Chaim; Klazas, Michal; Lahiani, Adi; Schumacher-Klinger, Adi; Merzbach, Shira; Naoum, Johnny N.; Ovadia, Haim; Rubin, Limor; Cornell-Kennon, Susan; Schaefer, Erik M.; Katzhendler, Jehoshua; Marcinkiewicz, Cezary; Hoffman, Amnon; Lazarovici, Philip 分享 收藏
Cyclizing Painkillers: Development of Backbone-Cyclic TAPS Analogs Talhami, Alaa; Swed, Avi; Hess, Shmuel; Ovadia, Oded; Greenberg, Sarit; Schumacher-Klinger, Adi; Rosenthal, David; Shalev, Deborah E.; Hurevich, Mattan; Lazarovici, Philip; Hoffman, Amnon; Gilon, Chaim 分享 收藏
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Overcoming the Lack of Oral Availability of Cyclic Hexapeptides: Design of a Selective and Orally Available Ligand for the Integrin αvβ3 Weinmueller, Michael; Rechenmacher, Florian; Marelli, Udaya Kiran; Reichart, Florian; Kapp, Tobias G.; Raeder, Andreas F. B.; Di Leva, Francesco Saverio; Marinelli, Luciana; Novellino, Ettore; Munoz-Felix, Jose M.; Hodivala-Dilke, Kairbaan; Schumacher, Adi; Fanous, Joseph; Gilon, Chaim; Hoffman, Amnon; Kessler, Horst 分享 收藏
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Inhibition of inositol monophosphatase (IMPase) at the calbindin-D28k binding site: Molecular and behavioural aspects (vol 23, pg 1806, 2013) Levi, Itzhak; Eskira, Yael; Eisenstein, Miriam; Gilon, Chaim; Hoffman, Amnon; Tal-Gan, Yftah; Fanous, Joseph; Bersudsky, Yuly; Belmaker, R. H.; Agam, Galila; Almog, Orna 分享 收藏
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