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Virtual Screening of a Chemically Diverse Superscaffold Library Enables Ligand Discovery for a Key GPCR Target 化学上多样化的超级支架文库的虚拟筛选可以发现关键GPCR靶标的配体 Grotsch, Katharina; Sadybekov, Anastasiia V.; Hiller, Sydney; Zaidi, Saheem; Eremin, Dmitry; Le, Austen; Liu, Yongfeng; Smith, Evan Carlton; Illiopoulis-Tsoutsouvas, Christos; Thomas, Joice; Aggarwal, Shubhangi; Pickett, Julie E.; Reyes, Cesar; Picazo, Elias; Roth, Bryan L.; Makriyannis, Alexandros; Katritch, Vsevolod; Fokin, Valery V. 分享 收藏
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Gold(I) Phosphine Derivatives with Improved Selectivity as Topically Active Drug Leads to Overcome 5-Nitroheterocyclic Drug Resistance in Trichomonas vaginalis Miyamoto, Yukiko; Aggarwal, Shubhangi; Celaje, Jeff Joseph A.; Ihara, Sozaburo; Ang, Jonathan; Eremin, Dmitry B.; Land, Kirkwood M.; Wrischnik, Lisa A.; Zhang, Liangfang; Fokin, Valery V.; Eckmann, Lars 分享 收藏
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Click chemistry-facilitated comprehensive identification of proteins adducted by antimicrobial 5-nitroimidazoles for discovery of alternative drug targets against giardiasis Lauwaet, Tineke; Miyamoto, Yukiko; Ihara, Sozaburo; Le, Christine; Kalisiak, Jaroslaw; Korthals, Keith A.; Ghassemian, Majid; Smith, Diane K.; Sharpless, K. Barry; Fokin, Valery V.; Eckmann, Lars 分享 收藏
Counteracting tabun inhibition by reactivation by pyridinium aldoximes that interact with active center gorge mutants of acetylcholinesterase 通过与乙酰胆碱酯酶的活性中心峡谷突变体相互作用的吡啶鎓醛肟的再活化来抵消塔本抑制 Kovarik, Zrinka; Hrvat, Nikolina Macek; Kalisiak, Jaroslaw; Katalinic, Maja; Sit, Rakesh K.; Zorbaz, Tamara; Radic, Zoran; Fokin, Valery V.; Sharpless, K. Barry; Taylor, Palmer 分享 收藏
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Pharmacology, Pharmacokinetics, and Tissue Disposition of Zwitterionic Hydroxyiminoacetamido Alkylamines as Reactivating Antidotes for Organophosphate Exposure Sit, Rakesh K.; Kovarik, Zrinka; Hrvat, Nikolina Macek; Zunec, Suzana; Green, Carol; Fokin, Valery V.; Sharpless, K. Barry; Radic, Zoran; Taylor, Palmer 分享 收藏
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Click Chemistry-Facilitated Structural Diversification of Nitrothiazoles, Nitrofurans, and Nitropyrroles Enhances Antimicrobial Activity against Giardia lamblia Kim, Wan Jung; Korthals, Keith A.; Li, Suhua; Le, Christine; Kalisiak, Jaroslaw; Sharpless, K. Barry; Fokin, Valery V.; Miyamoto, Yukiko; Eckmann, Lars 分享 收藏
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