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Chaim Gilon

The Hebrew University of Jerusalem

48H指数
316论文数
1.0W被引数
收录论文 68
发表时间
Application of Lipophilic Prodrug Charge Masking Strategy to Obtain Novel, Potential Oxytocin Prodrugs应用脂溶性前药电荷掩蔽策略以获得新型、潜在催产素前药
err2025-05-16
err0
errOAAI
errGitlin-Domagalska, Agata; Olejnik, Anna; Ruczynski, Jaroslaw; Starego, Dominika; Ptaszynska, Natalia; Legowska, Anna; Debowski, Dawid; Gilon, Chaim; Rolka, Krzysztof
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Anti-Inflammatory Effects of Clarstatin, a Shared-Epitope-Antagonistic Cyclic Peptide, on Experimental Autoimmune Uveitis in Mice
err2025-01-07
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errMerzbach, Shira; Schumacher-Klinger, Adi; Klazas, Michal; Hoffman, Amnon; Lazarovici, Philip; Gilon, Chaim; Nussbaum, Gabriel; Amer, Radgonde
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Development of Clarstatin, a Novel Drug Lead for the Therapy of Autoimmune Uveitis
err2024-05-27
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errOAAI
errMerzbach, Shira; Hoffman, Amnon; Lazarovici, Philip; Gilon, Chaim; Amer, Radgonde
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Structure-Activity Relationship of Synthetic Linear KTS-Peptides Containing Meta-Aminobenzoic Acid as Antagonists of α1β1 Integrin with Anti-Angiogenic and Melanoma Anti-Tumor Activities
err2024-04-24
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errNaamneh, Majdi Saleem; Momic, Tatjana; Klazas, Michal; Grosche, Julius; Eble, Johannes A.; Marcinkiewicz, Cezary; Khazanov, Netaly; Senderowitz, Hanoch; Hoffman, Amnon; Gilon, Chaim; Katzhendler, Jehoshua; Lazarovici, Philip
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Synthesis of Novel Arginine Building Blocks with Increased Lipophilicity Compatible with Solid-Phase Peptide Synthesis
err2023-11-25
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errGlavas, Mladena; Gitlin-Domagalska, Agata; Ptaszynska, Natalia; Starego, Dominika; Freza, Sylwia; Debowski, Dawid; Helbik-Maciejewska, Aleksandra; Legowska, Anna; Gilon, Chaim; Rolka, Krzysztof
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PH-Binding Motif in PAR4 Oncogene: From Molecular Mechanism to Drug Design
err2022-09-02
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errNag, Jeetendra Kumar; Malka, Hodaya; Sedley, Shoshana; Appasamy, Priyanga; Rudina, Tatyana; Levi, Tgst; Hoffman, Amnon; Gilon, Chaim; Uziely, Beatrice; Bar-Shavit, Rachel
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Synthesis and Pharmacological Characterization of Visabron, a Backbone Cyclic Peptide Dual Antagonist of α4β1 (VLA-4)/α9β1 Integrin for Therapy of Multiple Sclerosis用于治疗多发性硬化的 α4β1 (VLA-4)/α9β1整合素骨架环肽双拮抗剂Visabron的合成和药理表征
errJACS AU
IF8.7
err2021-11-24
err3
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errGilon, Chaim; Klazas, Michal; Lahiani, Adi; Schumacher-Klinger, Adi; Merzbach, Shira; Naoum, Johnny N.; Ovadia, Haim; Rubin, Limor; Cornell-Kennon, Susan; Schaefer, Erik M.; Katzhendler, Jehoshua; Marcinkiewicz, Cezary; Hoffman, Amnon; Lazarovici, Philip
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Cyclizing Painkillers: Development of Backbone-Cyclic TAPS Analogs
err2020-11-12
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errTalhami, Alaa; Swed, Avi; Hess, Shmuel; Ovadia, Oded; Greenberg, Sarit; Schumacher-Klinger, Adi; Rosenthal, David; Shalev, Deborah E.; Hurevich, Mattan; Lazarovici, Philip; Hoffman, Amnon; Gilon, Chaim
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Diffusion-Enhanced Amide Bond Formation on a Solid Support固体支持物上扩散增强的酰胺键形成
err2019-11-08
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errNaoum, Johnny N.; Alshanski, Israel; Gitlin-Domagalska, Agata; Bentolila, Moshe; Gilon, Chaim; Hurevich, Mattan
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Deciphering Direct and Indirect Effects of Neurokinin B and GnRH in the Brain-Pituitary Axis of Tilapia
err2019-07-12
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errMizrahi, Naama; Gilon, Chaim; Atre, Ishwar; Ogawa, Satoshi; Parhar, Ishwar S.; Levavi-Sivan, Berta
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Enhancing the Efficiency of the Solid Phase Peptide Synthesis (SPPS) Process by High Shear Mixing
err2018-09-04
err15
PREAI
errAlshanski, Israel; Bentolila, Moshe; Gitlin-Domagalska, Agata; Zamir, Dolev; Zorsky, Shir; Joubran, Salim; Hurevich, Mattan; Gilon, Chaim
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Development of a Novel Backbone Cyclic Peptide Inhibitor of the Innate Immune TLR/IL1R Signaling Protein MyD88
err2018-06-21
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errDishon, Shira; Schumacher, Adi; Fanous, Joseph; Talhami, Alaa; Kassis, Ibrahim; Karussis, Dimitrios; Gilon, Chaim; Hoffmann, Amnon; Nussbaum, Gabriel
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Oxytocin-Monolayer-Based Impedimetric Biosensor for Zinc and Copper Ions
err2017-12-08
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errTadi, Kiran Kumar; Alshanski, Israel; Mervinetsky, Evgeniy; Marx, Gerard; Petrou, Panayiota; Dimitrios, Karussis M.; Gilon, Chaim; Hurevich, Mattan; Yitzchaik, Shlomo
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Overcoming the Lack of Oral Availability of Cyclic Hexapeptides: Design of a Selective and Orally Available Ligand for the Integrin αvβ3
err2017-11-23
err29
PREAI
errWeinmueller, Michael; Rechenmacher, Florian; Marelli, Udaya Kiran; Reichart, Florian; Kapp, Tobias G.; Raeder, Andreas F. B.; Di Leva, Francesco Saverio; Marinelli, Luciana; Novellino, Ettore; Munoz-Felix, Jose M.; Hodivala-Dilke, Kairbaan; Schumacher, Adi; Fanous, Joseph; Gilon, Chaim; Hoffman, Amnon; Kessler, Horst
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Superiority of the S,S conformation in diverse pharmacological processes: Intestinal transport and entry inhibition activity of novel anti-HIV drug lead
err2015-11-01
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PREAI
errFanous, Joseph; Swed, Avi; Joubran, Salim; Hurevich, Mattan; Britan-Rosich, Elena; Kotler, Moshe; Gilon, Chaim; Hoffman, Amnon
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Inhibition of inositol monophosphatase (IMPase) at the calbindin-D28k binding site: Molecular and behavioural aspects (vol 23, pg 1806, 2013)
err2015-11-01
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errLevi, Itzhak; Eskira, Yael; Eisenstein, Miriam; Gilon, Chaim; Hoffman, Amnon; Tal-Gan, Yftah; Fanous, Joseph; Bersudsky, Yuly; Belmaker, R. H.; Agam, Galila; Almog, Orna
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Mechanistic Studies of Malonic Acid-Mediated In Situ Acylation
err2015-09-24
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PREAI
errChandra, Koushik; Naoum, Johnny N.; Roy, Tapta Kanchan; Gilon, Chaim; Gerber, R. Benny; Friedler, Assaf
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cis-Peptide Bonds: A Key for Intestinal Permeability of Peptides?
err2015-09-04
err33
PREAI
errMarelli, Udaya Kiran; Ovadia, Oded; Frank, Andreas Oliver; Chatterjee, Jayanta; Gilon, Chaim; Hoffman, Amnon; Kessler, Horst
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Shared Epitope-Antagonistic Ligands: A New Therapeutic Strategy in Mice With Erosive Arthritis
err2015-07-28
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errLing, Song; Liu, Ying; Fu, Jiaqi; Colletta, Alessandro; Gilon, Chaim; Holoshitz, Joseph
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